中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共275条,第1-10条 帮助

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NIR-II fluorescence-guided liver cancer surgery by a small molecular HDAC6 targeting probe 期刊论文  OAI收割
EBIOMEDICINE, 2023, 卷号: 98, 页码: 18
作者:  
Wang, Bo;  Tang, Chu;  Lin, En;  Jia, Xiaohua;  Xie, Ganyuan
  |  收藏  |  浏览/下载:14/0  |  提交时间:2024/02/22
TI17, a novel compound, exerts anti-MM activity by impairing Trip13 function of DSBs repair and enhancing DNA damage 期刊论文  OAI收割
CANCER MEDICINE, 2023, 页码: 14
作者:  
Chang, Shuaikang;  Xiao, Wenqin;  Xie, Yongsheng;  Xu, Zhijian;  Li, Bo
  |  收藏  |  浏览/下载:7/0  |  提交时间:2023/12/11
Design, synthesis of auristatins-glucuronide conjugates targeting the β-glucuronidase in tumor microenvironment 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2023, 卷号: 95, 页码: 5
作者:  
Wang, Yujie;  Xu, Keshi;  Liu, Hongchun;  Zhang, Wei;  Hu, Chun
  |  收藏  |  浏览/下载:4/0  |  提交时间:2023/12/19
Design, synthesis, and biological evaluation of novel spirocyclic compounds as potential anti-glioblastoma agents 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 258, 页码: 22
作者:  
Zhu, Heping;  Song, Xiaomin;  Pan, Yihui;  Li, Ming;  Chen, Liang
  |  收藏  |  浏览/下载:11/0  |  提交时间:2023/10/17
[68Ga]Ga-AUNP-12 PET imaging to assess the PD-L1 status in preclinical and first-in-human study 期刊论文  OAI收割
EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING, 2023, 页码: 11
作者:  
Zhou, Ming;  Xiang, Shijun;  Zhao, Yajie;  Tang, Yongxiang;  Yang, Jinhui
  |  收藏  |  浏览/下载:6/0  |  提交时间:2023/11/16
Discovery of ARD-1676 as a Highly Potent and Orally Efficacious AR PROTAC Degrader with a Broad Activity against AR Mutants for the Treatment of AR plus Human Prostate Cancer 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 18, 页码: 13280-13303
作者:  
Xiang, Weiguo;  Zhao, Lijie;  Han, Xin;  Xu, Tianfeng;  Kregel, Steven
  |  收藏  |  浏览/下载:9/0  |  提交时间:2023/12/08
Discovery, structural optimization, and anti-tumor bioactivity evaluations of betulinic acid derivatives as a new type of ROR & gamma; antagonists 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 257, 页码: 15
作者:  
  |  收藏  |  浏览/下载:39/0  |  提交时间:2023/10/17
Discovery of 2-Aminopyrimidine Derivatives as Potent Dual FLT3/CHK1 Inhibitors with Significantly Reduced hERG Inhibitory Activities 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 23
作者:  
Li, Xuemei;  Wang, Peipei;  Wang, Chang;  Jin, Tingting;  Xu, Ran
  |  收藏  |  浏览/下载:14/0  |  提交时间:2023/10/17
Novel thieno[2,3-b]quinoline-procaine hybrid molecules: A new class of allosteric SHP-1 activators evolved from PTP1B inhibitors 期刊论文  OAI收割
CHINESE CHEMICAL LETTERS, 2023, 卷号: 34, 期号: 8, 页码: 6
作者:  
Xu, Lei;  Xuyan, Xuyang;  Minmi, Minmin;  Wang, Zhiji;  Shee, Chao
  |  收藏  |  浏览/下载:27/0  |  提交时间:2023/10/17
Fibroblast Activation Protein Targeting Probe with Gly-Pro Sequence for PET of Glioblastoma 期刊论文  OAI收割
MOLECULAR PHARMACEUTICS, 2023, 卷号: 20, 期号: 8, 页码: 4120-4128
作者:  
Lai, Chaoquan;  Cao, Rui;  Li, Renda;  He, Chunfeng;  Wang, Xiao
  |  收藏  |  浏览/下载:19/0  |  提交时间:2023/10/17