中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [97]
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Design, Synthesis, and Anti-tuberculosis Activity of Streptomycin Derivatives
期刊论文
OAI收割
LETTERS IN DRUG DESIGN & DISCOVERY, 2024, 卷号: 21, 期号: 4, 页码: 738-748
作者:
Zhang, Yinyong
;
Zhao, Wenhao
;
Yang, Yushe
;
Zhou, Xianli
;
Guo, Bin
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2024/03/06
Multidrug-resistant
hydrazine
hydrazide
sulfonyl hydrazide
siderophore
synthesis
anti-tuberculosis activity
A facile and selective derivatization approach on kynurenine-NH2 in daptomycin, leading to the discovery of hexakynomycin to combat multidrug-resistant Gram-positive pathogens especially daptomycin-resistant bacteria
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 259, 页码: 14
作者:
Guan, Dongliang
;
Li, Jian
;
Chen, Feifei
;
Li, Jiaqi
;
Bian, Xiaolei
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2023/10/17
Lipopeptide
Daptomycin derivatives
Multidrug-resistant bacteria
Kynurenine
Hexakynomycin
Resin glycosides from Merremia hederacea with multidrug-resistant reversal activities
期刊论文
OAI收割
PHYTOCHEMISTRY LETTERS, 2023, 卷号: 54, 页码: 14-17
作者:
Li, Chen-Yue
;
Fang, Jie
;
Li, Guang-Yao
;
Wang, Wen-Qiong
;
Xuan, Li-Jiang
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2023/10/17
Merremia hederacea
Resin glycoside
Multidrug-resistant reversal activity
Efficient Kilogram-Scale Synthesis of a Novel Oxazolidinone Antibacterial Candidate YG-056SP
期刊论文
OAI收割
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2023, 页码: 12
作者:
Zhang, Yinyong
;
Yang, Yushe
;
Meng, Xin
;
Zhou, Xianli
;
Guo, Bin
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2023/04/10
oxazolidinone
asymmetric reduction
fused ring
process development
crystal transformation
Anti-infective therapy using species-specific activators of Staphylococcus aureus ClpP
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2022, 卷号: 13, 期号: 1, 页码: 16
作者:
Wei, Bingyan
;
Zhang, Tao
;
Wang, Pengyu
;
Pan, Yihui
;
Li, Jiahui
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2023/04/10
Drug Degradation Caused by mce3R Mutations Confers Contezolid (MRX-I) Resistance in Mycobacterium tuberculosis
期刊论文
OAI收割
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 2022, 卷号: 66, 期号: 10, 页码: 11
作者:
Pi, Rui
;
Chen, Xiaomin
;
Meng, Jian
;
Liu, Qingyun
;
Chen, Yiwang
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2022/11/11
Mycobacterium tuberculosis
drug resistance
contezolid
Mce3R
Rv1936
degradation
drug resistance mechanisms
Potentiation of Vancomycin: Creating Cooperative Membrane Lysis through a "Derivatization-for-Sensitization" Approach
期刊论文
OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2022, 卷号: 144, 期号: 23, 页码: 10622-10639
作者:
Lei, E.
;
Tao, Huanyu
;
Jiao, Shang
;
Yang, Anming
;
Zhou, Yu
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2022/08/16
Novel niclosamide-derived adjuvants elevating the efficacy of polymyxin B against MDR Pseudomonas aeruginosa DK2
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 236, 页码: 114318
作者:
Lu, Taotao
;
Zheng, Xinyu
;
Mao, Fei
;
Cao, Qiao
;
Cao, Qin
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/03/21
Pseudomonas aeruginosa DK2
Polymyxin B
Niclosamide
Adjuvants
Drug repurposing
A Short Peptide of Autotransporter Ata Is a Promising Protective Antigen for Vaccination Against Acinetobacter baumannii
期刊论文
OAI收割
FRONTIERS IN IMMUNOLOGY, 2022, 卷号: 13, 页码: 12
作者:
Sun, Peng
;
Li, Xin
;
Pan, Chao
;
Liu, Zhicheng
;
Wu, Jun
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2023/02/24
Acinetobacter baumannii
acinetobacter trimeric autotransporter adhesin (Ata)
CpG
CTB
subunit vaccine
Diverse antibiotic resistance genes and potential pathogens inhabit in the phyllosphere of fresh vegetables
期刊论文
OAI收割
SCIENCE OF THE TOTAL ENVIRONMENT, 2022, 卷号: 815, 期号: 0, 页码: 152851
作者:
Yin, Yue
;
Zhu, Dong
;
Yang, Guang
;
Su, Jianqiang
;
Duan, Guilan
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2022/11/07
ESCHERICHIA-COLI
IRRIGATION WATER
CROSS-CONTAMINATION
SALMONELLA
BACTERIA
PRODUCE
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COMMUNITIES
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