中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [45]
采集方式
OAI收割 [45]
内容类型
期刊论文 [45]
发表日期
2024 [1]
2020 [3]
2019 [3]
2018 [7]
2017 [10]
2016 [2]
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专题:上海药物研究所
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Structure-Guided Design, Synthesis, and Antivirulence Assessment of Covalent
Staphylococcus aureus
Sortase A Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 2, 页码: 1127-1146
作者:
Yue, Chuan
;
Yuan, Ziqi
;
Xu, Guobin
;
Guan, Xiang-Na
;
Wei, Bingyan
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2024/02/27
BRD4 as a therapeutic target for nonfunctioning and growth hormone pituitary adenoma
期刊论文
OAI收割
NEURO-ONCOLOGY, 2020, 卷号: 22, 期号: 8, 页码: 1114-1125
作者:
Shi, Chengzhang
;
Ye, Zhao
;
Han, Jie
;
Ye, Xiaoqing
;
Lu, Wenchao
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2024/03/21
High-throughput screening campaign identifies a small molecule agonist of the relaxin family peptide receptor 4
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 9
作者:
Lin, Guang-yao
;
Lin, Lin
;
Cai, Xiao-qing
;
Dai, An-tao
;
Zhu, Yue
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2020/07/01
RXFP4
INSL5
high-throughput screening
agonist
JK1
A Novel G Protein-Biased and Subtype-Selective Agonist for a G Protein-Coupled Receptor Discovered from Screening Herbal Extracts
期刊论文
OAI收割
ACS CENTRAL SCIENCE, 2020, 卷号: 6, 期号: 2, 页码: 213-225
作者:
Zhang, Bingjie
;
Zhao, Simeng
;
Yang, Dehua
;
Wu, Yiran
;
Xin, Ye
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2020/07/01
Tetramerized Sesquiterpenoid Ainsliatetramers A and B from Ainsliaea fragrans and Their Cytotoxic Activities
期刊论文
OAI收割
ORGANIC LETTERS, 2019, 卷号: 21, 期号: 20, 页码: 8211-8214
作者:
Zhang, Rui
;
Tang, Chunping
;
Liu, Hong-Chun
;
Ren, Yongmei
;
Ke, Chang-Qiang
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2020/07/01
17-nor-Cephalotane-Type Diterpenoids from Cephalotaxus fortunei
期刊论文
OAI收割
JOURNAL OF NATURAL PRODUCTS, 2019, 卷号: 82, 期号: 6, 页码: 1565-1575
作者:
Ge, Zhan-Peng
;
Liu, Hong-Chun
;
Wang, Guo-Cai
;
Liu, Qun-Fang
;
Xu, Cheng-Hui
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2020/07/01
Structure and dynamics of the active human parathyroid hormone receptor-1
期刊论文
OAI收割
SCIENCE, 2019, 卷号: 364, 期号: 6436, 页码: 148-+
作者:
Zhao, Li-Hua
;
Ma, Shanshan
;
Sutkeviciute, Ieva
;
Shen, Dan-Dan
;
Zhou, X. Edward
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2020/07/01
From hit to lead: Structure-based discovery of naphthalene-1 sulfonamide derivatives as potent and selective inhibitors of fatty acid binding protein 4
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 154, 页码: 44-59
作者:
Gao, Ding-Ding
;
Dou, Hui-Xia
;
Su, Hai-Xia
;
Zhang, Ming-Ming
;
Wang, Ting
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2019/01/08
FABP4 inhibitors
FABP3 sparing
Structure-based design strategy
X-ray crystallography
The synthesis and antistaphylococcal activity of N-sulfonaminoethyloxime derivatives of dehydroabietic acid
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2018, 卷号: 28, 期号: 10, 页码: 1943-1948
作者:
Zhang, Wen-Ming
;
Yao, Yang
;
Yang, Teng
;
Wang, Xue-Ying
;
Zhu, Zhen-Yun
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2019/01/08
Antistaphylococcal
Multidrug-resistant
Synthesis
Oxime
Dehydroabietic acid
Exploring lipid markers of the quality of coix seeds with different geographical origins using supercritical fluid chromatography mass spectrometry and chemometrics
期刊论文
OAI收割
PHYTOMEDICINE, 2018, 卷号: 45, 页码: 1-7
作者:
Hou, Jin-Jun
;
Cao, Chun-Mei
;
Xu, Yong-wei
;
Yao, Shuai
;
Cai, Lu-Ying
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2019/01/08
Quality marker
Coicis semen
Triglyceride
Diglyceride
Ultra-performance convergence chromatography
Quadrupole/time-of-flight hybrid mass spectrometry