中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [7]
中国科学院大学 [1]
海洋研究所 [1]
上海生物化学与细胞生... [1]
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OAI收割 [9]
iSwitch采集 [1]
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期刊论文 [10]
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2022 [2]
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2019 [2]
2017 [2]
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2008 [1]
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Biotechnol... [1]
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Absorption, distribution, metabolism, and excretion of [C-14]Mefuparib (CVL218), a novel PARP1/2 inhibitor, in rats
期刊论文
OAI收割
CANCER CHEMOTHERAPY AND PHARMACOLOGY, 2022, 页码: 12
作者:
Li, Xin-mei
;
Zheng, Yuan-dong
;
Zhang, Yi-fan
;
Huan, Xia-juan
;
Yang, Chen
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2022/12/13
[C-14]Mefuparib
Mefuparib (CVL218)
Blood-brain barrier
Mass balance
Tissue distribution
GastroPlus simulation
Metabolite profiles and mass balance of fuzuloparib, a novel poly (ADP-ribose) polymerase inhibitor, in subjects with advanced solid cancers
期刊论文
OAI收割
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 2022, 页码: 14
作者:
Bian, Yicong
;
Meng, Jian
;
Ma, Sheng
;
Li, Guangze
;
Wang, Yuya
  |  
收藏
  |  
浏览/下载:79/0
  |  
提交时间:2022/06/15
fuzuloparib
mass balance
metabolite profiles
PARP
pharmacokinetics
PARP14 inhibits microglial activation via LPAR5 to promote post-stroke functional recovery
期刊论文
OAI收割
AUTOPHAGY, 2021, 卷号: 17, 期号: 10, 页码: 2905-2922
作者:
Tang, Ying
;
Liu, Jinchang
;
Wang, Yu
;
Yang, Li
;
Han, Bing
  |  
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2022/01/04
Autophagy
functional recovery
ischemic stroke
lysophosphatidic acid receptor 5
microglial activation
poly (ADP-ribose) polymerase 14
BOS-93, a novel bromophenol derivative, induces apoptosis and autophagy in human A549 lung cancer cells via PI3K/Akt/mTOR and MAPK signaling pathway
期刊论文
OAI收割
EXPERIMENTAL AND THERAPEUTIC MEDICINE, 2019, 卷号: 17, 期号: 5, 页码: 3848-3858
作者:
Guo, Chuanlong
;
Wang, Lijun
;
Zhao, Yue
;
Jiang, Bo
;
Luo, Jiao
  |  
收藏
  |  
浏览/下载:117/0
  |  
提交时间:2019/08/28
bromophenol
apoptosis
autophagy
phosphoinositide 3-kinase
protein kinase B
mechanistic target of rapamycin signaling
reactive oxygen species
Pharmacologic characterization of fluzoparib, a novel poly(ADP-ribose) polymerase inhibitor undergoing clinical trials
期刊论文
OAI收割
CANCER SCIENCE, 2019, 卷号: 110, 期号: 3, 页码: 1064-1075
作者:
Wang, Lei
;
Yang, Changyong
;
Xie, Chengying
;
Jiang, Jiahua
;
Gao, Mingzhao
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2020/07/01
antitumor activity
fluzoparib
pharmacokinetics
poly(ADP-ribose) polymerase
toxicity
Discovery of potent 2,4-difluoro-linker poly(ADP-ribose) polymerase 1 inhibitors with enhanced water solubility and in vivo anticancer efficacy
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2017, 卷号: 38, 期号: 11, 页码: 1521-1532
作者:
Chen, Wen-hua
;
Song, Shan-shan
;
Qi, Ming-hui
;
Huan, Xia-juan
;
Wang, Ying-qing
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2019/01/08
PARP-1 inhibitor
olaparib
breast cancer
BRCA-deficient tumors
Discovery, mechanism and metabolism studies of 2,3-difluorophenyl-linker-containing PARP1 inhibitors with enhanced in vivo efficacy for cancer therapy
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 138, 页码: 514-531
作者:
Chen, Wenhua
;
Guo, Ne
;
Qi, Minghui
;
Dai, Haiying
;
Hong, Minghuang
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2019/01/08
Antitumor drug
BRCA1/2
PARP inhibitors
Molecular docking
Mixed galactolipid anomers accentuate apoptosis of multiple myeloma cells by inducing DNA damage
期刊论文
OAI收割
CARBOHYDRATE RESEARCH, 2015, 卷号: 408, 页码: 114-118
作者:
Deng, Si-Si
;
Zhang, Chao
;
Wang, Huan
;
Zang, Yi
;
Li, Jia
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2019/01/08
Multiple myeloma
Glycolipid
Anomer
Synergism
Apoptosis
Experimental therapy of hepatoma with artemisinin and its derivatives: in vitro and in vivo activity, chemosensitization, and mechanisms of action
期刊论文
iSwitch采集
Clinical cancer research, 2008, 卷号: 14, 期号: 17, 页码: 5519-5530
作者:
Hou, Junmei
;
Wang, Disong
;
Zhang, Ruiwen
;
Wang, Hui
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2019/05/10
Potent antitumor efficacy of XAF1 delivered by conditionally replicative adenovirus vector via caspase-independent apoptosis
期刊论文
OAI收割
CANCER GENE THERAPY, 2007, 卷号: 14, 期号: 1, 页码: 82-90
作者:
Qi, R
;
Gu, J
;
Zhang, Z
;
Yang, K
;
Li, B
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2015/07/22
XAF1
ZD55
caspase-independent apoptosis
gene-virotherapy