中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共10条,第1-10条 帮助

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Design, synthesis of auristatins-glucuronide conjugates targeting the β-glucuronidase in tumor microenvironment 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2023, 卷号: 95, 页码: 5
作者:  
Wang, Yujie;  Xu, Keshi;  Liu, Hongchun;  Zhang, Wei;  Hu, Chun
  |  收藏  |  浏览/下载:4/0  |  提交时间:2023/12/19
Preclinical Evaluation of 9MW2821, a Site-Specific Monomethyl Auristatin E-based Antibody-Drug Conjugate for Treatment of Nectin-4-expressing Cancers 期刊论文  OAI收割
MOLECULAR CANCER THERAPEUTICS, 2023, 卷号: 22, 期号: 8, 页码: 913-925
作者:  
Zhou, Wei;  Fang, Peng;  Yu, Dongan;  Ren, Hongyuan;  You, Meng
  |  收藏  |  浏览/下载:11/0  |  提交时间:2023/10/17
Enzyme-linked immunosorbent assays for quantification of MMAE-conjugated ADCs and total antibodies in cynomolgus monkey sera 期刊论文  OAI收割
JOURNAL OF PHARMACEUTICAL ANALYSIS, 2022, 卷号: 12, 期号: 4, 页码: 645-652
作者:  
Pei, Min;  Liu, Tingting;  Ouyang, Lu;  Sun, Jianhua;  Deng, Xiaojie
  |  收藏  |  浏览/下载:37/0  |  提交时间:2022/11/11
CD71-Specific Aptamer Conjugated with Monomethyl Auristatin E for the Treatment of Uveal Melanoma 期刊论文  OAI收割
ACS APPLIED MATERIALS & INTERFACES, 2021
作者:  
Zhang, Hui;  Jin, Cheng;  Zhang, Lin;  Peng, Bo;  Zhang, Yibin
  |  收藏  |  浏览/下载:36/0  |  提交时间:2022/02/14
An antibody-drug conjugate targeting a GSTA glycosite-signature epitope of MUC1 expressed by non-small cell lung cancer 期刊论文  OAI收割
CANCER MEDICINE, 2020, 页码: 12
作者:  
Pan, Deng;  Tang, Yubo;  Tong, Jiao;  Xie, Chengmei;  Chen, Jiaxi
  |  收藏  |  浏览/下载:33/0  |  提交时间:2020/12/24
Construction of Bispecific Aptamer-Drug Conjugate by a Hybrid Chemical and Biological Approach 期刊论文  OAI收割
BIOCONJUGATE CHEMISTRY, 2020, 卷号: 31
作者:  
Sun, Yang;  Gao, Fei;  Yang, Cai;  Li, Yingying;  Jin, Cheng
  |  收藏  |  浏览/下载:38/0  |  提交时间:2020/11/26
Aberrant intracellular metabolism of T-DM1 confers T-DM1 resistance in human epidermal growth factor receptor 2-positive gastric cancer cells 期刊论文  OAI收割
CANCER SCIENCE, 2017, 卷号: 108, 期号: 7, 页码: 1458-1468
作者:  
Wang, Hongbin;  Wang, Wenqian;  Xu, Yongping;  Yang, Yong;  Chen, Xiaoyan
  |  收藏  |  浏览/下载:30/0  |  提交时间:2019/01/08
HER2-targeted antibody drug conjugates for ovarian cancer therapy 期刊论文  OAI收割
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2016, 卷号: 93, 页码: 274-286
作者:  
Jiang, Jing;  Dong, Lihou;  Wang, Lei;  Wang, Ling;  Zhang, Jing
  |  收藏  |  浏览/下载:52/0  |  提交时间:2019/01/08
Structural Insights into the Pharmacophore of Vinca Domain Inhibitors of Microtubules 期刊论文  OAI收割
MOLECULAR PHARMACOLOGY, 2016, 卷号: 89, 期号: 2, 页码: 233—242
作者:  
Wang, YX;  Benz, FW;  Wu, YP;  Wang, QS;  Chen, YF
收藏  |  浏览/下载:29/0  |  提交时间:2016/09/12
An anti-HER2 antibody conjugated with monomethyl auristatin E is highly effective in HER2-positive human gastric cancer 期刊论文  OAI收割
CANCER BIOLOGY & THERAPY, 2016, 卷号: 17, 期号: 4, 页码: 346-354
作者:  
Li, Hongwen;  Yu, Chao;  Jiang, Jing;  Huang, Changjiang;  Yao, Xuejing
  |  收藏  |  浏览/下载:29/0  |  提交时间:2019/01/08