中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [18]
采集方式
OAI收割 [18]
内容类型
期刊论文 [16]
会议论文 [2]
发表日期
2023 [1]
2022 [3]
2021 [2]
2019 [2]
2018 [2]
2017 [3]
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专题:上海药物研究所
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Rational Design of RNA Demethylase FTO Inhibitors with Enhanced Antileukemia Drug-Like Properties
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 22
作者:
Xiao, Pan
;
Duan, Zongliang
;
Liu, Zeyu
;
Chen, Liang
;
Zhang, Deyan
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2023/10/17
Aberrant human ClpP activation disturbs mitochondrial proteome homeostasis to suppress pancreatic ductal adenocarcinoma
期刊论文
OAI收割
CELL CHEMICAL BIOLOGY, 2022, 卷号: 29, 期号: 9, 页码: 1396-+
作者:
Wang, Pengyu
;
Zhang, Tao
;
Wang, Xinjing
;
Xiao, Hongying
;
Li, Huiti
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2022/12/13
Dual-modified nanoparticles overcome sequential absorption barriers for oral insulin delivery
期刊论文
OAI收割
JOURNAL OF CONTROLLED RELEASE, 2022, 卷号: 342, 页码: 1-13
作者:
Xi, Ziyue
;
Ahmad, Ejaj
;
Zhang, Wei
;
Li, Jingyi
;
Wang, Aohua
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2022/06/15
Absorption barriers
Sequential delivery
Transcytosis
Intracellular trafficking
Insulin
Discovery of seneciobipyrrolidine derivatives for the amelioration of glucose homeostasis disorders through 4E-BP1/Akt/AMPK signaling activation
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 228, 页码: 25
作者:
Che, Jinxin
;
Ma, Canliang
;
Lu, Jialiang
;
Chen, Binhui
;
Shi, Qiuqiu
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2022/06/15
Seneciobipyrrolidine
Phenotypic screening
Glucose homeostasis
Proteomic analysis
L6 myotubes
4E-BP1
Twin drug design, synthesis and evaluation of diosgenin derivatives as multitargeted agents for the treatment of vascular dementia
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 37, 页码: 16
作者:
Yang, Gui-Xiang
;
Sun, Jia-Min
;
Zheng, Lu-Lu
;
Zhang, Li
;
Li, Jie
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2021/06/11
Vascular dementia
Diosgenin
Antioxidant
Anti-cholinesterase
Multi-target-directed ligands
Biscaesalmins A and B from Caesalpinia minax, highly oxidized dimeric cassane diterpenoids as interleukin-1 beta inhibitors
期刊论文
OAI收割
CHINESE CHEMICAL LETTERS, 2021, 卷号: 32, 期号: 4, 页码: 1475-1479
作者:
Xu, Yunshao
;
Zhang, Tian
;
Feng, Lu
;
Feng, Zheling
;
Zhang, Qingwen
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2021/08/17
Caesalpinia minax
IL-1 beta
Dimeric cassane diterpenoids
NLRP3
TD-DFT
Cancer Cell Membrane-Camouflaged Nanorods with Endoplasmic Reticulum Targeting for Improved Antitumor Therapy
期刊论文
OAI收割
ACS APPLIED MATERIALS & INTERFACES, 2019, 卷号: 11, 期号: 50, 页码: 46614-46625
作者:
Zhang, Wei
;
Yu, Miaorong
;
Xi, Ziyue
;
Nie, Di
;
Dai, Zhuo
  |  
收藏
  |  
浏览/下载:44/0
  |  
提交时间:2020/07/01
rod shape
endoplasmic reticulum-tatgeted
cancer cell membrane coating
intracellular trafficking
pancreatic tumor delivery
Lycodine-type alkaloids from Lycopodiastrum casuarinoides and their acetylcholinesterase inhibitory activity
期刊论文
OAI收割
FITOTERAPIA, 2019, 卷号: 139, 页码: 7
作者:
Feng, Zheling
;
Chen, Shixin
;
Wang, Wei
;
Feng, Lu
;
Dong, Yanyan
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2020/07/01
Lycopodiastrum casuarinoides
Lycopodiaceae
Lycodine-type alkaloids
TD-DFT
ECD
Characteristics of hERG and hNav1.5 channel blockade by sulcardine sulfate, a novel anti-arrhythmic compound
期刊论文
OAI收割
European journal of pharmacology, 2018, 卷号: 844, 页码: 130-138
作者:
Chen, Weihai
;
Gan, Lu
;
Wang, Yiping
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2019/01/08
Rapid transport of deformation-tuned nanoparticles across biological hydrogels and cellular barriers
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2018, 卷号: 9
作者:
Yu, Miaorong
;
Xu, Lu
;
Tian, Falin
;
Su, Qian
;
Zheng, Nan
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2019/01/08