中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 上海药物研究所 [48]
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A first-in-human phase 1 study of simnotrelvir, a 3CL-like protease inhibitor for treatment of COVID-19, in healthy adult subjects 期刊论文  OAI收割
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2023, 卷号: 191, 页码: 9
作者:  
Yang, Xin-Mei;  Yang, Yang;  Yao, Bu-Fan;  Ye, Pan-Pan;  Xu, Yan
  |  收藏  |  浏览/下载:11/0  |  提交时间:2023/12/11
Prime editing-based gene correction alleviates the hyperexcitable phenotype and seizures of a genetic epilepsy mouse model 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 页码: 4
作者:  
Cao, Bi-rong;  Huang, Yi-ming;  Tian, Fu-yun;  Li, Jin-hui;  Xu, Chun-long
  |  收藏  |  浏览/下载:26/0  |  提交时间:2023/10/17
Controlled sequential in situ self-assembly and disassembly of a fluorogenic cisplatin prodrug for cancer theranostics 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 1
作者:  
Xidan Wen;  Rui Zhang;  Yuxuan Hu;  Luyan Wu;  He Bai
  |  收藏  |  浏览/下载:14/0  |  提交时间:2023/05/22
Caulophyine A, a Rare Azapyrene Alkaloid from the Roots of Caulophyllum robustum 期刊论文  OAI收割
CHEMICAL & PHARMACEUTICAL BULLETIN, 2022, 卷号: 70, 期号: 4, 页码: 283-285
作者:  
Wei, Wei;  Yuan, Ya-Hong;  Jiao, Fu-Rong;  Zhao, Xiang;  Xiao, Lei
  |  收藏  |  浏览/下载:21/0  |  提交时间:2022/06/15
A propolis-derived small molecule ameliorates metabolic syndrome in obese mice by targeting the CREB/CRTC2 transcriptional complex 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2022, 卷号: 13, 期号: 1, 页码: 20
作者:  
Chen, Yaqiong;  Wang, Jiang;  Wang, Yibing;  Wang, Pengfei;  Zhou, Zan
  |  收藏  |  浏览/下载:29/0  |  提交时间:2022/06/15
Rapamycin recruits SIRT2 for FKBP12 deacetylation during mTOR activity modulation in innate immunity 期刊论文  OAI收割
ISCIENCE, 2021, 卷号: 24, 期号: 11, 页码: 22
作者:  
Hu, Lin;  Chen, Fuxian;  Wu, Chao;  Wang, Jun;  Chen, Si-si
  |  收藏  |  浏览/下载:54/0  |  提交时间:2022/01/18
Sinunanolobatone A, an Anti-inflammatory Diterpenoid with Bicyclo[13.1.0]pentadecane Carbon Scaffold, and Related Casbanes from the Sanya Soft Coral Sinularia nanolobata 期刊论文  OAI收割
ORGANIC LETTERS, 2021, 卷号: 23, 期号: 19, 页码: 7575-7579
作者:  
Zeng, Zi-Rong;  Li, Wang-Sheng;  Nay, Bastien;  Hu, Pei;  Zhang, Hai-Yan
  |  收藏  |  浏览/下载:14/0  |  提交时间:2021/12/01
Anti-DLBCL efficacy of DCZ0825 in vitro and in vivo: involvement of the PI3K-AKT-mTOR/JNK pathway 期刊论文  OAI收割
ACTA BIOCHIMICA ET BIOPHYSICA SINICA, 2021, 卷号: 53, 期号: 5, 页码: 575-583
作者:  
Hu, Ke;  Li, Bo;  Ma, Ruye;  Yi, Hongfei;  Xu, Zhijian
  |  收藏  |  浏览/下载:38/0  |  提交时间:2021/06/11
PI3K alpha inhibitor CYH33 triggers antitumor immunity in murine breast cancer by activating CD8(+)T cells and promoting fatty acid metabolism 期刊论文  OAI收割
JOURNAL FOR IMMUNOTHERAPY OF CANCER, 2021, 卷号: 9, 期号: 8, 页码: 16
作者:  
Sun, Pu;  Zhang, Xi;  Wang, Rong-Jing;  Ma, Qing-Yang;  Xu, Lan
  |  收藏  |  浏览/下载:24/0  |  提交时间:2021/11/04
A novel silicone derivative of natural osalmid (DCZ0858) induces apoptosis and cell cycle arrest in diffuse large B-cell lymphoma via the JAK2/STAT3 pathway 期刊论文  OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2020, 卷号: 5, 期号: 1, 页码: 11
作者:  
Lu, Kang;  Li, Bo;  Zhang, Hui;  Xu, Zhijian;  Song, Dongliang
  |  收藏  |  浏览/下载:29/0  |  提交时间:2020/07/01