中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共182条,第1-10条 帮助

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Discovery of novel antimyeloma agents targeting TRIP13 by molecular modeling and bioassay 期刊论文  OAI收割
RSC MEDICINAL CHEMISTRY, 2025, 页码: 14
作者:  
Bunu, Samuel Jacob;  Cai, Haiyan;  Zhou, Zhaoyin;  Zhang, Yanlei;  Lai, Yue
  |  收藏  |  浏览/下载:7/0  |  提交时间:2025/06/23
Dynamically chiral phosphonic acid-type metallo-β-lactamase inhibitors 期刊论文  OAI收割
COMMUNICATIONS CHEMISTRY, 2025, 卷号: 8, 期号: 1, 页码: 13
作者:  
Gulyas, Kinga Virag;  Zhou, Liping;  Salamonsen, Daniel;  Prester, Andreas;  Bartels, Kim
  |  收藏  |  浏览/下载:8/0  |  提交时间:2025/06/23
REG3A secreted by peritumoral acinar cells enhances pancreatic ductal adenocarcinoma progression via activation of EGFR signaling 期刊论文  OAI收割
CELL COMMUNICATION AND SIGNALING, 2025, 卷号: 23, 期号: 1, 页码: 19
作者:  
Ren, Xiaojing;  Teng, Yunfei;  Xie, Kunxin;  He, Xiao;  Chen, Gang
  |  收藏  |  浏览/下载:31/0  |  提交时间:2025/04/01
Discovery of peptidomimetic spiropyrrolidine derivatives as novel 3CLpro inhibitors against SARS-CoV-2 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 281, 页码: 22
作者:  
Guma, Samuel Desta;  Zhou, Zhaoyin;  Song, Kang;  Yang, Feipu;  Suo, Jin
  |  收藏  |  浏览/下载:19/0  |  提交时间:2024/12/11
F-CPI: A Multimodal Deep Learning Approach for Predicting Compound Bioactivity Changes Induced by Fluorine Substitution 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 13
作者:  
Zhang, Qian;  Yin, Wenhai;  Chen, Xinyao;  Zhou, Aimin;  Zhang, Guixu
  |  收藏  |  浏览/下载:23/0  |  提交时间:2025/02/28
Identification of USP2 as a novel target to induce degradation of KRAS in myeloma cells 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2024, 卷号: 14, 期号: 12, 页码: 5235-5248
作者:  
Wang, Yingying;  Zhang, Youping;  Luo, Hao;  Wei, Wei;  Liu, Wanting
  |  收藏  |  浏览/下载:24/0  |  提交时间:2025/04/01
Slow Metabolism-Driven Amplification of Hepatic PPARγ Agonism Mediates Benzbromarone-Induced Obesity-Specific Liver Injury 期刊论文  OAI收割
ADVANCED SCIENCE, 2024, 页码: 14
作者:  
Li, Guanting;  Hu, Yourong;  Zhao, Han;  Peng, Ziyu;  Shang, Xin
  |  收藏  |  浏览/下载:26/0  |  提交时间:2025/01/06
TRIP13-a potential drug target in cancer pharmacotherapy 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 151, 页码: 11
作者:  
Bunu, Samuel Jacob;  Cai, Haiyan;  Wu, Leyun;  Zhang, Hui;  Zhou, Zhaoyin
  |  收藏  |  浏览/下载:18/0  |  提交时间:2024/09/26
Development of ketalized unsaturated saccharides as multifunctional cysteine-targeting covalent warheads 期刊论文  OAI收割
COMMUNICATIONS CHEMISTRY, 2024, 卷号: 7, 期号: 1, 页码: 10
作者:  
Dong, Sanfeng;  Huang, Hui;  Li, Jintian;  Li, Xiaomei;  Bunu, Samuel Jacob
  |  收藏  |  浏览/下载:21/0  |  提交时间:2024/10/21
Synthesis and biological evaluation of multimodal monoaminergic arylpiperazine derivatives with potential antidepressant profile 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 275, 页码: 16
作者:  
Zheng, Jiefang;  Zhou, Liping;  Gong, Xudong;  Yang, Feipu;  Cheng, Jiaxin
  |  收藏  |  浏览/下载:19/0  |  提交时间:2024/08/22