中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [59]
采集方式
OAI收割 [59]
内容类型
期刊论文 [59]
发表日期
2023 [6]
2022 [7]
2020 [2]
2019 [4]
2018 [11]
2017 [2]
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专题:上海药物研究所
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Discovery of a novel GPR35 agonist with high and equipotent species potency for oral treatment of IBD
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2023, 卷号: 96, 页码: 12
作者:
Song, Zhaoxiang
;
Lu, Dan
;
Sun, Jun
;
Ye, Yangliang
;
Fang, Jiahui
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2024/01/16
GPR35
IBD
Lodoxamide
Functional ProTracer identifies patterns of cell proliferation in tissues and underlying regulatory mechanisms
期刊论文
OAI收割
NPJ REGENERATIVE MEDICINE, 2023, 卷号: 8, 期号: 1, 页码: 7
作者:
Liu, Xiuxiu
;
Han, Maoying
;
Weng, Wendong
;
Li, Yan
;
Pu, Wenjuan
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2023/10/17
The PIWI-specific insertion module helps load longer piRNAs for translational activation essential for male fertility
期刊论文
OAI收割
SCIENCE CHINA-LIFE SCIENCES, 2023, 页码: 23
作者:
Wang, Xin
;
Lin, Di-Hang
;
Yan, Yue
;
Wang, An-Hui
;
Liao, Jiaoyang
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2023/10/17
PIWI
piRNAs
PIWI-Ins
translational activation
spermatid development
male fertility
Photochemically controlled activation of STING by CAIX-targeting photocaged agonists to suppress tumor cell growth
期刊论文
OAI收割
CHEMICAL SCIENCE, 2023, 卷号: 14, 期号: 22, 页码: 5956-5964
作者:
Ding, Chunyong
;
Du, Mengyan
;
Xiong, Zhi
;
Wang, Xue
;
Li, Hongji
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2023/10/17
Structural insights into ligand recognition and activation of the medium-chain fatty acid-sensing receptor GPR84
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 14
作者:
Liu, Heng
;
Zhang, Qing
;
He, Xinheng
;
Jiang, Mengting
;
Wang, Siwei
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2023/10/17
Intranasal delivery of replicating mRNA encoding hACE2-targeting antibody against SARS-CoV-2 Omicron infection in the hamster
期刊论文
OAI收割
ANTIVIRAL RESEARCH, 2023, 卷号: 209, 页码: 9
作者:
Zhang, Ya-Nan
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2023/04/10
Omicron
VEEV VRP
Replicable mRNA
Molecular recognition of two endogenous hormones by the human parathyroid hormone receptor-1
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2022, 页码: 11
作者:
Zhao, Li-hua
;
Yuan, Qing-ning
;
Dai, An-tao
;
He, Xin-heng
;
Chen, Chuan-wei
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2023/04/10
G protein- coupled receptors
parathyroid hormone
PTH-related peptide
PTH receptor-1
cryo-electron microscopy structure
osteoporosis
Mass spectrometry imaging: new eyes on natural products for drug research and development
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2022, 页码: 16
作者:
Hou, Jin-jun
;
Zhang, Zi-jia
;
Wu, Wen-yong
;
He, Qing-qing
;
Zhang, Teng-qian
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2022/11/11
natural product
mass spectrometry imaging
MALDI
DESI
molecular imaging
ion mobility
Artemisinin analog SM934 alleviates epithelial barrier dysfunction via inhibiting apoptosis and caspase-1-mediated pyroptosis in experimental colitis
期刊论文
OAI收割
FRONTIERS IN PHARMACOLOGY, 2022, 卷号: 13, 页码: 18
作者:
Shao, Meijuan
;
Yan, Yuxi
;
Zhu, Fenghua
;
Yang, Xiaoqian
;
Qi, Qing
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2022/11/11
SM934
colitis
intestinal epithelial barrier
apoptosis
pyroptosis
NLRP3/caspase-1/GSDMD
MAPK/NF-kB
Rational Design and Identification of Novel Piperine Derivatives as Multichitinase Inhibitors
期刊论文
OAI收割
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2022, 卷号: 70, 期号: 33, 页码: 10326-10336
作者:
Jiang, Zhiyang
;
Shi, Dongmei
;
Li, Huilin
;
He, Danchan
;
Zhu, Kai
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2022/09/30
Asian corn borer
chitinase
piperine derivate
multichitinase inhibitor
insect growth regulator (IGR)