中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [43]
新疆理化技术研究所 [4]
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OAI收割 [57]
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期刊论文 [57]
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F-CPI: A Multimodal Deep Learning Approach for Predicting Compound Bioactivity Changes Induced by Fluorine Substitution
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 13
作者:
Zhang, Qian
;
Yin, Wenhai
;
Chen, Xinyao
;
Zhou, Aimin
;
Zhang, Guixu
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2025/02/28
Discovery of the potent covalent inhibitor with an acrylate warhead for SARS-CoV-2 3CL protease
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 112, 页码: 5
作者:
Shen, Wen
;
Chen, Xinyao
;
Zhou, Liping
;
Cheng, Yan
;
Zhang, Yan
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2024/10/21
COVID-19
SARS-CoV-2 3CL pro inhibitor
Drug design
Antiviral activities
Identification of Dihydrobenzofuran Neolignans as Novel PDE4 Inhibitors and Evaluation of Antiatopic Dermatitis Efficacy in DNCB-Induced Mice Model
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 6, 页码: 4855-4869
作者:
Gu, Chenming
;
Liu, Jiayuan
;
Qian, Fei
;
Yu, Wenchao
;
Huang, Doudou
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/05/07
Cannabidiol exhibits anxiolytic-like effects and antipsychotic-like effects in mice models
期刊论文
OAI收割
NEUROSCIENCE LETTERS, 2024, 卷号: 826, 页码: 8
作者:
Shu, Guangzhao
;
He, Yang
;
Suo, Jin
;
Wu, Chunhui
;
Gong, Xudong
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2024/06/27
Cannabidiol
Stress-induced hyperthermia
Phencyclidine-induced negative symptoms of
schizophrenia model
5-HT 1A receptor
Oral Simnotrelvir for Adult Patients with Mild-to-Moderate Covid-19
期刊论文
OAI收割
NEW ENGLAND JOURNAL OF MEDICINE, 2024, 卷号: 390, 期号: 3, 页码: 230-241
作者:
Cao, Bin
;
Wang, Yeming
;
Lu, Hongzhou
;
Huang, Chaolin
;
Yang, Yumei
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2024/05/07
Glimepiride, a novel soluble epoxide hydrolase inhibitor, protects against heart failure via increasing epoxyeicosatrienoic acids
期刊论文
OAI收割
JOURNAL OF MOLECULAR AND CELLULAR CARDIOLOGY, 2023, 卷号: 185, 页码: 13-25
作者:
Zhao, Chengcheng
;
Jiang, Xiangrui
;
Peng, Liyuan
;
Zhang, Yan
;
Li, Huihui
  |  
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2024/01/16
Heart failure
Hypertrophy
Epoxyeicosatrienoic acids
Soluble epoxide hydrolase
Discovery and Timing of Millisecond Pulsars in the Globular Cluster M5 with FAST and Arecibo
期刊论文
OAI收割
ASTROPHYSICAL JOURNAL SUPPLEMENT SERIES, 2023, 卷号: 269, 期号: 2
作者:
Zhang, Lei
;
Freire, Paulo C. C.
;
Ridolfi, Alessandro
;
Pan, Zhichen
;
Zhao, Jiaqi
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2024/03/29
Structure-based development and preclinical evaluation of the SARS-CoV-2 3C-like protease inhibitor simnotrelvir
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 15
作者:
Jiang, Xiangrui
;
Su, Haixia
;
Shang, Weijuan
;
Zhou, Feng
;
Zhang, Yan
  |  
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2024/03/25
Design, synthesis and biological evaluation of covalent peptidomimetic 3CL protease inhibitors containing nitrile moiety
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2023, 卷号: 87, 页码: 12
作者:
Zhu, Mengwei
;
Fu, Tiantian
;
You, Mengyuan
;
Cao, Junyuan
;
Yang, Hanxi
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2023/10/17
COVID-19
SARS-CoV-2
3CL protease
Nirmatrelvir
Peptidomimetic inhibitors
Lift of a bio-inspired flapping wing with a dynamic trailing-edge flap in forward flight
期刊论文
OAI收割
PHYSICS OF FLUIDS, 2023, 卷号: 35, 期号: 4, 页码: 41709
作者:
Chen YX(陈一鑫)
;
Wang CY(王春雨)
;
Zhao, Jingshan
;
Wang SZ(王士召)
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2023/07/17