中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [42]
采集方式
OAI收割 [42]
内容类型
期刊论文 [42]
发表日期
2022 [1]
2021 [5]
2020 [5]
2019 [5]
2018 [4]
2017 [5]
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专题:上海药物研究所
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Optimization of Brigatinib as New Wild-Type Sparing Inhibitors of EGFR(T790M/C797S) Mutants
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2022, 页码: 7
作者:
Li, Shan
;
Zhang, Tao
;
Zhu, Su-Jie
;
Lei, Chong
;
Lai, Mengzhen
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2022/06/15
Epidermal Growth Factor Receptor (EGFR)
Resistant Mutation
C797S
Antitumor
Constitutive signal bias mediated by the human GHRHR splice variant 1
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2021, 卷号: 118, 期号: 40, 页码: 10
作者:
Cong, Zhaotong
;
Zhou, Fulai
;
Zhang, Chao
;
Zou, Xinyu
;
Zhang, Huibing
  |  
收藏
  |  
浏览/下载:57/0
  |  
提交时间:2021/12/01
class B1 GPCR
receptor bias
cancer
cell proliferation
Myelocytomatosis-Protein Arginine N-Methyltransferase 5 Axis Defines the Tumorigenesis and Immune Response in Hepatocellular Carcinoma
期刊论文
OAI收割
HEPATOLOGY, 2021, 卷号: 74, 期号: 4, 页码: 1932-1951
作者:
Luo, Yuhong
;
Gao, Yuqing
;
Liu, Weiwei
;
Yang, Yuan
;
Jiang, Jie
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/03/21
Discovery of Cyclic Peptidomimetic Ligands Targeting the Extracellular Domain of EGFR
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 15, 页码: 11219-11228
作者:
Zheng, Mengmeng
;
Li, Chunpu
;
Zhou, Mi
  |  
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2021/11/04
Intestinal MYC modulates obesity-related metabolic dysfunction
期刊论文
OAI收割
NATURE METABOLISM, 2021, 页码: 37
作者:
Luo, Yuhong
;
Yang, Shoumei
;
Wu, Xuan
;
Takahashi, Shogo
;
Sun, Lulu
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2021/08/17
Targeting p300/CBP Attenuates Hepatocellular Carcinoma Progression through Epigenetic Regulation of Metabolism
期刊论文
OAI收割
CANCER RESEARCH, 2021, 卷号: 81, 期号: 4, 页码: 860-872
作者:
Cai, Ling-Yan
;
Chen, Shi-Jie
;
Xiao, Sen-Hao
;
Sun, Qin-Juan
;
Ding, Chen-Hong
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2024/03/21
Capsaicin derivatives with nitrothiophene substituents: Design, synthesis and antibacterial activity against multidrug-resistant S. aureus
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 198, 页码: 11
作者:
Wang, Zhi-Cheng
;
Wei, Bingyan
;
Pei, Fang-Ning
;
Yang, Teng
;
Tang, Jie
  |  
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2020/12/24
Capsaicin
Nitrothiophene
Multidrug-resistant S. aureus
Antibacterial agent
2-Oxo-3,4-dihydropyrimido[4,5-d] pyrimidines as new reversible inhibitors of EGFR C797S (Cys797 to Ser797) mutant
期刊论文
OAI收割
CHINESE CHEMICAL LETTERS, 2020, 卷号: 31, 期号: 5, 页码: 1281-1287
作者:
Hu, Xianglong
;
Xun, Qiuju
;
Zhang, Tao
;
Zhu, Su-Jie
;
Li, Qian
  |  
收藏
  |  
浏览/下载:80/0
  |  
提交时间:2020/07/01
EGFR(C797S) mutant
SARs
2-Oxo-3,4-dihydropyrimido[4,5-d] pyrimidine
Clinical resistance
Fourth-generation inhibitors
BRD4 as a therapeutic target for nonfunctioning and growth hormone pituitary adenoma
期刊论文
OAI收割
NEURO-ONCOLOGY, 2020, 卷号: 22, 期号: 8, 页码: 1114-1125
作者:
Shi, Chengzhang
;
Ye, Zhao
;
Han, Jie
;
Ye, Xiaoqing
;
Lu, Wenchao
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2024/03/21
High-throughput screening campaign identifies a small molecule agonist of the relaxin family peptide receptor 4
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 9
作者:
Lin, Guang-yao
;
Lin, Lin
;
Cai, Xiao-qing
;
Dai, An-tao
;
Zhu, Yue
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2020/07/01
RXFP4
INSL5
high-throughput screening
agonist
JK1