中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [22]
生态环境研究中心 [2]
合肥物质科学研究院 [2]
地理科学与资源研究所 [1]
计算技术研究所 [1]
西双版纳热带植物园 [1]
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采集方式
OAI收割 [34]
内容类型
期刊论文 [34]
发表日期
2022 [34]
学科主题
Biotechnol... [1]
Cell Biolo... [1]
Genetics &... [1]
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浏览/检索结果:
共34条,第1-10条
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发表日期:2022
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Optimized Synthesis of a Key Intermediate of Nirmatrelvir
期刊论文
OAI收割
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2022, 页码: 6
作者:
Qin, Hongjian
;
Jin, Chen
;
Odilov, Abdullajon
;
Bonku, Emmanuel Mintah
;
Zhu, Fuqiang
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/04/10
alpha-cyanomethylation
neodymium chloride
hydrogenation
one-pot
cyclic glutamine analog
Nirmatrelvir
In vitro and in vivo evaluation of the main protease inhibitor FB2001 against SARS-CoV-2
期刊论文
OAI收割
ANTIVIRAL RESEARCH, 2022, 卷号: 208, 页码: 10
作者:
Shang, Weijuan
;
Dai, Wenhao
;
Yao, Cheng
;
Xu, Ling
;
Tao, Xiangming
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2023/04/10
SARS-CoV-2
SARS-CoV-2 variants
FB2001
Main protease
PBPK
Anti-SARS-CoV-2 in vivo
Identification of Cysteine 270 as a Novel Site for Allosteric Modulators of SARS-CoV-2 Papain-Like Protease
期刊论文
OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2022, 页码: 10
作者:
Hu, Hangchen
;
Wang, Qian
;
Su, Haixia
;
Shao, Qiang
;
Zhao, Wenfeng
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/04/10
Allosteric Modulator
Cysteine 270
Drug Design
Papain-Like Protease
SARS-CoV-2
Anti-infective therapy using species-specific activators of Staphylococcus aureus ClpP
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2022, 卷号: 13, 期号: 1, 页码: 16
作者:
Wei, Bingyan
;
Zhang, Tao
;
Wang, Pengyu
;
Pan, Yihui
;
Li, Jiahui
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2023/04/10
Metagenomic analysis reveals the microbial degradation mechanism during kitchen waste biodrying
期刊论文
OAI收割
CHEMOSPHERE, 2022, 卷号: 307, 页码: 10
作者:
Cai, Lu
;
Guo, Han-Tong
;
Zheng, Guo-Di
;
Wang, Xin-Yu
;
Wang, Kan
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2022/09/26
Kitchen waste biodrying
Metagenomic
Functional microorganisms
Organic matter degradation
Metabolic functions
Structure-based design of a novel inhibitor of the ZIKA virus NS2B/ NS3 protease
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2022, 卷号: 128, 页码: 7
作者:
Xiong, Yanchao
;
Cheng, Fei
;
Zhang, Junyi
;
Su, Haixia
;
Hu, Hangchen
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2022/11/11
Zika virus
Fragment -based hit screening
Protein -inhibitor interactions
NS2B
NS3 protease
Crystal structure
A designed antimicrobial peptide with potential ability against methicillin resistant Staphylococcus aureus
期刊论文
OAI收割
FRONTIERS IN MICROBIOLOGY, 2022, 卷号: 13
作者:
Yuan, Bingqian
;
Lu, Xiaoyu
;
Yang, Min
;
He, Qiyi
;
Cha, Zhuocen
  |  
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2022/12/23
Staphylococcus aureus
cathelicidin
antimicrobial peptides
GW18
drug-resistant
Discovery of potent ebola entry inhibitors with (3S,4aS,8aS)-2-(3-amino-2-hydroxypropyl) decahydroisoquinoline-3-carboxamide scaffold
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 240, 页码: 12
作者:
Han, Sheng
;
Li, Heng
;
Chen, Weixiong
;
Yang, Li
;
Tong, Xiankun
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2022/11/11
Ebola virus
Entry inhibitor
Structural optimization
Aberrant human ClpP activation disturbs mitochondrial proteome homeostasis to suppress pancreatic ductal adenocarcinoma
期刊论文
OAI收割
CELL CHEMICAL BIOLOGY, 2022, 卷号: 29, 期号: 9, 页码: 1396-+
作者:
Wang, Pengyu
;
Zhang, Tao
;
Wang, Xinjing
;
Xiao, Hongying
;
Li, Huiti
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2022/12/13
Artemisinin analog SM934 alleviates epithelial barrier dysfunction via inhibiting apoptosis and caspase-1-mediated pyroptosis in experimental colitis
期刊论文
OAI收割
FRONTIERS IN PHARMACOLOGY, 2022, 卷号: 13, 页码: 18
作者:
Shao, Meijuan
;
Yan, Yuxi
;
Zhu, Fenghua
;
Yang, Xiaoqian
;
Qi, Qing
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2022/11/11
SM934
colitis
intestinal epithelial barrier
apoptosis
pyroptosis
NLRP3/caspase-1/GSDMD
MAPK/NF-kB