中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [6]
南海海洋研究所 [1]
大连化学物理研究所 [1]
采集方式
OAI收割 [8]
内容类型
期刊论文 [7]
会议论文 [1]
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2022 [1]
2020 [1]
2018 [1]
2015 [2]
2014 [1]
2012 [1]
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学科主题
物理化学 [1]
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In vitro and in vivo evaluation of the main protease inhibitor FB2001 against SARS-CoV-2
期刊论文
OAI收割
ANTIVIRAL RESEARCH, 2022, 卷号: 208, 页码: 10
作者:
Shang, Weijuan
;
Dai, Wenhao
;
Yao, Cheng
;
Xu, Ling
;
Tao, Xiangming
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2023/04/10
SARS-CoV-2
SARS-CoV-2 variants
FB2001
Main protease
PBPK
Anti-SARS-CoV-2 in vivo
Physiologically Based Pharmacokinetic Model for the Biotransportation of Arsenic in Marine Medaka (Oryzias melastigma)
期刊论文
OAI收割
ENVIRONMENTAL SCIENCE & TECHNOLOGY, 2020, 卷号: 54, 期号: 12, 页码: 7485, 7493
作者:
Zhang, Wei
;
Song, Dongdong
;
Tan, Qiao-Guo
;
Wang, Wen-Xiong
;
Zhang, Li
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2020/09/22
Glycyrrhizin has a high likelihood to be a victim of drug-drug interactions mediated by hepatic organic anion-transporting polypeptide 1B1/1B3
期刊论文
OAI收割
BRITISH JOURNAL OF PHARMACOLOGY, 2018, 卷号: 175, 期号: 17, 页码: 3486-3503
作者:
Dong, Jiajia
;
Olaleye, Olajide E.
;
Jiang, Rongrong
;
Li, Jing
;
Lu, Chuang
  |  
收藏
  |  
浏览/下载:96/0
  |  
提交时间:2019/01/08
Preclinical pharmacokinetics of TPN729MA, a novel PDE5 inhibitor, and prediction of its human pharmacokinetics using a PBPK model
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2015, 卷号: 36, 期号: 12, 页码: 1528-1536
作者:
Gao, Zhi-wei
;
Zhu, Yun-ting
;
Yu, Ming-ming
;
Zan, Bin
;
Liu, Jia
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2019/01/08
TPN729MA
PDE5 inhibitor
erectile dysfunction
pharmacokinetics
human PK prediction
physiologically based pharmacokinetic model
preclinicalpharmacokineticsoftpn729maanovelpde5inhibitorandpredictionofitshumanpharmacokineticsusingapbpkmodel
期刊论文
OAI收割
actapharmacologicasinica, 2015, 卷号: 36, 期号: 12, 页码: 1528
作者:
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2020/07/01
HUMAN DRUG CLEARANCE
PHOSPHODIESTERASE-5 INHIBITORS
CLINICAL PHARMACOKINETICS
ERECTILE DYSFUNCTION
TISSUE DISTRIBUTION
ORAL PHARMACOKINETICS
RECEPTOR ANTAGONIST
DIVERSE COMPOUNDS
IN-VIVO
ABSORPTION
TPN729MA
PDE5 inhibitor
erectile dysfunction
pharmacokinetics
human PK prediction
physiologically based pharmacokinetic model
Predicting pharmacokinetics of anti-cancer drug, famitinib in human using physiologically based pharmacokinetic model
期刊论文
OAI收割
Acta Pharmaceutica Sinica, 2014, 卷号: 49, 期号: 12, 页码: 1684-1688
作者:
Yu Mingming
;
Gao Zhiwei
;
Chen Xiaoyan
;
Zhong Dafang
  |  
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2019/01/08
famitinib
physiologically based pharmacokinetic model
species extrapolation
tyrosine kinase inhibitor
Simulation of the pharmacokinetics of bisoprolol in healthy adults and patients with impaired renal function using whole-body physiologically based pharmacokinetic modeling
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2012, 卷号: 33, 期号: 11, 页码: 1359
作者:
Li Guofu
;
Wang Kun
;
Chen Rui
;
Zhao Haoru
;
Yang Jin
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2020/12/24
TISSUE DISTRIBUTION
DRUG DISCOVERY
INTRASUBJECT VARIABILITY
PBPK SIMULATION
P-GP
ABSORPTION
POPULATION
PREDICTION
BIOAVAILABILITY
IDENTIFICATION
bisoprolol
whole-body physiologically based pharmacokinetic model
drug absorption
drug distribution
renal function impairment
Hepatobiliary disposition of deoxyschizandrin in perfused rat livers in situ
会议论文
OAI收割
16th north american regional issx meeting, 美国, 2009-10-18
吴敬敬
;
张延延
;
葛广波
;
杨凌
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2011/07/11