中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 上海药物研究所 [42]
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Optimization of Brigatinib as New Wild-Type Sparing Inhibitors of EGFR(T790M/C797S) Mutants 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2022, 页码: 7
作者:  
Li, Shan;  Zhang, Tao;  Zhu, Su-Jie;  Lei, Chong;  Lai, Mengzhen
  |  收藏  |  浏览/下载:25/0  |  提交时间:2022/06/15
Constitutive signal bias mediated by the human GHRHR splice variant 1 期刊论文  OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2021, 卷号: 118, 期号: 40, 页码: 10
作者:  
Cong, Zhaotong;  Zhou, Fulai;  Zhang, Chao;  Zou, Xinyu;  Zhang, Huibing
  |  收藏  |  浏览/下载:57/0  |  提交时间:2021/12/01
Myelocytomatosis-Protein Arginine N-Methyltransferase 5 Axis Defines the Tumorigenesis and Immune Response in Hepatocellular Carcinoma 期刊论文  OAI收割
HEPATOLOGY, 2021, 卷号: 74, 期号: 4, 页码: 1932-1951
作者:  
Luo, Yuhong;  Gao, Yuqing;  Liu, Weiwei;  Yang, Yuan;  Jiang, Jie
  |  收藏  |  浏览/下载:9/0  |  提交时间:2024/03/21
Discovery of Cyclic Peptidomimetic Ligands Targeting the Extracellular Domain of EGFR 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 15, 页码: 11219-11228
作者:  
Zheng, Mengmeng;  Li, Chunpu;  Zhou, Mi
  |  收藏  |  浏览/下载:51/0  |  提交时间:2021/11/04
Intestinal MYC modulates obesity-related metabolic dysfunction 期刊论文  OAI收割
NATURE METABOLISM, 2021, 页码: 37
作者:  
Luo, Yuhong;  Yang, Shoumei;  Wu, Xuan;  Takahashi, Shogo;  Sun, Lulu
  |  收藏  |  浏览/下载:28/0  |  提交时间:2021/08/17
Targeting p300/CBP Attenuates Hepatocellular Carcinoma Progression through Epigenetic Regulation of Metabolism 期刊论文  OAI收割
CANCER RESEARCH, 2021, 卷号: 81, 期号: 4, 页码: 860-872
作者:  
Cai, Ling-Yan;  Chen, Shi-Jie;  Xiao, Sen-Hao;  Sun, Qin-Juan;  Ding, Chen-Hong
  |  收藏  |  浏览/下载:19/0  |  提交时间:2024/03/21
Capsaicin derivatives with nitrothiophene substituents: Design, synthesis and antibacterial activity against multidrug-resistant S. aureus 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 198, 页码: 11
作者:  
Wang, Zhi-Cheng;  Wei, Bingyan;  Pei, Fang-Ning;  Yang, Teng;  Tang, Jie
  |  收藏  |  浏览/下载:42/0  |  提交时间:2020/12/24
2-Oxo-3,4-dihydropyrimido[4,5-d] pyrimidines as new reversible inhibitors of EGFR C797S (Cys797 to Ser797) mutant 期刊论文  OAI收割
CHINESE CHEMICAL LETTERS, 2020, 卷号: 31, 期号: 5, 页码: 1281-1287
作者:  
Hu, Xianglong;  Xun, Qiuju;  Zhang, Tao;  Zhu, Su-Jie;  Li, Qian
  |  收藏  |  浏览/下载:80/0  |  提交时间:2020/07/01
BRD4 as a therapeutic target for nonfunctioning and growth hormone pituitary adenoma 期刊论文  OAI收割
NEURO-ONCOLOGY, 2020, 卷号: 22, 期号: 8, 页码: 1114-1125
作者:  
Shi, Chengzhang;  Ye, Zhao;  Han, Jie;  Ye, Xiaoqing;  Lu, Wenchao
  |  收藏  |  浏览/下载:18/0  |  提交时间:2024/03/21
High-throughput screening campaign identifies a small molecule agonist of the relaxin family peptide receptor 4 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 9
作者:  
Lin, Guang-yao;  Lin, Lin;  Cai, Xiao-qing;  Dai, An-tao;  Zhu, Yue
  |  收藏  |  浏览/下载:23/0  |  提交时间:2020/07/01