机构

• 上海药物研究所 [27]

采集方式

• OAI收割 [27]

内容类型

• 期刊论文 [27]

发表日期

• 2021 [27]

学科主题

筛选

浏览/检索结果: 共27条，第1-10条 帮助 限定条件 发表日期：2021    专题：上海药物研究所    第一署名单位    第一作者单位    通讯作者单位     条数/页： 5101520253035404550556065707580859095100 排序方式： 请选择提交时间升序提交时间降序题名升序题名降序作者升序作者降序发表日期升序发表日期降序 Design, synthesis and biological evaluation of a novel spiro oxazolidinedione as potent p300/CBP HAT inhibitor for the treatment of ovarian cancer 期刊论文  OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 52, 页码: 12 作者:  Ding, Hong;  Pei, Yuan;  Li, Yuanqing;  Xu, Wen;  Mei, Lianghe   |  收藏  |  浏览/下载：37/0  |  提交时间：2022/06/15 Epigenetics  Histone acetyltransferase  P300/CBP  Ovarian cancer   Structure-Based Discovery of Potent CARM1 Inhibitors for Solid Tumor and Cancer Immunology Therapy 期刊论文  OAI收割 JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 22, 页码: 16650-16674 作者:  Zhang, Zhuqing;  Guo, Zuhao;  Xu, Xiaowei;  Cao, Danyan;  Yang, Hong   |  收藏  |  浏览/下载：25/0  |  提交时间：2022/06/15 Discovery of a novel DDRs kinase inhibitor XBLJ-13 for the treatment of idiopathic pulmonary fibrosis 期刊论文  OAI收割 ACTA PHARMACOLOGICA SINICA, 2021, 页码: 11 作者:  Dong, Ying;  Tang, Bi-xi;  Wang, Qi;  Zhou, Li-wei;  Li, Cong   |  收藏  |  浏览/下载：53/0  |  提交时间：2022/01/04 idiopathic pulmonary fibrosis  DDRs  kinase inhibitor  indazole derivatives  XBLJ-13  nintedanib  bleomycin-induced pulmonary fibrosismouse model   Inhibition of Autophagy by a Small Molecule through Covalent Modification of the LC3 Protein 期刊论文  OAI收割 ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2021, 页码: 11 作者:  Fan, Shijie   |  收藏  |  浏览/下载：98/0  |  提交时间：2021/12/16 covalent modification  probes  proteome  LC3  post-translational modification   PARP14 inhibits microglial activation via LPAR5 to promote post-stroke functional recovery 期刊论文  OAI收割 AUTOPHAGY, 2021, 卷号: 17, 期号: 10, 页码: 2905-2922 作者:  Tang, Ying;  Liu, Jinchang;  Wang, Yu;  Yang, Li;  Han, Bing   |  收藏  |  浏览/下载：42/0  |  提交时间：2022/01/04 Autophagy  functional recovery  ischemic stroke  lysophosphatidic acid receptor 5  microglial activation  poly (ADP-ribose) polymerase 14   Discovery of a subtype-selective, covalent inhibitor against palmitoylation pocket of TEAD3 期刊论文  OAI收割 ACTA PHARMACEUTICA SINICA B, 2021, 卷号: 11, 期号: 10, 页码: 3206-3219 作者:  Lu, Tian;  Li, Yong;  Lu, Wenchao;  Spitters, Twgm;  Fang, Xueyu   |  收藏  |  浏览/下载：45/0  |  提交时间：2021/12/01 Hippo pathway  TEAD3  Covalent inhibitor  Palmitoylation inhibitor   Ketamine activated glutamatergic neurotransmission by GABAergic disinhibition in the medial prefrontal cortex 期刊论文  OAI收割 NEUROPHARMACOLOGY, 2021, 卷号: 194, 页码: 10 作者:  Zhang, Bing;  Yang, Xili;  Ye, Luyu;  Liu, Rui;  Ye, Binglu   |  收藏  |  浏览/下载：31/0  |  提交时间：2021/08/17 Spiro ent-Clerodane Dimers: Discovery and Green Approaches for a Scalable Biomimetic Synthesis 期刊论文  OAI收割 ORGANIC LETTERS, 2021, 卷号: 23, 期号: 15, 页码: 5647-5651 作者:  Li, Xing-Ren;  Yan, Bing-Chao;  Hu, Kun;  He, Shijun;  Sun, Han-Dong   |  收藏  |  浏览/下载：26/0  |  提交时间：2021/11/04 Discovery of SARS-CoV-2-E channel inhibitors as antiviral candidates 期刊论文  OAI收割 ACTA PHARMACOLOGICA SINICA, 2021, 页码: 7 作者:  Wang, Yi;  Fang, Sui;  Wu, Yan;  Cheng, Xi;  Zhang, Lei-ke   |  收藏  |  浏览/下载：67/0  |  提交时间：2021/08/17 SARS-CoV-2  envelope protein (2-E)  cation channel  high-throughput screening (HTS)  anti-virus   A new mechanism of obeticholic acid on NASH treatment by inhibiting NLRP3 inflammasome activation in macrophage 期刊论文  OAI收割 METABOLISM-CLINICAL AND EXPERIMENTAL, 2021, 卷号: 120, 页码: 12 作者:  Huang, Suling;  Wu, Yanwei;  Zhao, Zhuohui;  Wu, Bing;  Sun, Kai   |  收藏  |  浏览/下载：108/0  |  提交时间：2021/08/17 Macrophage  NLRP3 inflammasome  Hepatic lipid accumulation  NASH  FXR