中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共10条,第1-10条 帮助

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Absorption, distribution, metabolism, and excretion of [C-14]Mefuparib (CVL218), a novel PARP1/2 inhibitor, in rats 期刊论文  OAI收割
CANCER CHEMOTHERAPY AND PHARMACOLOGY, 2022, 页码: 12
作者:  
Li, Xin-mei;  Zheng, Yuan-dong;  Zhang, Yi-fan;  Huan, Xia-juan;  Yang, Chen
  |  收藏  |  浏览/下载:30/0  |  提交时间:2022/12/13
Metabolite profiles and mass balance of fuzuloparib, a novel poly (ADP-ribose) polymerase inhibitor, in subjects with advanced solid cancers 期刊论文  OAI收割
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 2022, 页码: 14
作者:  
Bian, Yicong;  Meng, Jian;  Ma, Sheng;  Li, Guangze;  Wang, Yuya
  |  收藏  |  浏览/下载:79/0  |  提交时间:2022/06/15
PARP14 inhibits microglial activation via LPAR5 to promote post-stroke functional recovery 期刊论文  OAI收割
AUTOPHAGY, 2021, 卷号: 17, 期号: 10, 页码: 2905-2922
作者:  
Tang, Ying;  Liu, Jinchang;  Wang, Yu;  Yang, Li;  Han, Bing
  |  收藏  |  浏览/下载:42/0  |  提交时间:2022/01/04
BOS-93, a novel bromophenol derivative, induces apoptosis and autophagy in human A549 lung cancer cells via PI3K/Akt/mTOR and MAPK signaling pathway 期刊论文  OAI收割
EXPERIMENTAL AND THERAPEUTIC MEDICINE, 2019, 卷号: 17, 期号: 5, 页码: 3848-3858
作者:  
Guo, Chuanlong;  Wang, Lijun;  Zhao, Yue;  Jiang, Bo;  Luo, Jiao
  |  收藏  |  浏览/下载:117/0  |  提交时间:2019/08/28
Pharmacologic characterization of fluzoparib, a novel poly(ADP-ribose) polymerase inhibitor undergoing clinical trials 期刊论文  OAI收割
CANCER SCIENCE, 2019, 卷号: 110, 期号: 3, 页码: 1064-1075
作者:  
Wang, Lei;  Yang, Changyong;  Xie, Chengying;  Jiang, Jiahua;  Gao, Mingzhao
  |  收藏  |  浏览/下载:21/0  |  提交时间:2020/07/01
Discovery of potent 2,4-difluoro-linker poly(ADP-ribose) polymerase 1 inhibitors with enhanced water solubility and in vivo anticancer efficacy 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2017, 卷号: 38, 期号: 11, 页码: 1521-1532
作者:  
Chen, Wen-hua;  Song, Shan-shan;  Qi, Ming-hui;  Huan, Xia-juan;  Wang, Ying-qing
  |  收藏  |  浏览/下载:26/0  |  提交时间:2019/01/08
Discovery, mechanism and metabolism studies of 2,3-difluorophenyl-linker-containing PARP1 inhibitors with enhanced in vivo efficacy for cancer therapy 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 138, 页码: 514-531
作者:  
Chen, Wenhua;  Guo, Ne;  Qi, Minghui;  Dai, Haiying;  Hong, Minghuang
  |  收藏  |  浏览/下载:29/0  |  提交时间:2019/01/08
Mixed galactolipid anomers accentuate apoptosis of multiple myeloma cells by inducing DNA damage 期刊论文  OAI收割
CARBOHYDRATE RESEARCH, 2015, 卷号: 408, 页码: 114-118
作者:  
Deng, Si-Si;  Zhang, Chao;  Wang, Huan;  Zang, Yi;  Li, Jia
  |  收藏  |  浏览/下载:15/0  |  提交时间:2019/01/08
Experimental therapy of hepatoma with artemisinin and its derivatives: in vitro and in vivo activity, chemosensitization, and mechanisms of action 期刊论文  iSwitch采集
Clinical cancer research, 2008, 卷号: 14, 期号: 17, 页码: 5519-5530
作者:  
Hou, Junmei;  Wang, Disong;  Zhang, Ruiwen;  Wang, Hui
收藏  |  浏览/下载:24/0  |  提交时间:2019/05/10
Potent antitumor efficacy of XAF1 delivered by conditionally replicative adenovirus vector via caspase-independent apoptosis 期刊论文  OAI收割
CANCER GENE THERAPY, 2007, 卷号: 14, 期号: 1, 页码: 82-90
作者:  
Qi, R;  Gu, J;  Zhang, Z;  Yang, K;  Li, B
收藏  |  浏览/下载:16/0  |  提交时间:2015/07/22