中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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昆明动物研究所 [39]
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Structure-Based Design of Tropane Derivatives as a Novel Series of CCR5 Antagonists with Broad-Spectrum Anti-HIV-1 Activities and Improved Oral Bioavailability
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 24, 页码: 16526-16540
作者:
Xie, Xiong
;
Zheng, Yu-Gui
;
Chen, Huan
;
Li, Jian
;
Luo, Rong-Hua
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2023/04/10
Natural products for infectious microbes and diseases: an overview of sources, compounds, and chemical diversities
期刊论文
OAI收割
SCIENCE CHINA-LIFE SCIENCES, 2022, 卷号: 65, 期号: 6, 页码: 1123-1145
作者:
Luo, Lu
;
Yang, Jun
;
Wang, Cheng
;
Wu, Jie
;
Li, Yafang
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/03/07
natural product
infectious pathogen
drug discovery
drug development
in silico analysis
Antitubercular Ilamycins from Marine-Derived Streptomyces atratus SCSIO ZH16 Delta ilaR
期刊论文
OAI收割
JOURNAL OF NATURAL PRODUCTS, 2020, 卷号: 83, 期号: 5, 页码: 1646, 1657
作者:
Sun, Changli
;
Liu, Zhiyong
;
Zhu, Xiangcheng
;
Fan, Zhiying
;
Huang, Xuanmei
  |  
收藏
  |  
浏览/下载:63/0
  |  
提交时间:2020/09/22
Configurationally Stable (S)- and (R)--Methylproline-Derived Ligands for the Direct Chemical Resolution of Free Unprotected (3)-Amino Acids
期刊论文
OAI收割
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2018, 期号: 15, 页码: 1821-1832
作者:
Zhou, Shengbin
;
Wang, Shuni
;
Wang, Jiang
;
Nian, Yong
;
Peng, Panfeng
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2019/01/08
Amino acids
Chemical resolution
Nickel
Nonracemizable ligands
Antiviral agents
Hit optimization studies of 3-hydroxy-indolin-2-one analogs as potential anti-HIV-1 agents
期刊论文
OAI收割
Bioorganic chemistry, 2018, 期号: 79, 页码: 212-222
作者:
Subhash Chander
;
Murugesan Sankaranarayanan
;
Ashok Penta
;
Ping Wang
;
Deepak P. Bhagwat
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2018/09/19
Aids
Reverse Transcriptase
Toxicity
Virtual Screening
Sar
Docking
14-Formyl-15-aryloxy/methoxymatrine and 14-Aryloxymethylidenyl-mat- rine Derivatives as Anti-HIV-1 Agents
期刊论文
OAI收割
Medicinal Chemistry, 2018, 期号: 14, 页码: 249-252
作者:
Jiulin Huang
;
Liu-Meng Yang
;
Yuanyuan Zhang
;
Yong-Tang Zheng
;
Hui Xu
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2018/09/20
Matrine Derivatives
Aids
Hiv-1
Inhibitors
Antiretroviral Drugs
Peptide Drugs
Matrines
Novel tetrahydrofuran derivatives from Trigonostemon howii with their potential anti-HIV-1 activities
期刊论文
OAI收割
Bioorganic Chemistry, 2018, 期号: 79, 页码: 111–114
作者:
Xing-Yang Feng
;
Wan-Hui Zhao
;
Yan-Ping Liu
;
Yong-Tang Zheng
;
Zhi-Guo Sun
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2018/09/25
Trigonostemon Howii
Tetrahydrofuran Derivatives
Trigonohowine
Anti-hiv-1 Activities
Synthesis and Biological Evaluation of Benzophenone Derivatives as Poten- tial HIV-1 Inhibitors
期刊论文
OAI收割
Medicinal Chemistry, 2017, 卷号: 13, 期号: X, 页码: 98-405
作者:
Zhen YH
;
xiaodong.ma@139.com
;
Wang RR
;
Wang CY
;
Huang SS
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2017/10/19
Activity
Aids
Analogues
Benzophenone
Hiv-1
Inhibitor
Synthesis and Anti-HIV-1 Activity Evaluation for Novel 3a,6a-Dihydro-1H-pyrrolo[3,4-c]pyrazole-4,6-dione Derivatives
期刊论文
OAI收割
MOLECULES, 2016, 卷号: 21, 期号: 9
作者:
Liu, Guan-Nan
;
Luo, Rong-Hua
;
Zhou, Yu
;
Zhang, Xing-Jie
;
Li, Jian
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2019/01/08
anti-HIV-1
integrase
synthesis
SAR
AIDS
Design, synthesis and anti-HIV-1 evaluation of hydrazide-based peptidomimetics as selective gelatinase inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 9, 页码: 2125-2136
作者:
Yang L
;
Wang P
;
Pang W
;
Li YG
;
Shen YM
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2016/04/05
Hydrazide derivatives
Quinoxalinone
Selective gelatinase inhibitors
Peptidomimetics
Anti-HIV activity