中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [21]
新疆理化技术研究所 [1]
中国科学院大学 [1]
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OAI收割 [22]
iSwitch采集 [1]
内容类型
期刊论文 [23]
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2023 [5]
2022 [1]
2021 [3]
2020 [2]
2019 [3]
2018 [2]
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Glimepiride, a novel soluble epoxide hydrolase inhibitor, protects against heart failure via increasing epoxyeicosatrienoic acids
期刊论文
OAI收割
JOURNAL OF MOLECULAR AND CELLULAR CARDIOLOGY, 2023, 卷号: 185, 页码: 13-25
作者:
Zhao, Chengcheng
;
Jiang, Xiangrui
;
Peng, Liyuan
;
Zhang, Yan
;
Li, Huihui
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2024/01/16
Heart failure
Hypertrophy
Epoxyeicosatrienoic acids
Soluble epoxide hydrolase
An efficient synthesis of the last step key intermediate for telmisartan via Pd-catalyzed carbonylative cyclization
期刊论文
OAI收割
TETRAHEDRON, 2023, 卷号: 148, 页码: 8
作者:
Odilov, Abdullajon
;
Qin, Hongjian
;
Bonku, Emmanuel Mintah
;
Zhu, Fuqiang
;
Yang, Feipu
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2023/12/19
Telmisartan
Benzimidazole
Pd-catalyzed
Carbonylative/cyclization
Structure-based development and preclinical evaluation of the SARS-CoV-2 3C-like protease inhibitor simnotrelvir
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 15
作者:
Jiang, Xiangrui
;
Su, Haixia
;
Shang, Weijuan
;
Zhou, Feng
;
Zhang, Yan
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2024/03/25
Efficient Large-Scale Process for Tecovirimat via Reactive Distillation for the Preparation of Cycloheptatriene
期刊论文
OAI收割
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2023, 页码: 8
作者:
Bonku, Emmanuel Mintah
;
Qin, Hongjian
;
Odilov, Abdullajon
;
Yang, Feipu
;
Xing, Xinglong
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2023/12/08
tecovirimat
monkeypox
cycloheptatriene
antiviral drug
reactive distillation
Pharmacokinetics,mass balance,and metabolism of 14C TPN171,a novel PDE5 inhibitor,in humans for the treatment of pulmonary arterial hypertension
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 卷号: 44, 期号: 1, 页码: 221
作者:
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2023/05/22
TPN171
14CTPN171
PDE5 inhibitor
pulmonary arterial hypertension
healthy volunteers
pharmacokinetics
metabolite identification
mass balance
An Efficient and Scalable Synthesis of Hydroxyglimepiride and Carboxyl Glimepiride: Main Metabolites of Glimepiride
期刊论文
OAI收割
INDIAN JOURNAL OF HETEROCYCLIC CHEMISTRY, 2022, 卷号: 32, 期号: 4, 页码: 417-421
作者:
Khakimov, Makhmudjon
;
Jiang, Xiangrui
;
Yang, Feipu
;
Shen, Jingshan
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2023/04/10
Facile and Cost-Effective Route for the Synthesis of Simmerafil
期刊论文
OAI收割
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2021, 卷号: 25, 期号: 11, 页码: 2432-2437
作者:
Odilov, Abdullajon
;
Liu, Yin
;
Hu, Tianwen
;
Jiang, Xiangrui
;
Suo, Jin
  |  
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2022/01/18
simmerafil
PDE5 inhibitor
salicylamide
synthesis
TPN672: A Novel Serotonin-Dopamine Receptor Modulator for the Treatment of Schizophrenia
期刊论文
OAI收割
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2021, 卷号: 378, 期号: 1, 页码: 20-30
作者:
Wang, Yu
;
He, Yang
;
Yang, Feipu
;
Abame, Melkamu Alemu
;
Wu, Chunhui
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2021/11/04
SARS-CoV-2 envelope protein causes acute respiratory distress syndrome (ARDS)-like pathological damages and constitutes an antiviral target
期刊论文
OAI收割
CELL RESEARCH, 2021, 页码: 14
作者:
Xia, Bingqing
;
Shen, Xurui
;
He, Yang
;
Pan, Xiaoyan
;
Liu, Feng-Liang
  |  
收藏
  |  
浏览/下载:74/0
  |  
提交时间:2021/08/17
Automated design and optimization of multitarget schizophrenia drug candidates by deep learning
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 204, 页码: 16
作者:
Tan, Xiaoqin
;
Jiang, Xiangrui
;
He, Yang
;
Zhong, Feisheng
;
Li, Xutong
  |  
收藏
  |  
浏览/下载:52/0
  |  
提交时间:2020/12/21
Schizophrenia
Multitarget antipsychotic drugs
Recurrent neural network
Multitask deep neural network
Automated drug design