中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
首页
机构
成果
学者
登录
注册
登陆
×
验证码:
换一张
忘记密码?
记住我
×
校外用户登录
CAS IR Grid
机构
上海药物研究所 [9]
采集方式
OAI收割 [9]
内容类型
期刊论文 [9]
发表日期
2021 [9]
学科主题
筛选
浏览/检索结果:
共9条,第1-9条
帮助
限定条件
发表日期:2021
专题:上海药物研究所
第一署名单位
第一作者单位
通讯作者单位
条数/页:
5
10
15
20
25
30
35
40
45
50
55
60
65
70
75
80
85
90
95
100
排序方式:
请选择
提交时间升序
提交时间降序
题名升序
题名降序
作者升序
作者降序
发表日期升序
发表日期降序
GLP-1 mimetics as a potential therapy for nonalcoholic steatohepatitis
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 11
作者:
Chen, Yan
;
Xu, Ying-na
;
Ye, Chen-yu
;
Feng, Wen-bo
;
Zhou, Qing-tong
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2022/06/15
NAFLD
NASH
GLP-1R
GLP-1 mimetics
dual agonists
triple agonists
GPCR
Theoretical study and application of 2-phenyl-1,3,4-thiadiazole derivatives with optical and inhibitory activity against SHP1
期刊论文
OAI收割
PHYSICAL CHEMISTRY CHEMICAL PHYSICS, 2021, 页码: 14
作者:
Zhang, Chun
;
Sun, Yi-Tao
;
Gao, Li-Xin
;
Feng, Bo
;
Yan, Xue
  |  
收藏
  |  
浏览/下载:48/0
  |  
提交时间:2022/01/18
Synthesis and biological evaluation of 2,5-diaryl-1,3,4-oxadiazole derivatives as novel Src homology 2 domain-containing protein tyrosine phosphatase 2 (SHP2) inhibitors
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2021, 卷号: 116, 页码: 13
作者:
Meng, Xiang-Dong
;
Gao, Li-Xin
;
Wang, Zhi-Jia
;
Feng, Bo
;
Zhang, Chun
  |  
收藏
  |  
浏览/下载:61/0
  |  
提交时间:2021/12/01
2,5-diphenyl-1,3,4-oxadiazole derivatives
SHP2
Inhibitors
Structure-activity relationships (SAR)
Kynurenine derivative 3-HAA is an agonist ligand for transcription factor YY1
期刊论文
OAI收割
Journal of Hematology & Oncology, 2021, 卷号: 14, 期号: 1
作者:
Shi,Zhaopeng
;
Gan,Guifang
;
Xu,Xiang
;
Zhang,Jieying
;
Yuan,Yuan
  |  
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2021/11/04
3-Hydroxyanthronic acid (3-HAA)
Kynurenine
YY1
DUSP6
Hepatocellular carcinoma (HCC)
Tryptophan metabolism
DOT1L Regulates Thermogenic Adipocyte Differentiation and Function via Modulating H3K79 Methylation
期刊论文
OAI收割
DIABETES, 2021, 卷号: 70, 期号: 6, 页码: 1317-1333
作者:
Shuai, Lin
;
Li, Bo-Han
;
Jiang, Hao-Wen
;
Yang, Lin
;
Li, Jia
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2021/08/17
Natural product 1,2,3,4,6-penta-O-galloyl-beta-D-glucopyranose is a reversible inhibitor of glyceraldehyde 3-phosphate dehydrogenase
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 13
作者:
Li, Wen
;
Liao, Li-ping
;
Song, Ning
;
Liu, Yan-jun
;
Ding, Yi-luan
  |  
收藏
  |  
浏览/下载:44/0
  |  
提交时间:2021/06/11
glyceraldehyde 3-phosphate dehydrogenase
1,2,3,4,6-penta-O-galloyl-beta-D-glucopyranose
hydrogen deuterium exchange mass spectrometry
reversible inhibitor
glycolysis
Natural product 1,2,3,4,6-penta-O-galloyl-beta-D-glucopyranose is a reversible inhibitor of glyceraldehyde 3-phosphate dehydrogenase
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 13
作者:
Li, Wen
;
Liao, Li-ping
;
Song, Ning
;
Liu, Yan-jun
;
Ding, Yi-luan
  |  
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2021/06/11
glyceraldehyde 3-phosphate dehydrogenase
1,2,3,4,6-penta-O-galloyl-beta-D-glucopyranose
hydrogen deuterium exchange mass spectrometry
reversible inhibitor
glycolysis
Downregulation of c-Myc expression confers sensitivity to CHK1 inhibitors in hematologic malignancies
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 9
作者:
Jiang, Kai-long
;
Tong, Le-xian
;
Wang, Tao
;
Wang, Han-lin
;
Hu, Xiao-bei
  |  
收藏
  |  
浏览/下载:49/0
  |  
提交时间:2021/05/24
CHK1 inhibitors
PY34
drug sensitivity
c-Myc
hematologic malignancies
Synthesis of 2-ethoxycarbonylthieno[2,3-b]quinolines in biomass-derived solvent gamma-valerolactone and their biological evaluation against protein tyrosine phosphatase 1B
期刊论文
OAI收割
RSC ADVANCES, 2021, 卷号: 11, 期号: 6, 页码: 3216-3220
作者:
Mu, Xu-Yang
;
Wang, Zhi-Jia
;
Feng, Bo
;
Xu, Lei
;
Gao, Li-Xin
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2021/05/24