中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [18]
西北高原生物研究所 [9]
上海生物化学与细胞生... [6]
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Development of the novel ACLY inhibitor 326E as a promising treatment for hypercholesterolemia
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13, 期号: 2, 页码: 739-753
作者:
Xie, Zhifu
;
Zhang, Mei
;
Song, Qian
;
Cheng, Long
;
Zhang, Xinwen
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2024/03/27
Hypercholesterolemia
Atherosclerosis
Liver
ATP-Citrate lyase (ACLY)
Lipogenesis
Cholesterol efflux
ACLY inhibitor
Discovery of Novel Long-Chain Alkenyl Diacid Derivatives as ACLY Inhibitors
期刊论文
OAI收割
CHINESE JOURNAL OF CHEMISTRY, 2022, 页码: 8
作者:
Song, Gao-Lei
;
Cao, Lei
;
Zhang, Mei
;
Yang, Yu-Rou
;
Ma, Jie
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2022/09/30
Alkenyl diacid derivatives
Cancer
ACLY inhibitors
Acetyl-CoA
Structure-activity relationships
Identification and evaluation of a lipid-lowering small compound in preclinical models and in a Phase I trial
期刊论文
OAI收割
CELL METABOLISM, 2022, 卷号: 34, 期号: 5, 页码: 667-+
作者:
Wang, Jiang
;
Zhao, Jing
;
Yan, Cong
;
Xi, Cong
;
Wu, Chenglin
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2022/08/16
Oxidized Low-Density Lipoprotein Links Hypercholesterolemia and Bladder Cancer Aggressiveness by Promoting Cancer Stemness
期刊论文
OAI收割
CANCER RESEARCH, 2021, 卷号: 81, 期号: 22, 页码: 5720-5732
作者:
Yang, Lin
;
Sun, Jingya
;
Li, Meiqian
;
Long, Yiming
;
Zhang, Dianzheng
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2022/01/04
23,24-Dihydrocucurbitacin B promotes lipid clearance by dual transcriptional regulation of LDLR and PCSK9
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2020, 卷号: 41, 期号: 3, 页码: 327-335
作者:
Li, Hui-hui
;
Li, Jun
;
Zhang, Xian-jing
;
Li, Jiao-meng
;
Xi, Cong
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2020/07/01
23,24-dihydrocucurbitacin B
lipid-lowering agent
LDLR
PCSK9
HNF1 alpha
SREBP2
Phytochemical and biological studies on rare and endangered plants endemic to China. Part XV. Structurally diverse diterpenoids and sesquiterpenoids from the vulnerable conifer Pseudotsuga sinensis
期刊论文
OAI收割
PHYTOCHEMISTRY, 2020, 卷号: 169, 页码: 14
作者:
Huang, Ting
;
Ying, Sheng-Hui
;
Li, Jing-Ya
;
Chen, Hao-Wei
;
Zang, Yi
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2020/07/01
Pseudotsuga sinensis dode
Pinaceae
Rare and endangered plants (REPs)
Degraded diterpenoids
Pseudosinins
ATP-Citrate lyase (ACL)
PAQR3 modulates blood cholesterol level by facilitating interaction between LDLR and PCSK9
期刊论文
OAI收割
METABOLISM-CLINICAL AND EXPERIMENTAL, 2019, 卷号: 94, 期号: -, 页码: 88-95
作者:
Huang, Meiqin
;
Zhao, Zilong
;
Cao, Qianqian
;
Wei, Siying
;
Zhao, Jingyu
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2020/12/09
Low-density lipoprotein cholesterol
LDLR
PCSK9
Endosome
Protein degradation
The first pediatric case of glucagon receptor defect due to biallelic mutations in GCGR is identified by newborn screening of elevated arginine
期刊论文
OAI收割
MOLECULAR GENETICS AND METABOLISM REPORTS, 2018, 卷号: 17, 页码: 46-52
作者:
Li, Hong
;
Zhao, Lihua
;
Singh, Rani
;
Ham, J. Nina
;
Fadoju, Doris O.
  |  
收藏
  |  
浏览/下载:84/0
  |  
提交时间:2019/01/08
Glucagon receptor
Newborn screening
GCGR mutation
Hyperaminoacidemia
Mahvash disease
Pancreatic alpha cell hyperplasia (ACH)
Pancreatic neuroendocrine tumor (PNET)
Proteomics analysis reveals a potential new target protein for the lipid-lowering effect of Berberine8998
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 9, 页码: 1473-1482
作者:
Yu, Cheng-yin
;
Liu, Gang-yi
;
Liu, Xiao-hui
;
Gui, Yu-zhou
;
Liu, Hai-ming
  |  
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2019/01/08
berberine
berberine8998
proteomics
lipid-lowering
cholesterol
triglycerides
LDL-C
fatty acid metabolism
hypercholesterolemia
obesity
Effect of Medium-chain Fatty Acid-sensing Receptor GPR84 on Glucose and Lipid Metabolism in Mice
期刊论文
OAI收割
PROGRESS IN BIOCHEMISTRY AND BIOPHYSICS, 2018, 卷号: 45, 期号: 8, 页码: 853-864
作者:
Fang You-Chen
;
Zheng Yang
;
Zheng Qing
;
Li Jing
;
Xie Xin
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2019/01/08
GPR84
medium-chain fatty acid-sensing receptor
obesity
lipid metabolism
hypercholesterolemia