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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [844]
采集方式
OAI收割 [844]
内容类型
期刊论文 [844]
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2024 [6]
2023 [49]
2022 [57]
2021 [61]
2020 [67]
2019 [48]
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Biochemist... [6]
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浏览/检索结果:
共844条,第1-10条
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存缴方式:oaiharvest
内容类型:期刊论文
专题:上海药物研究所
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Palladium(II)-Catalyzed Tandem γ-C(sp
2
)-H Arylation and Cyclization for the Construction of Natural Product-Like Polycyclic Fused
ortho
-Quinone Scaffolds
期刊论文
OAI收割
ORGANIC LETTERS, 2024, 页码: 6
作者:
Li, Xingjun
;
Chen, Yu
;
Xie, Xiong
;
Li, Jing
;
Wang, Jiang
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/05/22
Discovery and Optimization of Novel Nonbile Acid FXR Agonists as Preclinical Candidates for the Treatment of Inflammatory Bowel Disease
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 7, 页码: 5642-5661
作者:
Li, Yuan
;
Xu, Tingting
;
Zhao, Yue
;
Zhang, Hui
;
Liu, Zesheng
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2024/05/07
Palladium(II)-Catalyzed Heck Coupling: Direct Stereoselective Synthesis of
C
-Aryl Glycosides from Nonactivated Glycals and Thianthrenium Salts
期刊论文
OAI收割
ORGANIC LETTERS, 2024, 页码: 5
作者:
Wei, Xinxin
;
Zeng, Mingjie
;
Li, Yazhou
;
Wang, Dechuan
;
Wang, Jiang
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2024/05/07
Structure-based design of pan-coronavirus inhibitors targeting host cathepsin L and calpain-1
期刊论文
OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2024, 卷号: 9, 期号: 1, 页码: 14
作者:
Xie, Xiong
;
Lan, Qiaoshuai
;
Zhao, Jinyi
;
Zhang, Sulin
;
Liu, Lu
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/05/07
Ent-labdane-type diterpene glycosides obtained from
Rubus
chingii
Hu and their inhibitory effects on PDE5A activity
期刊论文
OAI收割
FITOTERAPIA, 2024, 卷号: 173, 页码: 14
作者:
Yu, Jun-dong
;
Wang, Jing-Yi
;
Liu, Jia-yuan
;
Xu, Ye-chun
;
Zhang, Xue
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/02/27
diterpene glycosides
Rubus Chingii Hu
PDE5A inhibitory activity
ent-labdane
Discovery, Optimization, and Evaluation of Novel Pyridin-2(1
H
)-one Analogues as Potent TRK Inhibitors for Cancer Treatment
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 2, 页码: 1168-1183
作者:
Xu, Zichao
;
Peng, Xia
;
Zhang, Renjie
;
Ji, Yinchun
;
You, Mengke
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2024/02/27
Recognition of methamphetamine and other amines by trace amine receptor TAAR1
期刊论文
OAI收割
NATURE, 2023, 卷号: 624, 期号: 7992, 页码: 663-+
作者:
Liu, Heng
;
Zheng, You
;
Wang, Yue
;
Wang, Yumeng
;
He, Xinheng
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2024/03/25
Safety, tolerability and pharmacokinetics of forsythin in healthy subjects: a double-blinded, placebo-controlled single-dose and multiple-dose escalation and food effect study
期刊论文
OAI收割
ANNALS OF MEDICINE, 2023, 卷号: 55, 期号: 2, 页码: 9
作者:
Li, Cuiyun
;
Wu, Min
;
Zhang, Hong
;
Zhu, Xiaoxue
;
Fu, Li
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2024/01/16
Forsythin
pharmacokinetics
safety
tolerability
food effect
Substrate- and Catalyst-Controlled C-H Bond Activation/Annulation for Construction of Pyrido[2,3,4-
de
]quinazolinones and Indolo[1,2-
c
]quinazolinones
期刊论文
OAI收割
ADVANCED SYNTHESIS & CATALYSIS, 2023, 页码: 8
作者:
Hou, Xinjiao
;
Wang, Run
;
Zhou, Jianhui
;
Li, Yuan
;
Li, Jiyuan
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/01/16
C-H bond activation
Fused heterocycles
Rh(III) catalysis
Ru(II) catalysis
A first-in-human phase 1 study of simnotrelvir, a 3CL-like protease inhibitor for treatment of COVID-19, in healthy adult subjects
期刊论文
OAI收割
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2023, 卷号: 191, 页码: 9
作者:
Yang, Xin-Mei
;
Yang, Yang
;
Yao, Bu-Fan
;
Ye, Pan-Pan
;
Xu, Yan
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/12/11
COVID-19
Simnotrelvir
Safety
Pharmacokinetics
Healthy subjects