中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [8]
兰州化学物理研究所 [2]
金属研究所 [1]
新疆理化技术研究所 [1]
合肥物质科学研究院 [1]
采集方式
OAI收割 [13]
内容类型
期刊论文 [13]
发表日期
2020 [13]
学科主题
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发表日期:2020
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DW14383 is an irreversible pan-FGFR inhibitor that suppresses FGFR-dependent tumor growth in vitro and in vivo
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 9
作者:
Dai, Meng-di
;
Wang, Yue-liang
;
Fan, Jun
;
Dai, Yang
;
Ji, Yin-chun
  |  
收藏
  |  
浏览/下载:66/0
  |  
提交时间:2021/05/24
receptor tyrosine kinase
FGFR inhibitor
DW14383
antitumor activity
Design, synthesis and anti-tumor activities of carbamate derivatives of cinobufagin
期刊论文
OAI收割
STEROIDS, 2020, 卷号: 164, 页码: 11
作者:
Zhou, Yang
;
Hou, Jinjun
;
Long, Huali
;
Zhang, Zijia
;
Lei, Min
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2021/05/24
Cardiac glycosides
Cinobufagin
Natural product
Cytotoxicity
Antiproliferative activities
The dual HDAC-PI3K inhibitor CUDC-907 displays single-agent activity and synergizes with PARP inhibitor olaparib in small cell lung cancer
期刊论文
OAI收割
JOURNAL OF EXPERIMENTAL & CLINICAL CANCER RESEARCH, 2020, 卷号: 39
作者:
Ma, Liying
;
Bian, Xing
;
Lin, Wenchu
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2020/11/30
SCLC
PI3K
HDAC
CUDC-907
PARP1
Olaparib
DSB repair
Combination treatment
Rational Design and Evaluation of 6-(Pyrimidin-2-ylamino)-3,4-dihydroquinoxalin-2(1H)-ones as Polypharmacological Inhibitors of BET and Kinases
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 17, 页码: 9787-9802
作者:
Lv, Kaikai
;
Chen, Weicong
;
Chen, Danqi
;
Mou, Jie
;
Zhang, Huijie
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2020/12/21
Synthesis of oleandrin derivatives and their cytotoxic activity
期刊论文
OAI收割
STEROIDS, 2020, 卷号: 159, 页码: 7
作者:
Zhang, Yanzhi
;
Chen, Xubing
;
Zhou, Yang
;
Hou, Jinjun
;
Long, Huali
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2020/12/24
Cardiac glycosides
Oleandrin (OL)
Natural product
OL-4 '-yl ester
Cytotoxicity
Bungsteroid A: One Unusual C 34 Pentacyclic Steroid Analogue from Zanthoxylum bungeanum Maxim
期刊论文
OAI收割
the Journal of Organic Chemistry, 2020, 卷号: 85, 期号: 16, 页码: 10806−10812
作者:
Meng XH(孟宪华)
;
Chai T(柴甜)
;
Shi YP(师彦平)
;
Yang JL(杨军丽)
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2020/11/16
Zanthoxylum bungeanum Maxim
quantum-chemical 13C NMR
ECD
antiproliferative effect
steroid
Design, synthesis and antiproliferative activity evaluation of a series of pyrrolo [2,1-f] [1,2,4] triazine derivatives
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 卷号: 30, 期号: 12, 页码: 4
作者:
Xiang, Hao-Yue
;
Chen, Yan-Hong
;
Wang, Yi
;
Zhang, Xi
;
Ding, Jian
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2020/07/01
Antiproliferative
Cancer
Therapy
PI3K inhibitors
Pyrrolo [2,1-f][1,2,4] triazine
Kinase
Design and synthesis of new lenalidomide analogs via Suzuki cross-coupling reaction
期刊论文
OAI收割
ARCHIV DER PHARMAZIE, 2020, 页码: 10
作者:
Xiao, Donghuai
;
Wang, Yu-jie
;
Wang, Han-lin
;
Zhou, Yu-bo
;
Li, Jia
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2020/07/01
antitumor
arylboronic acid
lenalidomide
Suzuki cross-coupling
Co-Prodrugs of 7-Ethyl-10-hydroxycamptothecin and Vorinostat with in Vitro Hydrolysis and Anticancer Effects
期刊论文
OAI收割
ACS OMEGA, 2020, 卷号: 5, 期号: 1, 页码: 350-357
作者:
Liu, Shuangxi
;
Hu, Zonglong
;
Zhang, Qiumeng
;
Zhu, Qiwen
;
Chen, Yi
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2020/07/01
Antiproliferative abietane quinone diterpenoids from the roots of Salvia deserta
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2020, 卷号: 104, 期号: 11, 页码: 1-12
作者:
Zheng, XF (Zheng, Xiaofeng)[ 1 ]
;
Kadir, A (Kadir, Abdukriem)[ 1,2 ]
;
Zheng, GJ (Zheng, Guijuan)[ 1 ]
;
Jin, PF (Jin, Pengfei)[ 1 ]
;
Qin, DM (Qin, Dongmei)[ 3 ]
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2021/01/05
Salvia deserta Schang (Lamiaceae)
Abietane quinone diterpenoids
Calculated C-13 NMR-DP4+analysis
Mo-2(OAc)(4)-induced ECD
Antiproliferative activity