中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [9]
采集方式
OAI收割 [9]
内容类型
期刊论文 [9]
发表日期
2023 [4]
2022 [3]
2021 [2]
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An efficient synthesis of the last step key intermediate for telmisartan via Pd-catalyzed carbonylative cyclization
期刊论文
OAI收割
TETRAHEDRON, 2023, 卷号: 148, 页码: 8
作者:
Odilov, Abdullajon
;
Qin, Hongjian
;
Bonku, Emmanuel Mintah
;
Zhu, Fuqiang
;
Yang, Feipu
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2023/12/19
Telmisartan
Benzimidazole
Pd-catalyzed
Carbonylative/cyclization
Optimized Synthesis of the Key Intermediate of Telmisartan via the Cyclization of 2-Bromoarylamine with
n
-Butyronitrile
期刊论文
OAI收割
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2023, 卷号: 27, 期号: 11, 页码: 2165-2173
作者:
Qin, Hongjian
;
Mintah Bonku, Emmanuel
;
Odilov, Abdullajon
;
Wu, Mingjun
;
Liu, Yongjian
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2024/02/27
bis-benzimidazole
cyclization
2-bromoarylamine
n-butyronitrile
telmisartan
design of experiments
Efficient Large-Scale Process for Tecovirimat via Reactive Distillation for the Preparation of Cycloheptatriene
期刊论文
OAI收割
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2023, 页码: 8
作者:
Bonku, Emmanuel Mintah
;
Qin, Hongjian
;
Odilov, Abdullajon
;
Yang, Feipu
;
Xing, Xinglong
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2023/12/08
tecovirimat
monkeypox
cycloheptatriene
antiviral drug
reactive distillation
Pharmacokinetics,mass balance,and metabolism of 14C TPN171,a novel PDE5 inhibitor,in humans for the treatment of pulmonary arterial hypertension
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 卷号: 44, 期号: 1, 页码: 221
作者:
He Yifei
;
Liu Yin
;
Yu Jinghua
;
Cheng Huan
;
Odilov Abdullajon
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2023/05/22
TPN171
14CTPN171
PDE5 inhibitor
pulmonary arterial hypertension
healthy volunteers
pharmacokinetics
metabolite identification
mass balance
Optimized Synthesis of a Key Intermediate of Nirmatrelvir
期刊论文
OAI收割
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2022, 页码: 6
作者:
Qin, Hongjian
;
Jin, Chen
;
Odilov, Abdullajon
;
Bonku, Emmanuel Mintah
;
Zhu, Fuqiang
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/04/10
alpha-cyanomethylation
neodymium chloride
hydrogenation
one-pot
cyclic glutamine analog
Nirmatrelvir
Facile Synthesis of Benzimidazoles via N-Arylamidoxime Cyclization
期刊论文
OAI收割
ACS OMEGA, 2022, 页码: 10
作者:
Qin, Hongjian
;
Odilov, Abdullajon
;
Bonku, Emmanuel Mintah
;
Zhu, Fuqiang
;
Hu, Tianwen
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2023/04/10
Pharmacokinetics, mass balance, and metabolism of [C-14]TPN171, a novel PDE5 inhibitor, in humans for the treatment of pulmonary arterial hypertension
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2022, 页码: 13
作者:
He, Yi-fei
;
Liu, Yin
;
Yu, Jing-hua
;
Cheng, Huan
;
Odilov, Abdullajon
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2022/08/16
TPN171
[C-14]TPN171
PDE5 inhibitor
pulmonary arterial hypertension
healthy volunteers
pharmacokinetics
metabolite identification
mass balance
Facile and Cost-Effective Route for the Synthesis of Simmerafil
期刊论文
OAI收割
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2021, 卷号: 25, 期号: 11, 页码: 2432-2437
作者:
Odilov, Abdullajon
;
Liu, Yin
;
Hu, Tianwen
;
Jiang, Xiangrui
;
Suo, Jin
  |  
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2022/01/18
simmerafil
PDE5 inhibitor
salicylamide
synthesis
Scalable Process for Making 5,7-Dichlorotetrahydroisoquinoline-6-carboxylic Acid Using Methylene as the Protecting Group
期刊论文
OAI收割
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2021, 卷号: 25, 期号: 11, 页码: 2447-2452
作者:
Xu, Wanbin
;
Gong, Xudong
;
Odilov, Abdullajon
;
Hu, Tianwen
;
Jiang, Xiangrui
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2022/01/18
5,7-dichlorotetrahydroisoquinoline-6-carboxylic acid
lifitegrast
methylene
atom utilization