中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
首页
机构
成果
学者
登录
注册
登陆
×
验证码:
换一张
忘记密码?
记住我
×
校外用户登录
CAS IR Grid
机构
上海药物研究所 [10]
合肥物质科学研究院 [2]
上海营养与健康研究所 [1]
采集方式
OAI收割 [13]
内容类型
期刊论文 [13]
发表日期
2023 [2]
2022 [1]
2021 [4]
2020 [2]
2019 [2]
2018 [1]
更多
学科主题
Biochemist... [1]
Biophysics [1]
筛选
浏览/检索结果:
共13条,第1-10条
帮助
条数/页:
5
10
15
20
25
30
35
40
45
50
55
60
65
70
75
80
85
90
95
100
排序方式:
请选择
提交时间升序
提交时间降序
发表日期升序
发表日期降序
题名升序
题名降序
作者升序
作者降序
Degradation of Cyclin-Dependent Kinase 9/Cyclin T1 by Optimized Microtubule-Associated Protein 1 Light Chain 3 Beta-Recruiting Coumarin Analogs
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 17
作者:
Zeng, Yanping
;
Xiao, Jian
;
Xu, Yuanxin
;
Wei, Fan
;
Tian, Lina
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2023/10/17
Predicting and overcoming resistance to CDK9 inhibitors for cancer therapy
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13
作者:
Hua, Chen
;
Shena, Lijuan
;
Zoua, Fengming
;
Wua, Yun
;
Wanga, Beilei
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/11/10
Acquired resistance mutations
CDK9 inhibitors
Transcription
Single nucleotide polymorphisms
BAY1251152
CDK9 inhibitors in cancer research
期刊论文
OAI收割
RSC MEDICINAL CHEMISTRY, 2022
作者:
Huang, Zhi
;
Wang, Tianqi
;
Wang, Cheng
;
Fan, Yan
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2022/12/23
Discovery of Potent and Selective CDK9 Degraders for Targeting Transcription Regulation in Triple-Negative Breast Cancer
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 19, 页码: 14822-14847
作者:
Wei, Dan
;
Wang, Hanlin
;
Zeng, Qinghe
;
Wang, Wenjing
;
Hao, Bingbing
  |  
收藏
  |  
浏览/下载:45/0
  |  
提交时间:2021/12/16
Rational Design and Development of Novel CDK9 Inhibitors for the Treatment of Acute Myeloid Leukemia
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 19, 页码: 14647-14663
作者:
Han, Xu
;
Song, Ning
;
Saidahmatov, Abdusaid
;
Wang, Peipei
;
Wang, Yong
  |  
收藏
  |  
浏览/下载:58/0
  |  
提交时间:2021/12/16
Efficient Synthesis and Docking Analysis of Selective CDK9 Inhibitor NVP-2
期刊论文
OAI收割
Pharmaceutical Fronts, 2021, 期号: 3, 页码: E50-E55
作者:
Saidahmatov, Abdusaid
;
Liang, Xue-Wu
;
Shi, Yuqiang
;
Han, Xu
;
Liu, Hong
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/03/14
NVP-2
CDK9 inhitor
efficient synthesis
docking analysis
Discovery of selective CDK9 degraders with enhancing antiproliferative activity through PROTAC conversion
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 211, 页码: 11
作者:
Qiu, Xiaqiu
;
Li, Yuanqing
;
Yu, Bin
;
Ren, Jie
;
Huang, Huidan
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2021/05/24
CDK9
Antitumor
PROTAC
AML
Degrader
Rational Design and Evaluation of 6-(Pyrimidin-2-ylamino)-3,4-dihydroquinoxalin-2(1H)-ones as Polypharmacological Inhibitors of BET and Kinases
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 17, 页码: 9787-9802
作者:
Lv, Kaikai
;
Chen, Weicong
;
Chen, Danqi
;
Mou, Jie
;
Zhang, Huijie
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2020/12/21
EZH2 inhibitors abrogate upregulation of trimethylation of H3K27 by CDK9 inhibitors and potentiate its activity against diffuse large B-cell lymphoma
期刊论文
OAI收割
HAEMATOLOGICA, 2020, 卷号: 105, 期号: 4, 页码: 1021-1031
作者:
Xie, Shao
;
Wei, Fan
;
Sun, Yi-ming
;
Gao, Ying-lei
;
Pan, Lu-lu
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2020/07/01
Design of wogonin-inspired selective cyclin-dependent kinase 9 (CDK9) inhibitors with potent in vitro and in vivo antitumor activity
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 178, 页码: 782-801
作者:
Wang, Jubo
;
Li, Tinghan
;
Zhao, Tengteng
;
Wu, Tizhi
;
Liu, Chuang
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2020/07/01
Wogonin
CDK9
AML
Flavonoid
Antitumor