中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [17]
采集方式
OAI收割 [17]
内容类型
期刊论文 [17]
发表日期
2021 [17]
学科主题
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浏览/检索结果:
共17条,第1-10条
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发表日期:2021
专题:上海药物研究所
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Sublyratins A-O, Labdane-Type Diterpenoids from Croton sublyratus
期刊论文
OAI收割
JOURNAL OF NATURAL PRODUCTS, 2021, 卷号: 84, 期号: 11, 页码: 2971-2980
作者:
Qi, Jing-Jing
;
Zhou, Jun-Su
;
Zhang, Yan
;
Fan, Yao-Yue
;
Zhou, Bin
  |  
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2022/01/18
Quantitative proteomic analysis uncovers inhibition of melanin synthesis by silk fibroin via MITF/tyrosinase axis in B16 melanoma cells
期刊论文
OAI收割
LIFE SCIENCES, 2021, 卷号: 284, 页码: 7
作者:
Wang, Yuqiu
;
Duan, Tianbi
  |  
收藏
  |  
浏览/下载:59/0
  |  
提交时间:2021/11/04
Silk fibroin
Quantitative proteomics
Melanin
Microphthalmia-associated transcription factor
Tyrosinase
Progression and Regression of Abdominal Aortic Aneurysms in Mice
期刊论文
OAI收割
CURRENT MEDICAL SCIENCE, 2021, 页码: 8
作者:
Ding, Yu-chao
;
Zhang, Xian-jing
;
Zhang, Ji-xiu
;
Zhai, Zi-yi
;
Zhang, Mei-xia
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2021/12/01
abdominal aortic aneurysm
disease progression
disease regression
elastogenesis
lysyl oxidase
Pharmacokinetics and Disposition of Contezolid in Humans: Resolution of a Disproportionate Human Metabolite for Clinical Development
期刊论文
OAI收割
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 2021, 卷号: 65, 期号: 11, 页码: 13
作者:
Wu, Xiaojie
;
Meng, Jian
;
Yuan, Hong
;
Zhong, Dafang
;
Yu, Jicheng
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2022/06/15
contezolid
disposition
metabolism
pharmacokinetics
Competitive CatSper Activators of Progesterone from Rhynchosia volubilis
期刊论文
OAI收割
PLANTA MEDICA, 2021, 页码: 10
作者:
Xiang, Jin
;
Kang, Hang
;
Li, Hong-Gang
  |  
收藏
  |  
浏览/下载:47/0
  |  
提交时间:2021/11/04
Leguminosae
Rhynchosia volubilis
CatSper
prenylated isoflavonoids
rhynchones A - E
Pharmacodynamic, pharmacokinetic, and phase 1a study of bisthianostat, a novel histone deacetylase inhibitor, for the treatment of relapsed or refractory multiple myeloma
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 9
作者:
Zhou, Yu-bo
;
Zhang, Yang-ming
;
Huang, Hong-hui
;
Shen, Li-jing
;
Han, Xiao-feng
  |  
收藏
  |  
浏览/下载:68/0
  |  
提交时间:2021/11/04
multiple myeloma
HDAC inhibitor
bisthianostat
pharmacodynamics
pharmacokinetics
phase 1a clinical trial
antitumor drug
Development of Potent NEDD8-Activating Enzyme Inhibitors Bearing a Pyrimidotriazole Scaffold
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 9, 页码: 6161-6178
作者:
Xiong, Chaodong
;
Zhou, Lina
;
Tan, Jing
;
Song, Shanshan
;
Bao, Xubin
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2021/08/17
Natural product 1,2,3,4,6-penta-O-galloyl-beta-D-glucopyranose is a reversible inhibitor of glyceraldehyde 3-phosphate dehydrogenase
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 13
作者:
Li, Wen
;
Liao, Li-ping
;
Song, Ning
;
Liu, Yan-jun
;
Ding, Yi-luan
  |  
收藏
  |  
浏览/下载:44/0
  |  
提交时间:2021/06/11
glyceraldehyde 3-phosphate dehydrogenase
1,2,3,4,6-penta-O-galloyl-beta-D-glucopyranose
hydrogen deuterium exchange mass spectrometry
reversible inhibitor
glycolysis
Natural product 1,2,3,4,6-penta-O-galloyl-beta-D-glucopyranose is a reversible inhibitor of glyceraldehyde 3-phosphate dehydrogenase
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 13
作者:
Li, Wen
;
Liao, Li-ping
;
Song, Ning
;
Liu, Yan-jun
;
Ding, Yi-luan
  |  
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2021/06/11
glyceraldehyde 3-phosphate dehydrogenase
1,2,3,4,6-penta-O-galloyl-beta-D-glucopyranose
hydrogen deuterium exchange mass spectrometry
reversible inhibitor
glycolysis
P300/CBP inhibition sensitizes mantle cell lymphoma to PI3K delta inhibitor idelalisib
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 13
作者:
Zhou, Xiao-ru
;
Li, Xiao
;
Liao, Li-ping
;
Han, Jie
;
Huang, Jing
  |  
收藏
  |  
浏览/下载:49/0
  |  
提交时间:2021/06/11
mantle cell lymphoma
idelalisib
drug resistance
P300
CBP
synergistic drug action
PI3Kδ
epigenetics