中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [6]
成都生物研究所 [1]
中国科学院大学 [1]
采集方式
OAI收割 [7]
iSwitch采集 [1]
内容类型
期刊论文 [8]
发表日期
2021 [1]
2019 [1]
2015 [2]
2011 [2]
2010 [2]
学科主题
Chemistry [1]
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Synthesis and Evaluation of 3-(Indol-3-yl)-4-(Pyrazolo[3,4-c]Pyridazin-3-yl)-Maleimides as Potent Mutant Isocitrate Dehydrogenase-1 Inhibitors
期刊论文
OAI收割
PHARMACEUTICAL CHEMISTRY JOURNAL, 2021, 卷号: 55, 期号: 7, 页码: 655-664
作者:
Xu, Jianghong
;
Hu, Yuanyuan
;
Liu, Xiaoqi
;
Gao, Anhui
;
Gao, Lixin
  |  
收藏
  |  
浏览/下载:55/0
  |  
提交时间:2021/12/01
IDH1-R132H inhibitors
synthesis
biological activity
docking
3-(indol-3-yl)-4-(pyrazolo-[3
4-c]pyridazin-3-yl)-maleimides
Synthesis and biological evaluation of 3-aryl-4-indolyl-maleimides as potent mutant isocitrate dehydrogenase-1 inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2019, 卷号: 27, 期号: 4, 页码: 589-603
作者:
Liu, Xiaoqi
;
Hu, Yuanyuan
;
Gao, Anhui
;
Xu, Meng
;
Gao, Lixin
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2020/07/01
3-Aryl-4-indolyl-maleimides
IDH1/R132H inhibitors
Tumor 2-HG
Synthesis
Synthesis and Evaluation of 3-(furo[2,3-b]pyridin-3-yl)-4-(1H-indol-3-yl)-maleimides as Novel GSK-3 Inhibitors and Anti-Ischemic Agents
期刊论文
OAI收割
CHEMICAL BIOLOGY & DRUG DESIGN, 2015, 卷号: 86, 期号: 4, 页码: 746-752
作者:
Ye, Qing
;
Li, Qiu
;
Zhou, Yubo
;
Xu, Lei
;
Mao, Weili
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2019/01/08
anti-ischemic agents
GSK-3 inhibitors
kinase activity
maleimides
Synthesis and biological evaluation of 3-([1,2,4]triazolo [4,3-a]pyridin-3-yl)-4-(indol-3-yl)-maleimides as potent, selective GSK-3 beta inhibitors and neuroprotective agents
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2015, 卷号: 23, 期号: 5, 页码: 1179-1188
作者:
Ye, Qing
;
Mao, Weili
;
Zhou, Yubo
;
Xu, Lei
;
Li, Qiu
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2019/01/08
GSK-3 beta inhibitors
Maleimides
Kinase activity
Neuroprotective agents
Chiral Pyrrolidine Sulfonamide Catalyzed Enantioselective Michael Addition of Cyclohexanones to Maleimides
期刊论文
OAI收割
SYNLETT, 2011, 期号: 4, 页码: 473-476
作者:
Wang, Jian
;
Zhang, Man-Man
;
Zhang, Shieli
;
Xu, Zi-An
;
Li, Hao
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/01/08
cyclic ketones
maleimides
Michael reaction
pyrrolidine sulfonamide
Thiourea-Catalyzed Highly Diastereo- and Enantioselective Conjugate Additions of alpha-Substituted Cyanoacetates to Maleimides: Efficient Construction of Vicinal Quaternary-Tertiary Stereocenters
期刊论文
OAI收割
ADVANCED SYNTHESIS & CATALYSIS, 2011, 卷号: 353, 期号: 10, 页码: 1720-1728
Liao, Yu-Hua
;
Liu, Xiong-Li
;
Wu, Zhi-Jun
;
Du, Xi-Lin
;
Zhang, Xiao-Mei
;
Yuan, Wei-Cheng
收藏
  |  
浏览/下载:1003/0
  |  
提交时间:2012/11/09
bifunctional thioureas
maleimides
Michael addition
organocatalysis
alpha-substituted cyanoacetates
Chiral primary amine thiourea promoted highly enantioselective michael reactions of isobutylaldehyde with maleimides
期刊论文
iSwitch采集
Tetrahedron, 2010, 卷号: 66, 期号: 46, 页码: 8928-8932
作者:
Bai, Jian-Fei
;
Peng, Lin
;
Wang, Liang-liang
;
Wang, Li-Xin
;
Xu, Xiao-Ying
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2019/05/10
Primary amine thiourea
Michael reactions
Isobutylaldehyde
Maleimides
Enantioselective
A Simple Primary Amine Thiourea Catalyzed Highly Enantioselective Conjugate Addition of alpha,alpha-Disubstituted Aldehydes to Maleimides
期刊论文
OAI收割
CHEMISTRY-A EUROPEAN JOURNAL, 2010, 卷号: 16, 期号: 27, 页码: 7979-7982
作者:
Xue, Fei
;
Liu, Lu
;
Zhang, Shilei
;
Duan, Wenhu
;
Wang, Wei
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2019/01/08
aldehydes
maleimides
Michael addition
organocatalysis