中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
机构
  • 上海药物研究所 [15]
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发表日期
  • 2019 [15]
学科主题
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LysargiNase and Chemical Derivatization Based Strategy for Facilitating In-Depth Profiling of C-Terminome 期刊论文  OAI收割
ANALYTICAL CHEMISTRY, 2019, 卷号: 91, 期号: 22, 页码: 14522-14529
作者:  
Hu, Hao;  Zhao, Wensi;  Zhu, Mengdi;  Zhao, Lei;  Zhai, Linhui
  |  收藏  |  浏览/下载:15/0  |  提交时间:2020/07/01
Comparison of high-resolution synchrotron-radiation-based phase-contrast imaging and absorption-contrast imaging for evaluating microstructure of vascular networks in rat brain: from 2D to 3D views 期刊论文  OAI收割
JOURNAL OF SYNCHROTRON RADIATION, 2019, 卷号: 26, 页码: 2024-2032
作者:  
Li, Hong-Lei;  Ding, Hui;  Yin, Xian-Zhen;  Chen, Zhuo-Hui;  Tang, Bin
  |  收藏  |  浏览/下载:34/0  |  提交时间:2020/07/01
Peptide Nanotube-Templated Biomineralization of Cu2-xS Nanoparticles for Combination Treatment of Metastatic Tumor 期刊论文  OAI收割
SMALL, 2019, 页码: 13
作者:  
Lai, Yi;  Xu, Zhiai;  Hu, Xianli;  Lei, Li;  Li, Lingling
  |  收藏  |  浏览/下载:19/0  |  提交时间:2020/07/01
fDiscovery of pyrazole-thiophene derivatives as highly Potent, orally active Akt inhibitors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 180, 页码: 72-85
作者:  
Zhan, Wenhu;  Che, Jinxin;  Xu, Lei;  Wu, Yizhe;  Hu, Xiaobei
  |  收藏  |  浏览/下载:20/0  |  提交时间:2020/07/01
Discovery of 3,4,6-Trisubstituted Piperidine Derivatives as Orally Active, Low hERG Blocking Akt Inhibitors via Conformational Restriction and Structure-Based Design 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 15, 页码: 7264-7288
作者:  
Dong, Xiaowu;  Zhan, Wenhu;  Zhao, Mengting;  Che, Jinxin;  Dai, Xiaoyang
  |  收藏  |  浏览/下载:26/0  |  提交时间:2020/07/01
Discovery of (R)-5-((5-(1-methyl-1H-pyrazol-4-yl)-4-(methylamino) pyrimidin-2-yl)amino)-3-(piperidin-3-yloxy)picolinonitrile, a novel CHK1 inhibitor for hematologic malignancies 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 173, 页码: 44-62
作者:  
Tong, Lexian;  Song, Pinrao;  Jiang, Kailong;  Xu, Lei;  Jin, Tingting
  |  收藏  |  浏览/下载:24/0  |  提交时间:2020/07/01
Bioinspired Multivalent Peptide Nanotubes for Sialic Acid Targeting and Imaging-Guided Treatment of Metastatic Melanoma 期刊论文  OAI收割
SMALL, 2019, 卷号: 15, 期号: 22, 页码: 11
作者:  
Lei, Li;  Xu, Zhiai;  Hu, Xianli;  Lai, Yi;  Xu, Jie
  |  收藏  |  浏览/下载:16/0  |  提交时间:2020/07/01
Small-Molecule Targeting of Oncogenic FTO Demethylase in Acute Myeloid Leukemia 期刊论文  OAI收割
CANCER CELL, 2019, 卷号: 35, 期号: 4, 页码: 677-+
作者:  
Huang, Yue;  Su, Rui;  Sheng, Yue;  Dong, Lei;  Dong, Ze
  |  收藏  |  浏览/下载:20/0  |  提交时间:2020/07/01
MiR-183-5p is required for non-small cell lung cancer progression by repressing PTEN 期刊论文  OAI收割
BIOMEDICINE & PHARMACOTHERAPY, 2019, 卷号: 111, 页码: 1103-1111
作者:  
Wang, Huimin;  Ma, Zhongliang;  Liu, Xiaomin;  Zhang, Caiyan;  Hu, Yanping
  |  收藏  |  浏览/下载:12/0  |  提交时间:2020/07/01
Covalent docking modelling-based discovery of tripeptidyl epoxyketone proteasome inhibitors composed of aliphatic-heterocycles 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 164, 页码: 602-614
作者:  
Dong, Xiao-Wu;  Zhang, Jian-Kang;  Xu, Lei;  Che, Jin-Xin;  Cheng, Gang
  |  收藏  |  浏览/下载:18/0  |  提交时间:2020/07/01