中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
机构
采集方式
内容类型
发表日期
学科主题
筛选

浏览/检索结果: 共177条,第1-10条 帮助

条数/页: 排序方式:
The Effects of Topiramate on Ethanol-Cocaine Interactions andDNA Methyltransferase Gene Expression in the Rat Prefrontal Cortex 期刊论文  OAI收割
出版物, 3111, 期号: 0, 页码: 1-39
作者:  
V.Echeverry-Alzate;  E. Gine;  K. M. Bühler;  J. Calleja-Conde;  P. Olmos
  |  收藏  |  浏览/下载:332/0  |  提交时间:2017/07/24
Development of (2-(Benzyloxy)phenyl)methanamine Derivatives as Potent and Selective Inhibitors of CARM1 for the Treatment of Melanoma 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 14
作者:  
Liu, Zhihao;  Lin, Min;  Liu, Chenyu;  Chen, Xin;  Chen, Qian
  |  收藏  |  浏览/下载:0/0  |  提交时间:2024/05/22
Structure-based discovery of a new series of nucleoside-derived ring-opening PRMT5 inhibitors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 267, 页码: 19
作者:  
Chen, Yuting;  Wang, Zekun;  Zhang, Junjie;  Shi, Qiongyu;  Yang, Hong
  |  收藏  |  浏览/下载:1/0  |  提交时间:2024/05/07
PRMT1 Inhibition Activates the Interferon Pathway to Potentiate Antitumor Immunity and Enhance Checkpoint Blockade Efficacy in Melanoma 期刊论文  OAI收割
CANCER RESEARCH, 2024, 卷号: 84, 期号: 3, 页码: 419-433
作者:  
Tao, Hongru;  Jin, Chen;  Zhou, Liyuan;  Deng, Zhenzhong;  Li, Xiao
  |  收藏  |  浏览/下载:16/0  |  提交时间:2024/04/09
Chemical Inhibitors Targeting the Oncogenic m6A Modifying Proteins 期刊论文  OAI收割
ACCOUNTS OF CHEMICAL RESEARCH, 2023, 卷号: 56, 期号: 21, 页码: 3010-3022
作者:  
Huang, Yue;  Xia, Wenyang;  Dong, Ze;  Yang, Cai-Guang
  |  收藏  |  浏览/下载:7/0  |  提交时间:2023/12/11
A patent review of PRMT5 inhibitors to treat cancer (2018-present) 期刊论文  OAI收割
EXPERT OPINION ON THERAPEUTIC PATENTS, 2023, 页码: 28
作者:  
Gao, Jing;  Yang, Jie;  Xue, Shengyu;  Ding, Hong;  Lin, Hua
  |  收藏  |  浏览/下载:12/0  |  提交时间:2023/10/17
PRMT6 promotes tumorigenicity and cisplatin response of lung cancer through triggering 6PGD/ENO1 mediated cell metabolism 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13, 期号: 1, 页码: 157-173
作者:  
Sun, Mingming;  Li, Leilei;  Niu, Yujia;  Wang, Yingzhi;  Yan, Qi
  |  收藏  |  浏览/下载:15/0  |  提交时间:2024/03/27
Design, synthesis, and biological evaluation of novel carbazole derivatives as potent DNMT1 inhibitors with reasonable PK properties 期刊论文  OAI收割
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2022, 卷号: 37, 期号: 1, 页码: 1537-1555
作者:  
Li, Ennian;  Wang, Kai;  Zhang, Bei;  Guo, Siqi;  Xiao, Senhao
  |  收藏  |  浏览/下载:37/0  |  提交时间:2022/08/16
Proteomic characterization of post-translational modifications in drug discovery 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2022, 页码: 18
作者:  
Zhai, Lin-hui;  Chen, Kai-feng;  Hao, Bing-bing;  Tan, Min-jia
  |  收藏  |  浏览/下载:13/0  |  提交时间:2023/04/10
Identification of PRMT5 inhibitors with novel scaffold structures through virtual screening and biological evaluations 期刊论文  OAI收割
JOURNAL OF MOLECULAR MODELING, 2022, 卷号: 28, 期号: 7, 页码: 184
作者:  
Zhang, Qian;  Zhang, Lun;  Jin, Jia;  Fan, Yaohua;  Wang, Xiaoguang
  |  收藏  |  浏览/下载:11/0  |  提交时间:2024/03/21