中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共13条,第1-10条 帮助

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Degradation of Cyclin-Dependent Kinase 9/Cyclin T1 by Optimized Microtubule-Associated Protein 1 Light Chain 3 Beta-Recruiting Coumarin Analogs 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 17
作者:  
Zeng, Yanping;  Xiao, Jian;  Xu, Yuanxin;  Wei, Fan;  Tian, Lina
  |  收藏  |  浏览/下载:7/0  |  提交时间:2023/10/17
Predicting and overcoming resistance to CDK9 inhibitors for cancer therapy 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13
作者:  
Hua, Chen;  Shena, Lijuan;  Zoua, Fengming;  Wua, Yun;  Wanga, Beilei
  |  收藏  |  浏览/下载:11/0  |  提交时间:2023/11/10
CDK9 inhibitors in cancer research 期刊论文  OAI收割
RSC MEDICINAL CHEMISTRY, 2022
作者:  
Huang, Zhi;  Wang, Tianqi;  Wang, Cheng;  Fan, Yan
  |  收藏  |  浏览/下载:10/0  |  提交时间:2022/12/23
Discovery of Potent and Selective CDK9 Degraders for Targeting Transcription Regulation in Triple-Negative Breast Cancer 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 19, 页码: 14822-14847
作者:  
Wei, Dan;  Wang, Hanlin;  Zeng, Qinghe;  Wang, Wenjing;  Hao, Bingbing
  |  收藏  |  浏览/下载:45/0  |  提交时间:2021/12/16
Rational Design and Development of Novel CDK9 Inhibitors for the Treatment of Acute Myeloid Leukemia 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 19, 页码: 14647-14663
作者:  
Han, Xu;  Song, Ning;  Saidahmatov, Abdusaid;  Wang, Peipei;  Wang, Yong
  |  收藏  |  浏览/下载:58/0  |  提交时间:2021/12/16
Efficient Synthesis and Docking Analysis of Selective CDK9 Inhibitor NVP-2 期刊论文  OAI收割
Pharmaceutical Fronts, 2021, 期号: 3, 页码: E50-E55
作者:  
Saidahmatov, Abdusaid;  Liang, Xue-Wu;  Shi, Yuqiang;  Han, Xu;  Liu, Hong
  |  收藏  |  浏览/下载:8/0  |  提交时间:2024/03/14
Discovery of selective CDK9 degraders with enhancing antiproliferative activity through PROTAC conversion 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 211, 页码: 11
作者:  
Qiu, Xiaqiu;  Li, Yuanqing;  Yu, Bin;  Ren, Jie;  Huang, Huidan
  |  收藏  |  浏览/下载:24/0  |  提交时间:2021/05/24
CDK9  Antitumor  PROTAC  AML  Degrader  
Rational Design and Evaluation of 6-(Pyrimidin-2-ylamino)-3,4-dihydroquinoxalin-2(1H)-ones as Polypharmacological Inhibitors of BET and Kinases 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 17, 页码: 9787-9802
作者:  
Lv, Kaikai;  Chen, Weicong;  Chen, Danqi;  Mou, Jie;  Zhang, Huijie
  |  收藏  |  浏览/下载:22/0  |  提交时间:2020/12/21
EZH2 inhibitors abrogate upregulation of trimethylation of H3K27 by CDK9 inhibitors and potentiate its activity against diffuse large B-cell lymphoma 期刊论文  OAI收割
HAEMATOLOGICA, 2020, 卷号: 105, 期号: 4, 页码: 1021-1031
作者:  
Xie, Shao;  Wei, Fan;  Sun, Yi-ming;  Gao, Ying-lei;  Pan, Lu-lu
  |  收藏  |  浏览/下载:27/0  |  提交时间:2020/07/01
Design of wogonin-inspired selective cyclin-dependent kinase 9 (CDK9) inhibitors with potent in vitro and in vivo antitumor activity 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 178, 页码: 782-801
作者:  
Wang, Jubo;  Li, Tinghan;  Zhao, Tengteng;  Wu, Tizhi;  Liu, Chuang
  |  收藏  |  浏览/下载:17/0  |  提交时间:2020/07/01