中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
机构
  • 上海药物研究所 [33]
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内容类型
发表日期
  • 2020 [33]
学科主题
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浏览/检索结果: 共33条,第1-10条 帮助

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Modulation of the G-Protein-Coupled Receptor 84 (GPR84) by Agonists and Antagonists 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 24, 页码: 15399-15409
作者:  
Chen, Lin-Hai;  Zhang, Qing;  Xie, Xin;  Nan, Fa-Jun
  |  收藏  |  浏览/下载:18/0  |  提交时间:2021/05/24
Liquid chromatography-tandem mass spectrometric assay for TPN171 in human plasma 期刊论文  OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2020, 卷号: 191, 页码: 8
作者:  
Zhang, Mengqi;  Liu, Haiming;  He, Jiajin;  Gui, Yuzhou;  Qian, Hongjie
  |  收藏  |  浏览/下载:38/0  |  提交时间:2020/12/24
Pharmacokinetics, mass balance, and metabolism of [C-14]vicagrel, a novel irreversible P2Y(12) inhibitor in humans 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 12
作者:  
Zheng, Yuan-dong;  Zhang, Hua;  Zhan, Yan;  Bian, Yi-cong;  Ma, Sheng
  |  收藏  |  浏览/下载:29/0  |  提交时间:2021/05/24
Discovery and Optimization of Non-bile Acid FXR Agonists as Preclinical Candidates for the Treatment of Nonalcoholic Steatohepatitis 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 21, 页码: 12748-12772
作者:  
Li, Junyou;  Liu, Mengqi;  Li, Yazhou;  Sun, Dan-dan;  Shu, Zhihao
  |  收藏  |  浏览/下载:25/0  |  提交时间:2021/05/24
Direct quantification of anorethidrani disuccinate and determination of sterol metabolites by chemical derivatization combined with LC-MS/MS: Application to a Phase I pharmacokinetic study in humans 期刊论文  OAI收割
JOURNAL OF CHROMATOGRAPHY B-ANALYTICAL TECHNOLOGIES IN THE BIOMEDICAL AND LIFE SCIENCES, 2020, 卷号: 1157, 页码: 9
作者:  
Jiang, Jinfang;  Li, Liang;  Lu, Youming;  Chen, Yunhui;  Chen, Xiaoyan
  |  收藏  |  浏览/下载:23/0  |  提交时间:2020/12/24
SAF-189s, a potent new-generation ROS1 inhibitor, is active against crizotinib-resistant ROS1 mutant-driven tumors 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 7
作者:  
Xia, Zong-jun;  Ji, Yin-chun;  Sun, De-qiao;  Peng, Xia;  Gao, Ying-lei
  |  收藏  |  浏览/下载:47/0  |  提交时间:2020/12/21
Intrinsic stability study of L-alpha-glycerylphosphorylcholine with HPLC method development and validation 期刊论文  OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2020, 卷号: 188, 页码: 6
作者:  
Zhao, Hongwei;  Sun, Ling;  Chen, Huanhuan;  Xiang, Lili;  Chen, Dongying
  |  收藏  |  浏览/下载:19/0  |  提交时间:2020/12/24
Machine-Driven Chemoenzymatic Synthesis of Glycopeptide 期刊论文  OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2020, 页码: 6
作者:  
Zhang, Jiabin;  Liu, Ding;  Saikam, Varma;  Gadi, Madhusudhan R.;  Gibbons, Christopher
  |  收藏  |  浏览/下载:36/0  |  提交时间:2020/12/24
Activation of unfolded protein response overcomes Ibrutinib resistance in diffuse large B-cell lymphoma 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 10
作者:  
Zhang, Xiao-tuan;  Hu, Xiao-bei;  Wang, Han-lin;  Kan, Wei-juan;  Xu, Lei
  |  收藏  |  浏览/下载:75/0  |  提交时间:2020/12/24
Design, synthesis and biological evaluation of potent EGFR kinase inhibitors against 19D/T790M/C797S mutation 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 卷号: 30, 期号: 16, 页码: 6
作者:  
Su, Zhicheng;  Yang, Tingyuan;  Wang, Jie;  Lai, Mengzhen;  Tong, Linjiang
  |  收藏  |  浏览/下载:62/0  |  提交时间:2020/12/24
EGFR  NSCLC  C797S