中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [60]
中国科学院大学 [1]
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期刊论文 [61]
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2026 [1]
2025 [14]
2024 [16]
2023 [7]
2022 [7]
2021 [4]
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Benchmarking
In Silico
Metabolite Prediction Tools against Human Radiolabeled ADME Data for Small-Molecule Drugs
期刊论文
OAI收割
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2026, 卷号: 66, 期号: 5, 页码: 2918-2928
作者:
Gao, Lei
;
Yan, Shu
;
Feng, Kaiyuan
;
Liu, Haonan
;
Zhang, Zihao
  |  
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Pharmacokinetics, mass balance, and metabolism of [
14
C]PLB1004, a selective and irreversible EGFR-TKI in humans
期刊论文
OAI收割
CANCER CHEMOTHERAPY AND PHARMACOLOGY, 2025, 卷号: 95, 期号: 1, 页码: 14
作者:
Liu, Donghui
;
Li, Qian
;
Yan, Shu
;
Zhang, Xinyue
;
Li, Weiqiang
  |  
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  |  
Pharmacokinetics, mass balance, and metabolism of [
14
C]FCN-437c, a selective and potent CDK4/6 inhibitor in humans
期刊论文
OAI收割
CANCER CHEMOTHERAPY AND PHARMACOLOGY, 2025, 卷号: 95, 期号: 1, 页码: 12
作者:
Gao, Lei
;
Ma, Sheng
;
Yan, Shu
;
Zhang, Hua
;
Tian, Ling
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  |  
Metabolism of the Total Flavonoid Extract of
Lithocarpus litseifolius
(Hance) Chun in Rats
期刊论文
OAI收割
BIOMEDICAL CHROMATOGRAPHY, 2025, 卷号: 39, 期号: 12, 页码: 10
作者:
Zhao, Yuqing
;
Yuan, Yali
;
Yan, Shu
;
Tang, Chongzhuang
  |  
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  |  
Pharmacokinetics, mass balance, and metabolism of [
14
C]SAF-189s, a potent anaplastic lymphoma kinase/c-ROS proto-oncogene 1 inhibitor in humans: Metabolism potentially affected by interaction of cytochrome P450 enzymes and intestinal microbiota
期刊论文
OAI收割
DRUG METABOLISM AND DISPOSITION, 2025, 卷号: 53, 期号: 9, 页码: 14
作者:
Yang, Ming
;
Diao, Lei
;
Yan, Shu
;
Tan, Yan
;
Liu, Donghui
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  |  
Development and Verification of a Physiologically Based Pharmacokinetic Model of Furmonertinib and Its Main Metabolite for Drug-Drug Interaction Predictions
期刊论文
OAI收割
CPT-PHARMACOMETRICS & SYSTEMS PHARMACOLOGY, 2025, 卷号: 14, 期号: 7, 页码: 1273-1284
作者:
Wu, Yali
;
Loer, Helena Leonie Hanae
;
Zhang, Yifan
;
Zhong, Dafang
;
Jiang, Yong
  |  
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  |  
Characterization of the specific proteins to which HH-A, a drug that alleviates ischemic brain injury, binds in rat plasma
期刊论文
OAI收割
DRUG METABOLISM AND DISPOSITION, 2025, 卷号: 53, 期号: 7, 页码: 15
作者:
Zhao, Jie
;
Zheng, Yuandong
;
Lei, Peng
;
Zhang, Yuying
;
Zhang, Pingping
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Absorption, distribution, metabolism, and excretion of [14C]SHEN211, a nonpeptidic small-molecule 3CLpro inhibitor, in rats
期刊论文
OAI收割
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2025, 卷号: 392, 期号: 7, 页码: 12
作者:
Zhang, Zihao
;
Jia, Mengting
;
Wang, Feiyu
;
Yang, Chen
;
Shi, Huanhuan
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Characterization of preclinical radio ADME properties of ARV-471 for predicting human PK using PBPK modeling
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL ANALYSIS, 2025, 卷号: 15, 期号: 5, 页码: 15
作者:
He, Yifei
;
Zhu, Chenggu
;
Lei, Peng
;
Yang, Chen
;
Zhang, Yifan
  |  
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  |  
Quantification of serum daratumumab in multiple myeloma patients by LC-MS/MS, comparison with ELISA
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2025, 卷号: 255, 页码: 7
作者:
Li, Weiqiang
;
Tian, Zhuoran
;
Yu, Xiong
;
Xu, Hongyu
;
Huang, Fang
  |  
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