中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [80]
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期刊论文 [196]
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Diterpenoids and diarylheptanoids from the fruits of
Alpinia
zerumbet
and their anti-inflammatory activity
期刊论文
OAI收割
FITOTERAPIA, 2025, 卷号: 184, 页码: 10
作者:
Zhang, Zhenghan
;
Li, Guangqian
;
Luo, Xin
;
Xiao, Fang
;
Zhang, Yan
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/08/20
Alpinia zerumbet
Labdane-type diterpenoid
Diarylheptanoid
Anti-inflammatory
ISG pathway
TDDFT ECD calculation
Structure-activity relationship analysis of meta-substituted N-cyclopropylmethyl-nornepenthones with mixed KOR/MOR activities
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 289, 页码: 15
作者:
Tang, Siyuan
;
Hu, Shuyang
;
Feng, Lijing
;
Kong, Linghui
;
Gui, Jiangwen
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2025/05/27
N-Cyclopropylmethyl-nornepenthones
Structure-activity relationship
MOR antagonist
KOR agonist
Substance use disorder
Direct Preparation of Site-Specific Antibody-Drug Conjugates with Unpurified Antibodies in Culture Medium
期刊论文
OAI收割
CHEMBIOCHEM, 2025, 页码: 7
作者:
Lu, Mengru
;
Zeng, Yue
;
Hang, Jiaying
;
Shi, Wei
;
Huang, Wei
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2025/05/27
cellular expression systems
K248 site-specific ADCs
one-pot
Macrophage SUCLA2 coupled glutaminolysis manipulates obesity through AMPK
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2025, 卷号: 16, 期号: 1, 页码: 20
作者:
Peng, Chang
;
Jiang, Haowen
;
Jing, Liya
;
Yang, Wenhua
;
Guan, Xiaotong
  |  
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2025/04/01
Discovery of novel biaryl urea derivatives against IL-1/3 release with low toxicity based on NEK7 inhibitor
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 283, 页码: 12
作者:
Wang, Leibo
;
Zhu, Kehan
;
Tian, Ziyang
;
Wang, Haoyu
;
Jia, Yulei
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2025/01/14
NLRP3 inflammasome
NEK7
NLRP3-NEK7
Inhibitors
Unveiling the binary nature of NGC 2323
期刊论文
OAI收割
ASTRONOMY & ASTROPHYSICS, 2025, 卷号: 693, 页码: A317
作者:
Qin, Songmei
;
Zhong, Jing
;
Tang, Tong
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2025/02/27
open clusters and associations: general
open clusters and associations: individual: NGC 2323
Harnessing acylhydrazone-oxime exchange reaction to achieve diverse synthesis of glycosite-specific antibody-drug conjugates
期刊论文
OAI收割
ORGANIC & BIOMOLECULAR CHEMISTRY, 2024, 页码: 9
作者:
Xia, Fei
;
Liu, Zhi
;
Hang, Jiaying
;
Xu, Hao
;
Xiao, Yuting
  |  
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2025/04/01
Synthesis and evaluation of hybrid molecules as RIPK1 and HDACs dual inhibitors
期刊论文
OAI收割
JOURNAL OF MOLECULAR STRUCTURE, 2024, 卷号: 1318, 页码: 13
作者:
Tang, Mingze
;
Zhou, Xuan
;
Shen, Qianqian
;
Fang, Chen
;
Peng, Xia
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2024/08/22
Receptor -interacting protein kinase 1
Histone deacetylases
Inhibitor
Molecular dynamics (MD) simulation
ADMET analysis
Design and development of a series of 4-(piperazin-1-yl)pyrimidines as irreversible menin inhibitors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 280, 页码: 20
作者:
Luo, Menglan
;
Ye, Yunfei
;
Tang, Lu
;
Kan, Weijuan
;
Chen, Lin
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2024/11/26
Menin
Covalent inhibitor
Antitumor
Degradation
Germacrane-type sesquiterpenes from Artemisia atrovirens and their anti-inflammatory activity
期刊论文
OAI收割
FITOTERAPIA, 2024, 卷号: 179, 页码: 11
作者:
Tang, Chunping
;
Zheng, Yongzhe
;
Shao, Zhengguang
;
Ke, Chang-Qiang
;
Feng, Zheling
  |  
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2024/11/26
Artemisia atrovirens
Atrovirenolides C -I
Atrovirenoic acid G
Diatrovirenolides A -B
DFT NMR calculation
TDDFT ECD calculation