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Chinese Academy of Sciences Institutional Repositories Grid
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上海药物研究所 [21]
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A patent review of PRMT5 inhibitors to treat cancer (2018-present)
期刊论文
OAI收割
EXPERT OPINION ON THERAPEUTIC PATENTS, 2023, 页码: 28
作者:
Gao, Jing
;
Yang, Jie
;
Xue, Shengyu
;
Ding, Hong
;
Lin, Hua
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2023/10/17
PRMT5
inhibitor
epigenetic target
cancer treatment
combined treatment
PRMT5 promotes ovarian cancer growth through enhancing Warburg effect by methylating ENO1
期刊论文
OAI收割
MedComm, 2023, 卷号: 4, 期号: 2, 页码: e245
作者:
Xie, Fei
;
Zhang, Han
;
Zhu, Kongkai
;
Jiang, Cheng-Shi
;
Zhang, Xiaoya
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/03/26
Structure-activity relationship study of a series of nucleoside derivatives bearing sulfonamide scaffold as potent and selective PRMT5 inhibitors
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2023, 卷号: 130, 页码: 20
作者:
Chen, Yuting
;
Shi, Qiongyu
;
Yang, Hong
;
Li, Jiayi
;
Zhou, Kaixin
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2023/04/10
Epigenetic
PRMT5 inhibitor
Nucleoside derivatives
Structure-activity Relationship Prodrug
Identification of PRMT5 inhibitors with novel scaffold structures through virtual screening and biological evaluations
期刊论文
OAI收割
JOURNAL OF MOLECULAR MODELING, 2022, 卷号: 28, 期号: 7, 页码: 184
作者:
Zhang, Qian
;
Zhang, Lun
;
Jin, Jia
;
Fan, Yaohua
;
Wang, Xiaoguang
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2024/03/21
PRMT5
Small-molecule inhibitors
Virtual screening
Molecular docking
Molecular dynamics simulations
Structure-Aided Design, Synthesis, and Biological Evaluation of Potent and Selective Non-Nucleoside Inhibitors Targeting Protein Arginine Methyltransferase 5
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 11, 页码: 7854-7875
作者:
Rong, Deqin
;
Zhou, Kaixin
;
Fang, Wei
;
Yang, Hong
;
Zhang, Yi
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2022/08/16
Myelocytomatosis-Protein Arginine N-Methyltransferase 5 Axis Defines the Tumorigenesis and Immune Response in Hepatocellular Carcinoma
期刊论文
OAI收割
HEPATOLOGY, 2021, 卷号: 74, 期号: 4, 页码: 1932-1951
作者:
Luo, Yuhong
;
Gao, Yuqing
;
Liu, Weiwei
;
Yang, Yuan
;
Jiang, Jie
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/03/21
Allosteric Modulation: Dynamics is Double-"E"dged
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 7, 页码: 3694-3696
作者:
Xiong, Bing
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2021/06/11
PRMT5 Is Involved in Spermatogonial Stem Cells Maintenance by Regulating Plzf Expression via Modulation of Lysine Histone Modifications
期刊论文
OAI收割
FRONTIERS IN CELL AND DEVELOPMENTAL BIOLOGY, 2021, 卷号: 9
作者:
Dong
;
Fangfang
;
Chen
;
Min
;
Chen
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2023/04/17
PRMT5 regulates ovarian follicle development by facilitating Wt1 translation
期刊论文
OAI收割
ELIFE, 2021, 卷号: 10
作者:
Chen Min
;
Dong Fangfang
;
Chen Min
;
Shen Zhiming
;
Wu Haowei
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2023/04/17
The cross-talk between methylation and phosphorylation in lymphoid-specific helicase drives cancer stem-like properties
期刊论文
OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2020, 卷号: 5, 期号: 1, 页码: 14
作者:
Liu, Na
;
Yang, Rui
;
Shi, Ying
;
Chen, Ling
;
Liu, Yating
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2020/12/21