中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共52条,第1-10条 帮助

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Discovery of novel triazine derivatives as potent retinoic acid receptor-related orphan receptor gamma t (ROR gamma t) inverse agonists 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 256, 页码: 18
作者:  
Lu, Lixue;  Chen, Song;  Yu, Mingcheng;  Zhou, Ronghui;  Guo, Siqi
  |  收藏  |  浏览/下载:15/0  |  提交时间:2023/10/17
Identification of methyl (5-(6-((4-(methylsulfonyl)piperazin-1-yl)methyl)-4-morpholinopyrrolo[2,1-f][1,2,4]triazin-2-yl)-4-(trifluoromethyl)pyridin-2-yl)carbamate (CYH33) as an orally bioavailable, highly potent, PI3K alpha inhibitor for the treatment of advanced solid tumors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 209, 页码: 10
作者:  
Xiang, Hao-Yue;  Wang, Xiang;  Chen, Yan-Hong;  Zhang, Xi;  Tan, Cun
  |  收藏  |  浏览/下载:24/0  |  提交时间:2021/05/24
Synthesis of Highly Fused Pyrano[2,3-b]pyridines via Rh(III)- Catalyzed C-H Activation and Intramolecular Cascade Annulation under Room Temperature 期刊论文  OAI收割
JOURNAL OF ORGANIC CHEMISTRY, 2020, 卷号: 85, 期号: 10, 页码: 6281-6294
作者:  
Han, Xu;  Gao, Feng;  Li, Chunpu;  Fang, Daqing;  Xie, Xiong
  |  收藏  |  浏览/下载:23/0  |  提交时间:2020/07/01
Novel oxacalix[2]arene[2]triazines with thermally activated delayed fluorescence and aggregation-induced emission properties 期刊论文  OAI收割
CHEMICAL COMMUNICATIONS, 2019, 卷号: 55, 期号: 64, 页码: 9559-9562
作者:  
Wang, Yin-Feng;  Lu, Hai-Yan;  Shen, Yi-Fan;  Li, Meng;  Chen, Chuan-Feng
  |  收藏  |  浏览/下载:41/0  |  提交时间:2019/09/30
Recent Developments in the Synthesis of Nitrogen-Containing Heterocycles through C-H/N-H Bond Functionalizations and Oxidative Cyclization 期刊论文  OAI收割
SYNLETT, 2019, 卷号: 30, 期号: 9, 页码: 1026-1036
作者:  
Liu, Xiang;  Huang, Yu
  |  收藏  |  浏览/下载:68/0  |  提交时间:2019/07/15
Low-cost and convenient ballpoint tip-protected liquid-phase microextraction for sensitive analysis of organic molecules in water samples 期刊论文  OAI收割
ANALYTICA CHIMICA ACTA, 2019, 卷号: 1006, 页码: 42-48
作者:  
Ji, Baocheng;  Xia, Bing;  Fu, Xian;  Lei, Shan;  Ye, Ye
  |  收藏  |  浏览/下载:18/0  |  提交时间:2020/12/24
Design, Synthesis and Pharmacological Evaluation of Novel Hsp90N-terminal Inhibitors Without Induction of Heat Shock Response 期刊论文  OAI收割
CHEMISTRYOPEN, 2019, 卷号: 8, 期号: 3, 页码: 344-353
作者:  
Liu, Peng;  Chen, Xiangling;  Zhu, Jianming;  Li, Bo;  Chen, Zhaoqiang
  |  收藏  |  浏览/下载:46/0  |  提交时间:2020/07/01
Design, Synthesis, and SAR Studies of Heteroarylpyrimidines and Heteroaryltriazines as CB2R Ligands 期刊论文  OAI收割
CHEMMEDCHEM, 2018, 卷号: 13, 期号: 22, 页码: 2455-2463
作者:  
Qian, Hai-Yan;  Wang, Zhi-Long;  Chen, Li-Li;  Pan, You-Lu;  Xie, Xiao-Yu
  |  收藏  |  浏览/下载:90/0  |  提交时间:2019/01/08
Silver-catalyzed [3+2+1] annulation of aryl amidines with benzyl isocyanide 期刊论文  OAI收割
TETRAHEDRON LETTERS, 2018, 卷号: 59, 期号: 4, 页码: 361-364
作者:  
Lu, Xiaodong;  Xin, Xiaoyi;  Wan, Boshun
  |  收藏  |  浏览/下载:15/0  |  提交时间:2019/06/20
Synthesis of carboxylate head-containing self-complementary building units and their anion- directed self-assembly 期刊论文  OAI收割
SUPRAMOLECULAR CHEMISTRY, 2018, 卷号: 30, 期号: 7, 页码: 568-574
作者:  
Xu, Rui-Bin;  Wang, Qi-Qiang;  Ao, Yu-Fei;  Wang, De-Xian
  |  收藏  |  浏览/下载:48/0  |  提交时间:2019/04/09