中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [22]
采集方式
OAI收割 [22]
内容类型
期刊论文 [22]
发表日期
2024 [1]
2021 [3]
2020 [3]
2019 [3]
2018 [1]
2017 [1]
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Chemistry [2]
Biochemist... [1]
Pharmacolo... [1]
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共22条,第1-10条
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专题:上海药物研究所
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Development and Validation of an ADA-Tolerant Assay for Quantification of an Exatecan-Based ADC in Monkey Plasma
期刊论文
OAI收割
MOLECULES, 2024, 卷号: 29, 期号: 3, 页码: 14
作者:
Tao, Yimin
;
Lu, Wei
;
Gao, Jinli
;
Yang, Shuangshuang
;
Ruan, Chaoyi
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2024/03/13
antibody-drug conjugate (ADC)
bioanalysis
anti-drug antibody (ADA)
ligand binding assay (LBA)
ADA-tolerant assay
GADD45 beta stabilized by direct interaction with HSP72 ameliorates insulin resistance and lipid accumulation
期刊论文
OAI收割
PHARMACOLOGICAL RESEARCH, 2021, 卷号: 173, 页码: 11
作者:
Dong, Yunxia
;
Ma, Ningning
;
Fan, Lei
;
Yuan, Luyang
;
Wu, Qian
  |  
收藏
  |  
浏览/下载:69/0
  |  
提交时间:2021/12/16
Non-alcoholic fatty liver disease
GADD45 beta
HSP72
Lipid accumulation
Insulin resistance
Kinetics-Driven Drug Design Strategy for Next-Generation Acetylcholinesterase Inhibitors to Clinical Candidate
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 4, 页码: 1844-1855
作者:
Zhou, Yu
;
Fu, Yan
;
Yin, Wanchao
;
Li, Jian
;
Wang, Wei
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2021/05/24
miR-552-3p modulates transcriptional activities of FXR and LXR to ameliorate hepatic glycolipid metabolism disorder
期刊论文
OAI收割
JOURNAL OF HEPATOLOGY, 2021, 卷号: 74, 期号: 1, 页码: 8-19
作者:
Fan, Lei
;
Lai, Rongtao
;
Ma, Ningning
;
Dong, Yunxia
;
Li, Yu
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2021/05/24
miR-552-3p
Transcriptional gene regulation
Intranuclear miRNAs
Glycolipid metabolic disease
NR1 subfamily
Geng et al. reply
期刊论文
OAI收割
CELL RESEARCH, 2020, 页码: 1
作者:
Wang, Xinyi
;
Sun, Guangqiang
;
Feng, Teng
;
Zhang, Jing
;
Huang, Xun
  |  
收藏
  |  
浏览/下载:73/0
  |  
提交时间:2020/12/24
Structure-Activity Relationship of SPOP Inhibitors against Kidney Cancer
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 9, 页码: 4849-4866
作者:
Dong, Ze
;
Wang, Zhen
;
Guo, Zhong-Qiang
;
Gong, Shouzhe
;
Zhang, Tao
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2020/07/01
Repurposing antimycotic ciclopirox olamine as a promising anti-ischemic stroke agent
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2020, 卷号: 10, 期号: 3, 页码: 434-446
作者:
Feng, Hongxuan
;
Hu, Linghao
;
Zhu, Hongwen
;
Tao, Lingxue
;
Wu, Lei
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2020/07/01
Blood-brain barrier
Brain ischemia
Cell cycle
Inflammation
Neuroprotection
Sodium oligomannate therapeutically remodels gut microbiota and suppresses gut bacterial amino acids-shaped neuroinflammation to inhibit Alzheimer's disease progression
期刊论文
OAI收割
CELL RESEARCH, 2019, 卷号: 29, 期号: 10, 页码: 787-803
作者:
Wang, Xinyi
;
Sun, Guangqiang
;
Feng, Teng
;
Zhang, Jing
;
Huang, Xun
  |  
收藏
  |  
浏览/下载:83/0
  |  
提交时间:2020/07/01
Emerging Approaches of Cell-Based Nanosystems to Target Cancer Metastasis
期刊论文
OAI收割
ADVANCED FUNCTIONAL MATERIALS, 2019, 页码: 36
作者:
Gong, Xiang
;
Li, Jie
;
Tan, Tao
;
Wang, Zhiwan
;
Wang, Hong
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2020/07/01
cancer metastasis
cell membranes
nanosystems
tumor targeting
Optimization of P2Y(12) Antagonist Ethyl 6-(4-((Benzylsulfonyl)carbarnoyl)piperidin-1-yl)-5-cyano-2-methylnicotinate (AZD1283) Led to the Discovery of an Oral Antiplatelet Agent with Improved Druglike Properties
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 6, 页码: 3088-3106
作者:
Kong, Deyu
;
Xue, Tao
;
Guo, Bin
;
Cheng, Jianjun
;
Liu, Shunyin
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2020/07/01