中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [5]
合肥物质科学研究院 [3]
采集方式
OAI收割 [8]
内容类型
期刊论文 [8]
发表日期
2023 [1]
2022 [3]
2020 [2]
2019 [1]
2018 [1]
学科主题
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Identification of [1,2,4]Triazolo[4,3-a]pyrazine PARP1 inhibitors with overcome acquired resistance activities
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 259, 页码: 19
作者:
Wang, Pingyuan
;
Zhu, Wen-Ting
;
Wang, Yajing
;
Song, Shan-Shan
;
Xi, Yong
  |  
收藏
  |  
浏览/下载:58/0
  |  
提交时间:2023/10/17
PARP1 inhibitor
Synthetic lethality
Drug resistance
Anticancer
Structure -activity relationship
Darinaparsin (ZIO-101) enhances the sensitivity of small-cell lung cancer to PARP inhibitors
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2022
作者:
Cao, Guo-Zhen
;
Ma, Li-Ying
;
Zhang, Zong-Hui
;
Wang, Xiao-Lin
;
Hua, Jing-Han
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2022/12/22
small-cell lung cancer
H3
3
PARP1
PARP inhibitor
darinaparsin
combination treatment
Design, synthesis and pharmacological evaluation of new PARP1 inhibitors by merging pharmacophores of olaparib and the natural product alantolactone
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 240, 页码: 114574
作者:
Kayumov, Muzaffar
;
Jia, Li
;
Pardaev, Azizbek
;
Song, Shan-Shan
;
Mirzaakhmedov, Sharafitdin
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2024/03/21
PARP1
Olaparib
Alantolactone
Syntheticlethality
BRCA1/2mutant
Repeated treatments of Capan-1 cells with PARP1 and Chk1 inhibitors promote drug resistance, migration and invasion
期刊论文
OAI收割
CANCER BIOLOGY & THERAPY, 2022, 页码: 14
作者:
Guo, Ne
;
Li, Meng-Zhu
;
Wang, Li-Min
;
Chen, Hua-Dong
;
Song, Shan-Shan
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2022/06/15
Combination therapy
PARP1
resistance
CXCL3-ERK1/2 signaling
migration and invasion
The dual HDAC-PI3K inhibitor CUDC-907 displays single-agent activity and synergizes with PARP inhibitor olaparib in small cell lung cancer
期刊论文
OAI收割
JOURNAL OF EXPERIMENTAL & CLINICAL CANCER RESEARCH, 2020, 卷号: 39
作者:
Ma, Liying
;
Bian, Xing
;
Lin, Wenchu
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2020/11/30
SCLC
PI3K
HDAC
CUDC-907
PARP1
Olaparib
DSB repair
Combination treatment
The MYC Paralog-PARP1 Axis as a Potential TherapeuticTarget in MYC Paralog-Activated Small Cell Lung Cancer
期刊论文
OAI收割
FRONTIERS IN ONCOLOGY, 2020, 卷号: 10
作者:
Bian, Xing
;
Wang, Xiaolin
;
Zhang, Qiuyan
;
Ma, Liying
;
Cao, Guozhen
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2020/11/30
small cell lung cancer
MYCparalog
PARP1
BET
DNA damage response
Increased PARP1-DNA binding due to autoPARylation inhibition of PARP1 on DNA rather than PARP1-DNA trapping is correlated with PARP1 inhibitor's cytotoxicity
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF CANCER, 2019, 卷号: 145, 期号: 3, 页码: 714-727
作者:
Chen, Hua-Dong
;
Chen, Chuan-Huizi
;
Wang, Yu-Ting
;
Guo, Ne
;
Tian, Yu-Nan
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2024/03/21
PARP1 inhibitor
PARP1-DNA binding
PARP1-DNA trapping
poly(ADP-ribose) polymerase activity
cytotoxicity
Design and synthesis of 2-(4,5,6,7-tetrahydrothienopyridin-2-yl)-benzoimidazole carboxamides as novel orally efficacious Poly(ADP-ribose)polymerase (PARP) inhibitors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 145, 页码: 389-403
作者:
Chen, Xuxing
;
Huan, Xiajuan
;
Liu, Qiufeng
;
Wang, Yuqin
;
He, Qian
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2019/01/08
PARP1/2 inhibitor
Benzimidazole
4,5,6,7-Tetrahydrothienopyridine
Co-crystal structure
Isothermal Titration Calorimetry