中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 上海药物研究所 [47]
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A first-in-human phase 1 study of simnotrelvir, a 3CL-like protease inhibitor for treatment of COVID-19, in healthy adult subjects 期刊论文  OAI收割
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2023, 卷号: 191, 页码: 9
作者:  
Yang, Xin-Mei;  Yang, Yang;  Yao, Bu-Fan;  Ye, Pan-Pan;  Xu, Yan
  |  收藏  |  浏览/下载:11/0  |  提交时间:2023/12/11
Design, Synthesis and Evaluation of Fluorescent Properties of Benzothiazole Derivatives 期刊论文  OAI收割
CHEMPHYSCHEM, 2023, 页码: 13
作者:  
Sun, Yi-Tao;  Zhang, Chun;  Gao, Li-Xin;  Liu, Min-Min;  Yang, Yuting
  |  收藏  |  浏览/下载:19/0  |  提交时间:2023/10/17
A study on optical properties of various hot drug molecules by 2020 期刊论文  OAI收割
NEW JOURNAL OF CHEMISTRY, 2023, 卷号: 47, 期号: 21, 页码: 10046-10060
作者:  
Zhang, Chun;  Yang, Yuting;  Yan, Xue;  Sun, Yi-Tao;  Shao, Andong
  |  收藏  |  浏览/下载:15/0  |  提交时间:2023/10/17
High-throughput screening of SARS-CoV-2 main and papain-like protease inhibitors 期刊论文  OAI收割
PROTEIN & CELL, 2023, 卷号: 14, 期号: 1, 页码: 17-27
作者:  
Zang, Yi;  Su, Mingbo;  Wang, Qingxing;  Cheng, Xi;  Zhang, Wenru
  |  收藏  |  浏览/下载:2/0  |  提交时间:2024/03/27
Engineered bioorthogonal POLY-PROTAC nanoparticles for tumour-specific protein degradation and precise cancer therapy 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2022, 卷号: 13, 期号: 1, 页码: 14
作者:  
Gao, Jing;  Hou, Bo;  Zhu, Qiwen;  Yang, Lei;  Jiang, Xingyu
  |  收藏  |  浏览/下载:41/0  |  提交时间:2022/08/30

A novel aromatic amide derivative SY-65 co-targeted tubulin and histone deacetylase 1 with potent anticancer activity in vitro and in vivo

期刊论文  OAI收割

BIOCHEMICAL PHARMACOLOGY, 2022, 卷号: 201, 页码: 12
作者:  
Li, Yin-Ru;  Liu, Fang-Fang;  Liu, Wen-Bo;  Zhang, Yi-Fan;  Tian, Xin-Yi
  |  收藏  |  浏览/下载:24/0  |  提交时间:2022/08/16
A novel aromatic amide derivative SY-65 co-targeted tubulin and histone deacetylase 1 with potent anticancer activity in vitro and in vivo 期刊论文  OAI收割
BIOCHEMICAL PHARMACOLOGY, 2022, 卷号: 201, 页码: 115070
作者:  
Li, Yin-Ru;  Liu, Fang-Fang;  Liu, Wen-Bo;  Zhang, Yi-Fan;  Tian, Xin-Yi
  |  收藏  |  浏览/下载:10/0  |  提交时间:2024/03/21
Dual-Channel Fluorescent Probe for the Simultaneous Monitoring of Peroxynitrite and Adenosine-5 '-triphosphate in Cellular Applications 期刊论文  OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2021, 页码: 10
作者:  
Wu, Luling;  Liu, Jihong;  Tian, Xue;  Groleau, Robin R.
  |  收藏  |  浏览/下载:37/0  |  提交时间:2022/06/15
Pharmacodynamic, pharmacokinetic, and phase 1a study of bisthianostat, a novel histone deacetylase inhibitor, for the treatment of relapsed or refractory multiple myeloma 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 9
作者:  
Zhou, Yu-bo;  Zhang, Yang-ming;  Huang, Hong-hui;  Shen, Li-jing;  Han, Xiao-feng
  |  收藏  |  浏览/下载:67/0  |  提交时间:2021/11/04
Anti-DLBCL efficacy of DCZ0825 in vitro and in vivo: involvement of the PI3K-AKT-mTOR/JNK pathway 期刊论文  OAI收割
ACTA BIOCHIMICA ET BIOPHYSICA SINICA, 2021, 卷号: 53, 期号: 5, 页码: 575-583
作者:  
Hu, Ke;  Li, Bo;  Ma, Ruye;  Yi, Hongfei;  Xu, Zhijian
  |  收藏  |  浏览/下载:38/0  |  提交时间:2021/06/11