中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 上海药物研究所 [844]
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  • OAI收割 [844]
内容类型
  • 期刊论文 [844]
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浏览/检索结果: 共844条,第1-10条 帮助

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Palladium(II)-Catalyzed Tandem γ-C(sp2)-H Arylation and Cyclization for the Construction of Natural Product-Like Polycyclic Fused ortho-Quinone Scaffolds 期刊论文  OAI收割
ORGANIC LETTERS, 2024, 页码: 6
作者:  
Li, Xingjun;  Chen, Yu;  Xie, Xiong;  Li, Jing;  Wang, Jiang
  |  收藏  |  浏览/下载:1/0  |  提交时间:2024/05/22
Discovery and Optimization of Novel Nonbile Acid FXR Agonists as Preclinical Candidates for the Treatment of Inflammatory Bowel Disease 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 7, 页码: 5642-5661
作者:  
Li, Yuan;  Xu, Tingting;  Zhao, Yue;  Zhang, Hui;  Liu, Zesheng
  |  收藏  |  浏览/下载:3/0  |  提交时间:2024/05/07
Palladium(II)-Catalyzed Heck Coupling: Direct Stereoselective Synthesis of C-Aryl Glycosides from Nonactivated Glycals and Thianthrenium Salts 期刊论文  OAI收割
ORGANIC LETTERS, 2024, 页码: 5
作者:  
Wei, Xinxin;  Zeng, Mingjie;  Li, Yazhou;  Wang, Dechuan;  Wang, Jiang
  |  收藏  |  浏览/下载:2/0  |  提交时间:2024/05/07
Structure-based design of pan-coronavirus inhibitors targeting host cathepsin L and calpain-1 期刊论文  OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2024, 卷号: 9, 期号: 1, 页码: 14
作者:  
Xie, Xiong;  Lan, Qiaoshuai;  Zhao, Jinyi;  Zhang, Sulin;  Liu, Lu
  |  收藏  |  浏览/下载:1/0  |  提交时间:2024/05/07
Ent-labdane-type diterpene glycosides obtained from Rubus chingii Hu and their inhibitory effects on PDE5A activity 期刊论文  OAI收割
FITOTERAPIA, 2024, 卷号: 173, 页码: 14
作者:  
Yu, Jun-dong;  Wang, Jing-Yi;  Liu, Jia-yuan;  Xu, Ye-chun;  Zhang, Xue
  |  收藏  |  浏览/下载:12/0  |  提交时间:2024/02/27
Discovery, Optimization, and Evaluation of Novel Pyridin-2(1H)-one Analogues as Potent TRK Inhibitors for Cancer Treatment 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 2, 页码: 1168-1183
作者:  
Xu, Zichao;  Peng, Xia;  Zhang, Renjie;  Ji, Yinchun;  You, Mengke
  |  收藏  |  浏览/下载:14/0  |  提交时间:2024/02/27
Recognition of methamphetamine and other amines by trace amine receptor TAAR1 期刊论文  OAI收割
NATURE, 2023, 卷号: 624, 期号: 7992, 页码: 663-+
作者:  
Liu, Heng;  Zheng, You;  Wang, Yue;  Wang, Yumeng;  He, Xinheng
  |  收藏  |  浏览/下载:20/0  |  提交时间:2024/03/25
Safety, tolerability and pharmacokinetics of forsythin in healthy subjects: a double-blinded, placebo-controlled single-dose and multiple-dose escalation and food effect study 期刊论文  OAI收割
ANNALS OF MEDICINE, 2023, 卷号: 55, 期号: 2, 页码: 9
作者:  
Li, Cuiyun;  Wu, Min;  Zhang, Hong;  Zhu, Xiaoxue;  Fu, Li
  |  收藏  |  浏览/下载:26/0  |  提交时间:2024/01/16
Substrate- and Catalyst-Controlled C-H Bond Activation/Annulation for Construction of Pyrido[2,3,4-de]quinazolinones and Indolo[1,2-c]quinazolinones 期刊论文  OAI收割
ADVANCED SYNTHESIS & CATALYSIS, 2023, 页码: 8
作者:  
Hou, Xinjiao;  Wang, Run;  Zhou, Jianhui;  Li, Yuan;  Li, Jiyuan
  |  收藏  |  浏览/下载:7/0  |  提交时间:2024/01/16
A first-in-human phase 1 study of simnotrelvir, a 3CL-like protease inhibitor for treatment of COVID-19, in healthy adult subjects 期刊论文  OAI收割
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2023, 卷号: 191, 页码: 9
作者:  
Yang, Xin-Mei;  Yang, Yang;  Yao, Bu-Fan;  Ye, Pan-Pan;  Xu, Yan
  |  收藏  |  浏览/下载:11/0  |  提交时间:2023/12/11