中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共12条,第1-10条 帮助

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Inhibition of the deubiquitinating enzyme USP47 as a novel targeted therapy for hematologic malignancies expressing mutant EZH2 期刊论文  OAI收割
LEUKEMIA, 2022
作者:  
Yang, Jing;  Weisberg, Ellen L.;  Qi, Shuang;  Ni, Wei;  Mei, Husheng
  |  收藏  |  浏览/下载:68/0  |  提交时间:2022/02/14
Targeting chaperon protein HSP70 as a novel therapeutic strategy for FLT3-ITD-positive acute myeloid leukemia 期刊论文  OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2021, 卷号: 6
作者:  
Hu, Chen;  Zou, Fengming;  Wang, Aoli;  Miao, Weili;  Liang, Qianmao
  |  收藏  |  浏览/下载:42/0  |  提交时间:2021/11/01
Selectively targeting FLT3-ITD mutants over FLT3-wt by a novel inhibitor for acute myeloid leukemia 期刊论文  OAI收割
HAEMATOLOGICA, 2021, 卷号: 106
作者:  
Wang, Aoli;  Hu, Chen;  Chen, Cheng;  Liang, Xiaofei;  Wang, Beilei
  |  收藏  |  浏览/下载:46/0  |  提交时间:2021/04/26
Repurposing of Kinase Inhibitors for Treatment of COVID-19 期刊论文  OAI收割
PHARMACEUTICAL RESEARCH, 2020, 卷号: 37
作者:  
Weisberg, Ellen;  Parent, Alexander;  Yang, Priscilla L.;  Sattler, Martin;  Liu, Qingsong
  |  收藏  |  浏览/下载:49/0  |  提交时间:2020/10/26
Discovery of N-(4-(6-Acetamidopyrimidin-4-yloxy)phenyl)-2-(2-(trifluoromethyl)phenyl)acetamide (CHMFL-FLT3-335) as a Potent FMS-like Tyrosine Kinase 3 Internal Tandem Duplication (FLT3-ITD) Mutant Selective Inhibitor for Acute Myeloid Leukemia 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 2, 页码: 875-892
作者:  
Liang, Xiaofei;  Wang, Beilei;  Chen, Cheng;  Wang, Aoli;  Hu, Chen
  |  收藏  |  浏览/下载:34/0  |  提交时间:2020/05/21
Structure-activity relationship investigation for benzonaphthyridinone derivatives as novel potent Bruton's tyrosine kinase (BTK) irreversible inhibitors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 137, 页码: 545-557
作者:  
Wang, Beilei;  Deng, Yuanxin;  Chen, Yongfei
  |  收藏  |  浏览/下载:39/0  |  提交时间:2018/08/16
Ibrutinib targets mutant-EGFR kinase with a distinct binding conformation 期刊论文  OAI收割
ONCOTARGET, 2016, 卷号: 7, 期号: 43, 页码: 69760-69769
作者:  
收藏  |  浏览/下载:77/0  |  提交时间:2017/11/21
Simultaneous inhibition of Vps34 kinase would enhance PI3K delta inhibitor cytotoxicity in the B-cell malignancies 期刊论文  OAI收割
ONCOTARGET, 2016, 卷号: 7, 期号: 33, 页码: 53515-53525
作者:  
Liu, Xiaochuan;  Wang, Aoli;  Liang, Xiaofei;  Liu, Juanjuan;  Zou, Fengming
收藏  |  浏览/下载:32/0  |  提交时间:2017/11/21
Characterization of selective and potent PI3K delta inhibitor (PI3KD-IN-015) for B-Cell malignances 期刊论文  OAI收割
ONCOTARGET, 2016, 卷号: 7, 期号: 22, 页码: 32641-32651
作者:  
Liu, Xiaochuan;  Wang, Aoli;  Liang, Xiaofei;  Chen, Cheng;  Liu, Juanjuan
收藏  |  浏览/下载:19/0  |  提交时间:2017/11/16
Dual Inhibition of AKT/FLT3-ITD by A674563 Overcomes FLT3 Ligand-Induced Drug Resistance in FLT3-ITD positive AML 期刊论文  OAI收割
ONCOTARGET, 2016, 卷号: 7, 期号: 20, 页码: 29131-29142
作者:  
Wang, Aoli;  Wu, Hong;  Chen, Cheng;  Hu, Chen;  Qi, Ziping
收藏  |  浏览/下载:15/0  |  提交时间:2017/11/16