中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [10]
采集方式
OAI收割 [10]
内容类型
期刊论文 [10]
发表日期
2021 [10]
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发表日期:2021
专题:上海药物研究所
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Discovery of a novel DDRs kinase inhibitor XBLJ-13 for the treatment of idiopathic pulmonary fibrosis
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 11
作者:
Dong, Ying
;
Tang, Bi-xi
;
Wang, Qi
;
Zhou, Li-wei
;
Li, Cong
  |  
收藏
  |  
浏览/下载:53/0
  |  
提交时间:2022/01/04
idiopathic pulmonary fibrosis
DDRs
kinase inhibitor
indazole derivatives
XBLJ-13
nintedanib
bleomycin-induced pulmonary fibrosismouse model
Sulfoximines Assisted Rh(III)-Catalyzed C-H Activation/Annulation Cascade to Synthesize Highly Fused Indeno-1,2-benzothiazines
期刊论文
OAI收割
JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 86, 期号: 21, 页码: 15217-15227
作者:
Li, Jian
;
Li, Hui
;
Fang, Daqing
;
Liu, Lingjun
;
Han, Xu
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2022/01/04
Identification of Novel Fused Heteroaromatics-Based MALT1 Inhibitors by High-Throughput Screening to Treat B Cell Lymphoma
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 13, 页码: 9217-9237
作者:
Liang, Xuewu
;
Sun, Chenxia
;
Li, Chunpu
;
Yu, Haolan
;
Wei, Xiaohui
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2021/08/17
Structures of human mGlu2 and mGlu7 homo- and heterodimers
期刊论文
OAI收割
NATURE, 2021, 卷号: 594, 期号: 7864, 页码: 589-+
作者:
Du, Juan
;
Wang, Dejian
;
Fan, Hongcheng
;
Xu, Chanjuan
;
Tai, Linhua
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2021/08/17
Natural product 1,2,3,4,6-penta-O-galloyl-beta-D-glucopyranose is a reversible inhibitor of glyceraldehyde 3-phosphate dehydrogenase
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 13
作者:
Li, Wen
;
Liao, Li-ping
;
Song, Ning
;
Liu, Yan-jun
;
Ding, Yi-luan
  |  
收藏
  |  
浏览/下载:44/0
  |  
提交时间:2021/06/11
glyceraldehyde 3-phosphate dehydrogenase
1,2,3,4,6-penta-O-galloyl-beta-D-glucopyranose
hydrogen deuterium exchange mass spectrometry
reversible inhibitor
glycolysis
Natural product 1,2,3,4,6-penta-O-galloyl-beta-D-glucopyranose is a reversible inhibitor of glyceraldehyde 3-phosphate dehydrogenase
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 13
作者:
Li, Wen
;
Liao, Li-ping
;
Song, Ning
;
Liu, Yan-jun
;
Ding, Yi-luan
  |  
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2021/06/11
glyceraldehyde 3-phosphate dehydrogenase
1,2,3,4,6-penta-O-galloyl-beta-D-glucopyranose
hydrogen deuterium exchange mass spectrometry
reversible inhibitor
glycolysis
A novel GPR120-selective agonist promotes insulin secretion and improves chronic inflammation
期刊论文
OAI收割
LIFE SCIENCES, 2021, 卷号: 269, 页码: 8
作者:
Yang, Liu
;
Lei, Xian-Tao
;
Huang, Qi
;
Wang, Ting
;
Sun, Hong-Bin
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2021/05/24
GPR120 agonist
Insulin secretion
Anti-inflammation
Insulin resistance
Type 2 diabetes mellitus
Dehydroberberine Analogue Nanoassemblies for Inducing and Self-Reporting Mitochondrial Dysfunction in Tumor Cells
期刊论文
OAI收割
ACS applied bio materials, 2021, 卷号: 4, 期号: 3, 页码: 2033-2043
作者:
Zhang, Rui
;
An, Ruibing
;
Gu, Zhanni
;
Sun, Haifeng
;
Ye, Deju
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/03/15
dehydroberberine
fluorescence
mitochondria
self-assembly
self-reporting
Novel bivalent BET inhibitor N2817 exhibits potent anticancer activity and inhibits TAF1
期刊论文
OAI收割
BIOCHEMICAL PHARMACOLOGY, 2021, 卷号: 185, 页码: 14
作者:
Wu, Qian
;
Chen, Dan-Qi
;
Sun, Lin
;
Huan, Xia-Juan
;
Bao, Xu-Bin
  |  
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2021/05/24
N2817
Bivalent BET inhibitors
Monovalent BET inhibitors
TAF1
Anticancer activity
Targeting p300/CBP Attenuates Hepatocellular Carcinoma Progression through Epigenetic Regulation of Metabolism
期刊论文
OAI收割
CANCER RESEARCH, 2021, 卷号: 81, 期号: 4, 页码: 860-872
作者:
Cai, Ling-Yan
;
Chen, Shi-Jie
;
Xiao, Sen-Hao
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2024/03/21