中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [7]
化学研究所 [1]
寒区旱区环境与工程研... [1]
上海有机化学研究所 [1]
青岛生物能源与过程研... [1]
中国科学院大学 [1]
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OAI收割 [15]
iSwitch采集 [2]
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期刊论文 [17]
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2023 [1]
2022 [2]
2018 [2]
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2016 [2]
2015 [1]
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Biochemist... [1]
生命有机化学 [1]
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Design, synthesis and biological evaluation of peptidomimetic benzothiazolyl ketones as 3CLpro inhibitors against SARS-CoV-2
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 257, 页码: 13
作者:
Yang, Hanxi
;
You, Mengyuan
;
Shu, Xiaoyang
;
Zhen, Jingyao
;
Zhu, Mengwei
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2023/10/17
Peptidomimetics
Benzothiazolyl ketone
3CLpro inhibitor
Pharmacokinetic properties
SARS-CoV-2
Synthesis of maleimide-braced peptide macrocycles and their potential anti-SARS-CoV-2 mechanisms
期刊论文
OAI收割
CHEMICAL COMMUNICATIONS, 2022, 页码: 4
作者:
Li, Jian
;
Sun, Jina
;
Zhang, Xianglei
;
Zhang, Ruxue
;
Wang, Qian
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2023/04/10
Metabolism guided optimization of peptidomimetics as non-covalent proteasome inhibitors for cancer treatment
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 233, 页码: 18
作者:
Cao, Yu
;
Tu, Yutong
;
Fu, Liping
;
Yu, Qian
;
Gao, Lixin
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2022/06/15
Metabolism
Design
Proteasome inhibitors
Non-covalent
Multiple myeloma
Oncolysis with DTT-205 and DTT-304 generates immunological memory in cured animals
期刊论文
iSwitch采集
CELL DEATH & DISEASE, 2018, 卷号: 9, 页码: 14
作者:
Zhou, Heng
;
Mondragon, Laura
;
Xie, Wei
;
Mauseth, Brynjar
;
Leduc, Marion
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2019/10/09
Oncolysis with DTT-205 and DTT-304 generates immunological memory in cured animals
期刊论文
OAI收割
CELL DEATH & DISEASE, 2018, 卷号: 9
作者:
Zhou, Heng
;
Mondragon, Laura
;
Xie, Wei
;
Mauseth, Brynjar
;
Leduc, Marion
  |  
收藏
  |  
浏览/下载:45/0
  |  
提交时间:2019/03/27
Peptidomimetic inhibitors of APC-Asef interaction block colorectal cancer migration
期刊论文
OAI收割
NATURE CHEMICAL BIOLOGY, 2017, 卷号: 13, 期号: 9, 页码: 994
作者:
Jiang, Haiming
;
Deng, Rong
;
Yang, Xiuyan
;
Shang, Jialin
;
Lu, Shaoyong
  |  
收藏
  |  
浏览/下载:54/0
  |  
提交时间:2018/12/29
Peptidomimetic inhibitors of APC-Asef interaction block colorectal cancer migration
期刊论文
OAI收割
NATURE CHEMICAL BIOLOGY, 2017, 卷号: 13, 期号: 9, 页码: 994-+
作者:
Jiang, Haiming
;
Deng, Rong
;
Yang, Xiuyan
;
Shang, Jialin
;
Lu, Shaoyong
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2020/12/09
Patient-derived tumor xenograft
gene expression profile
Monte Carlo feature selection
support vector machine
rule learning algorithm
3-Azidoazetidines as the first scaffolds for beta-amino azetidine carboxylic acid peptidomimetics: azetidine iminosugars containing an acetamido group do not inhibit beta-N-acetylhexosaminidases
期刊论文
OAI收割
TETRAHEDRON-ASYMMETRY, 2016, 卷号: 27, 期号: 17-18, 页码: 872-881
作者:
Liu, Zilei
;
Jenkinson, Sarah F.
;
Kato, Atsushi
;
Nakagawa, Shinpei
;
Wormald, Mark R.
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2016/12/29
Design, synthesis and anti-HIV-1 evaluation of hydrazide-based peptidomimetics as selective gelatinase inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 9, 页码: 2125-2136
作者:
Yang L
;
Wang P
;
Pang W
;
Li YG
;
Shen YM
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2016/04/05
Hydrazide derivatives
Quinoxalinone
Selective gelatinase inhibitors
Peptidomimetics
Anti-HIV activity
Asymmetric Synthesis of (2S,3S)-alpha-(1-Oxoisoindolin-3-yl)glycines under Low-Basicity "Kinetic" Control
期刊论文
OAI收割
JOURNAL OF ORGANIC CHEMISTRY, 2015, 卷号: 80, 期号: 22, 页码: 11275-11280
作者:
Li, Tingting
;
Zhou, Shengbin
;
Wang, Jiang
;
Acena, Jose Luis
;
Soloshonok, Vadim A.
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/01/08