中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [768]
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OAI收割 [768]
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期刊论文 [758]
会议论文 [9]
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Ent-labdane-type diterpene glycosides obtained from
Rubus
chingii
Hu and their inhibitory effects on PDE5A activity
期刊论文
OAI收割
FITOTERAPIA, 2024, 卷号: 173, 页码: 14
作者:
Yu, Jun-dong
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/02/27
diterpene glycosides
Rubus Chingii Hu
PDE5A inhibitory activity
ent-labdane
Discovery of GPX4 inhibitors through FP-based high-throughput screening
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 14
作者:
Cao, Yu
;
Wu, Bin
;
Xu, Ying
;
Wang, Mingchen
;
Wu, Xinyu
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2024/02/27
GPX4 inhibitor
HTS assay
Ferroptosis
Fluorescence polarization
Blocking tumor-platelet crosstalk to prevent tumor metastasis via reprograming glycolysis using biomimetic membrane-hybridized liposomes
期刊论文
OAI收割
JOURNAL OF CONTROLLED RELEASE, 2024, 卷号: 366, 页码: 328-341
作者:
Zhu, Jie
;
Wang, Rui
;
Yang, Chenxiao
;
Shao, Xinyue
;
Zhang, Yi
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2024/03/06
Platelet
Circulating tumor cells (CTCs)
Glycolysis
Metastasis
Hybrid-membrane liposome
Quercetin
Shikonin
Effects of aqueous extracts and volatile oils prepared from Huaxiang Anshen decoction on
p
-chlorophenylalanine-induced insomnia mice
期刊论文
OAI收割
JOURNAL OF ETHNOPHARMACOLOGY, 2024, 卷号: 319, 页码: 11
作者:
Li, Xinye
;
He, Chao
;
Shen, Min
;
Wang, Mingyun
;
Zhou, Jingwen
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2024/01/16
Huaxiang Anshen Decoction
Volatile oil
Sedative and hypnotic effects
beta-cyclodextrin inclusion complex
Stereoconvergent and Chemoenzymatic Synthesis of Tumor-Associated Glycolipid Disialosyl Globopentaosylceramide for Probing the Binding Affinity of Siglec-7
期刊论文
OAI收割
ACS CENTRAL SCIENCE, 2024, 卷号: 10, 期号: 2, 页码: 417-425
作者:
Liu, Yating
;
Yan, Mengkun
;
Wang, Minghui
;
Luo, Shiwei
;
Wang, Shasha
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2024/03/25
Design and synthesis of cantharidin derivative DCZ5418 as a TRIP13 inhibitor with anti-multiple myeloma activity
in
vitro
and
in
vivo
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 98, 页码: 7
作者:
Dong, Sanfeng
;
Hu, Ke
;
Shi, Yulong
;
Wang, Guanli
;
Yu, Dandan
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2024/02/19
Multiple myeloma
TRIP13 inhibitor
Cantharidin
DCZ5418
DCZ0415
Structure-Guided Design, Synthesis, and Antivirulence Assessment of Covalent
Staphylococcus aureus
Sortase A Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 2, 页码: 1127-1146
作者:
Yue, Chuan
;
Yuan, Ziqi
;
Xu, Guobin
;
Guan, Xiang-Na
;
Wei, Bingyan
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2024/02/27
The enzyme activity of sortase A is regulated by phosphorylation in Staphylococcus aureus
期刊论文
OAI收割
VIRULENCE, 2023, 卷号: 14, 期号: 1, 页码: 2171641
作者:
Chen, Feifei
;
Di, Hongxia
;
Wang, Yanhui
;
Peng, Chao
;
Chen, Rongrong
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2024/03/27
Staphylococcus aureus
Sortase A
protein phosphorylation
virulence
Discovery of Dual Function Agents That Exhibit Anticancer Activity via Catastrophic Nicotinamide Adenine Dinucleotide Depletion
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 24, 页码: 16694-16703
作者:
Fu, Yixian
;
Huang, Yahui
;
Zhou, Chenchen
;
Li, Xinge
;
Dong, Guoqiang
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2024/01/26
Discovery of 5-trifluoromethyl-2-aminopyrimidine derivatives as potent dual inhibitors of FLT3 and CHK1
期刊论文
OAI收割
RSC MEDICINAL CHEMISTRY, 2023, 页码: 14
作者:
Deng, Minjie
;
Gao, Yue
;
Wang, Peipei
;
Du, Wenjing
;
Xu, Gaoya
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/02/19