中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [4]
采集方式
OAI收割 [4]
内容类型
期刊论文 [4]
发表日期
2021 [1]
2014 [1]
2013 [2]
学科主题
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Third-generation EGFR inhibitor HS-10296 in combination with famitinib, a multi-targeted tyrosine kinase inhibitor, exerts synergistic antitumor effects through enhanced inhibition of downstream signaling in EGFR-mutant non-small cell lung cancer cells
期刊论文
OAI收割
THORACIC CANCER, 2021, 页码: 9
作者:
Zhang, Mi
;
Quan, Haitian
;
Fu, Li
;
Li, Yun
;
Fu, Haoyu
  |  
收藏
  |  
浏览/下载:66/0
  |  
提交时间:2021/05/24
EGFR‐
mutant non‐
small cell lung cancer
famitinib
HS‐
10296
multi‐
targeted tyrosine kinase inhibitor
third‐
generation EGFR inhibitor
Predicting pharmacokinetics of anti-cancer drug, famitinib in human using physiologically based pharmacokinetic model
期刊论文
OAI收割
Acta Pharmaceutica Sinica, 2014, 卷号: 49, 期号: 12, 页码: 1684-1688
作者:
Yu Mingming
;
Gao Zhiwei
;
Chen Xiaoyan
;
Zhong Dafang
  |  
收藏
  |  
浏览/下载:43/0
  |  
提交时间:2019/01/08
famitinib
physiologically based pharmacokinetic model
species extrapolation
tyrosine kinase inhibitor
Phase I study of the safety, pharmacokinetics and antitumor activity of famitinib
期刊论文
OAI收割
CANCER CHEMOTHERAPY AND PHARMACOLOGY, 2013, 卷号: 72, 期号: 5, 页码: 1043-1053
作者:
Zhou, Aiping
;
Zhang, Wen
;
Chang, Chunxiao
;
Chen, Xiaoyan
;
Zhong, Dafang
  |  
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2019/01/08
Famitinib
Phase I trial
Safety
Pharmacokinetics
Antitumor activity
Metabolism and bioactivation of famitinib, a novel inhibitor of receptor tyrosine kinase, in cancer patients
期刊论文
OAI收割
BRITISH JOURNAL OF PHARMACOLOGY, 2013, 卷号: 168, 期号: 7, 页码: 1687-1706
作者:
Xie, Cen
;
Zhou, Jialan
;
Guo, Zitao
;
Diao, Xingxing
;
Gao, Zhiwei
  |  
收藏
  |  
浏览/下载:62/0
  |  
提交时间:2019/01/08
famitinib
metabolism
bioactivation
quinone-imine
hepatotoxicity