中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 上海药物研究所 [7]
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A viral RNA-dependent RNA polymerase inhibitor VV116 broadly inhibits human coronaviruses and has synergistic potency with 3CLpro inhibitor nirmatrelvir 期刊论文  OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2023, 卷号: 8, 期号: 1, 页码: 10
作者:  
Zhang, Yumin;  Sun, Yuan;  Xie, Yuanchao;  Shang, Weijuan;  Wang, Zhen
  |  收藏  |  浏览/下载:6/0  |  提交时间:2023/12/08
Design, synthesis and biological evaluation of peptidomimetic benzothiazolyl ketones as 3CLpro inhibitors against SARS-CoV-2 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 257, 页码: 13
作者:  
Yang, Hanxi;  You, Mengyuan;  Shu, Xiaoyang;  Zhen, Jingyao;  Zhu, Mengwei
  |  收藏  |  浏览/下载:13/0  |  提交时间:2023/10/17
Discovery of novel non-peptidic and non-covalent small-molecule 3CL(pro) inhibitors as potential candidate for COVID-19 treatment 期刊论文  OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2023, 卷号: 8, 期号: 1, 页码: 4
作者:  
Jiang, Zhidong;  Feng, Bo;  Zhang, Yumin;  Nie, Tianqing;  Liu, Hong
  |  收藏  |  浏览/下载:9/0  |  提交时间:2023/10/17
Synthesis and anti-SARS-CoV-2 activity of deuterated GS-441524 analogs 期刊论文  OAI收割
TETRAHEDRON LETTERS, 2022, 卷号: 104, 页码: 9
作者:  
Zheng, Wei;  Hu, Tianwen;  Zhang, Yumin;  Wei, Daibao;  Xie, Yuanchao
  |  收藏  |  浏览/下载:17/0  |  提交时间:2022/11/11
Oral remdesivir derivative VV116 is a potent inhibitor of respiratory syncytial virus with efficacy in mouse model 期刊论文  OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2022, 卷号: 7, 期号: 1, 页码: 3
作者:  
Zhang, Ruxue;  Zhang, Yumin;  Zheng, Wei;  Shang, Weijuan;  Wu, Yan
  |  收藏  |  浏览/下载:23/0  |  提交时间:2022/06/15
Design and development of an oral remdesivir derivative VV116 against SARS-CoV-2 期刊论文  OAI收割
CELL RESEARCH, 2021, 页码: 3
作者:  
Xie, Yuanchao;  Yin, Wanchao;  Zhang, Yumin;  Shang, Weijuan;  Wang, Zhen
  |  收藏  |  浏览/下载:73/0  |  提交时间:2021/11/04
Identification of pyrogallol as a warhead in design of covalent inhibitors for the SARS-CoV-2 3CL protease 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2021, 卷号: 12, 期号: 1, 页码: 12
作者:  
Su, Haixia;  Yao, Sheng;  Zhao, Wenfeng;  Zhang, Yumin;  Liu, Jia
  |  收藏  |  浏览/下载:57/0  |  提交时间:2021/08/17