中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [14]
兰州化学物理研究所 [9]
地理科学与资源研究所 [7]
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植物研究所 [5]
南京地理与湖泊研究所 [4]
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OAI收割 [62]
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期刊论文 [58]
专利 [2]
会议论文 [1]
学位论文 [1]
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2025 [1]
2024 [4]
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2020 [9]
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Development of Orally Bioavailable Octahydroindole-Based Peptidomimetic Derivative as a Broad-Spectrum Inhibitor against HCoV-OC43 and SARS-CoV-2
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 11, 页码: 10823-10844
作者:
Hu, Shulei
;
Zhang, Yumin
;
Wang, Chenchen
;
Li, Jian
;
Su, Haixia
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2025/07/25
Discovery of Novel Nonpeptidic and Noncovalent Small Molecule 3CL
pro
Inhibitors as anti-SARS-CoV-2 Drug Candidate
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 15, 页码: 12760-12783
作者:
Jiang, Zhidong
;
Feng, Bo
;
Chen, Lu
;
Nie, Tianqing
;
Chen, Shizhao
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2024/09/26
Integrating a Physical Model with Multi-Objective Optimization for the Design of Optical Angle Nano-Positioning Mechanism
期刊论文
OAI收割
APPLIED SCIENCES-BASEL, 2024, 卷号: 14, 期号: 9
作者:
Jiang, Bo
;
Dong, Yiming
;
Zhang, Zijie
;
Li, Xiangyu
;
Wei, Yuxuan
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2024/08/22
nano-positioning mechanisms
synchrotron radiation facility
multi-objective optimization
Mapping the potential distribution of Asian elephants: Implications for conservation and human-elephant conflict mitigation in South and Southeast Asia
期刊论文
OAI收割
ECOLOGICAL INFORMATICS, 2024, 卷号: 80, 页码: 102518
作者:
Xu, Haixia
;
Jiang, Luguang
;
Liu, Ye
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2024/09/19
Asian elephant
Maximum entropy
Environmental features
Population characteristics
Assessing the Accuracy and Consistency of Cropland Products in the Middle Yangtze Plain
期刊论文
OAI收割
LAND, 2024, 卷号: 13, 期号: 3, 页码: 14
作者:
Xu, Haixia
;
Jiang, Luguang
;
Liu, Ye
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2024/05/06
cropland distribution
Middle Yangtze Plain
GLAD (Global Land Analysis & Discovery)
AGLC (Annual Global Land Cover)
CLCD (China Land Cover Dataset)
CACD (China's Annual Cropland Dataset)
Structure-based development and preclinical evaluation of the SARS-CoV-2 3C-like protease inhibitor simnotrelvir
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 15
作者:
Jiang, Xiangrui
;
Su, Haixia
;
Shang, Weijuan
;
Zhou, Feng
;
Zhang, Yan
  |  
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2024/03/25
Design, synthesis and biological evaluation of peptidomimetic benzothiazolyl ketones as 3CLpro inhibitors against SARS-CoV-2
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 257, 页码: 13
作者:
Yang, Hanxi
;
You, Mengyuan
;
Shu, Xiaoyang
;
Zhen, Jingyao
;
Zhu, Mengwei
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2023/10/17
Peptidomimetics
Benzothiazolyl ketone
3CLpro inhibitor
Pharmacokinetic properties
SARS-CoV-2
Discovery of novel non-peptidic and non-covalent small-molecule 3CL(pro) inhibitors as potential candidate for COVID-19 treatment
期刊论文
OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2023, 卷号: 8, 期号: 1, 页码: 4
作者:
Jiang, Zhidong
;
Feng, Bo
;
Zhang, Yumin
;
Nie, Tianqing
;
Liu, Hong
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2023/10/17
一种腐蚀磨损实验装置
专利
OAI收割
专利号: ZL 202320110565X, 申请日期: 2023-05-12,
作者:
王鹏
;
马鹏翔
;
江海霞
;
柴利强
;
张贝贝
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/12/22
Design, synthesis and biological evaluation of covalent peptidomimetic 3CL protease inhibitors containing nitrile moiety
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2023, 卷号: 87, 页码: 12
作者:
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2023/10/17
COVID-19
SARS-CoV-2
3CL protease
Nirmatrelvir
Peptidomimetic inhibitors