中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 2021 [21]
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Structure-Based Design of Dual-Acting Compounds Targeting Adenosine A(2A) Receptor and Histone Deacetylase as Novel Tumor Immunotherapeutic Agents 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 22, 页码: 16573-16597
作者:  
Yan, Wenzhong;  Ling, Lijun;  Wu, Yiran;  Yang, Kexin;  Liu, Ruiquan
  |  收藏  |  浏览/下载:16/0  |  提交时间:2022/06/15
The Novel RET Inhibitor SYHA1815 Inhibits RET-Driven Cancers and Overcomes Gatekeeper Mutations by Inducing G1 Cell-Cycle Arrest through c-Myc Downregulation 期刊论文  OAI收割
MOLECULAR CANCER THERAPEUTICS, 2021, 卷号: 20, 期号: 11, 页码: 2198-2206
作者:  
Jiang, Yuchen;  Peng, Xia;  Ji, Yinchun;  Dai, Yang;  Fang, Yanfen
  |  收藏  |  浏览/下载:34/0  |  提交时间:2021/12/16
Discovery and Development of a Potent, Selective, and Orally Bioavailable CHK1 Inhibitor Candidate: 5-((4-((3-Amino-3-methylbutyl)amino)-5-(trifluoromethyl)pyrimidin-2-yl)amino)picolinonitrile 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 20, 页码: 15069-15090
作者:  
Jin, Tingting;  Xu, Lei;  Wang, Peipei;  Hu, Xiaobei;  Zhang, Runyuan
  |  收藏  |  浏览/下载:27/0  |  提交时间:2022/01/04
Discovery and structure - activity relationship exploration of pyrazolo [1,5-a]pyrimidine derivatives as potent FLT3-ITD inhibitors 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 48, 页码: 13
作者:  
Chen, Yun;  Bai, Gang;  Li, Yan;  Ning, Yi;  Cao, Sufen
  |  收藏  |  浏览/下载:57/0  |  提交时间:2021/12/01
Rational Design and Development of Novel CDK9 Inhibitors for the Treatment of Acute Myeloid Leukemia 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 19, 页码: 14647-14663
作者:  
Han, Xu;  Song, Ning;  Saidahmatov, Abdusaid;  Wang, Peipei;  Wang, Yong
  |  收藏  |  浏览/下载:58/0  |  提交时间:2021/12/16
Myelocytomatosis-Protein Arginine N-Methyltransferase 5 Axis Defines the Tumorigenesis and Immune Response in Hepatocellular Carcinoma 期刊论文  OAI收割
HEPATOLOGY, 2021, 卷号: 74, 期号: 4, 页码: 1932-1951
作者:  
Luo, Yuhong;  Gao, Yuqing;  Liu, Weiwei;  Yang, Yuan;  Jiang, Jie
  |  收藏  |  浏览/下载:9/0  |  提交时间:2024/03/21
Clerodenoids A-F: C-ring Aromatized and/or Rearranged Abietane Diterpenoids from Clerodendrum chinense var. simplex 期刊论文  OAI收割
CHINESE JOURNAL OF CHEMISTRY, 2021, 页码: 7
作者:  
Qi, Jingjing;  Zhang, Yan;  Liu, Qunfang
  |  收藏  |  浏览/下载:27/0  |  提交时间:2021/08/17
In vitro studies of deferasirox derivatives as potential organelle-targeting traceable anti-cancer therapeutics 期刊论文  OAI收割
CHEMICAL COMMUNICATIONS, 2021, 页码: 4
作者:  
  |  收藏  |  浏览/下载:28/0  |  提交时间:2021/06/11
飞龙掌血化学成分及细胞毒活性研究 学位论文  OAI收割
2021
作者:  
陈姗姗
  |  收藏  |  浏览/下载:10/0  |  提交时间:2024/03/20
Rational drug design of benzothiazole-based derivatives as potent signal transducer and activator of transcription 3 (STAT3) signaling pathway inhibitors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 216, 页码: 20
作者:  
Gao, Dingding;  Jin, Nan;  Fu, Yixian;  Zhu, Yueyue;  Wang, Yujie
  |  收藏  |  浏览/下载:33/0  |  提交时间:2021/06/11