中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共53条,第1-10条 帮助

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Discovery of 2-tetrahydroisoquinoline substituted quinazoline derivatives as lysine methyltransferase G9a inhibitors with in vivo antitumor efficacy 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 300, 页码: 15
作者:  
Shao, Mengjie;  Gao, Lixin;  Xu, Jiahui;  Zhu, Lingfeng;  Lu, Yiting
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A pan-KRAS inhibitor and its derived degrader elicit multifaceted anti-tumor efficacy in KRAS-driven cancers 期刊论文  OAI收割
CANCER CELL, 2025, 卷号: 43, 期号: 10, 页码: 32
作者:  
Feng, Juanjuan;  Xiao, Xuanzheng;  Xia, Xinting;  Min, Jian;  Tang, Weiying
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Discovery of Hydrazineyl Amide Derivative of Pseudolaric Acid B for Reprogramming Tumor-Associated Macrophages Against Tumor Growth 期刊论文  OAI收割
MOLECULES, 2025, 卷号: 30, 期号: 10, 页码: 22
作者:  
Peng, Xia;  Yu, Siqi;  Xu, Lin;  Wang, Qinghua;  Yang, Lin
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Design, Synthesis, and Pharmacological Evaluation of Quinazoline and Quinoline Derivatives as Potent ENPP1 Inhibitors for Cancer Immunotherapy 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 页码: 18
作者:  
He, Jie;  Ma, Xiaoyu;  Sun, Jia;  Chen, Manman;  Xu, Lan
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Discovery of Urea Derivatives of Celastrol as Selective Peroxiredoxin 1 Inhibitors against Colorectal Cancer Cells 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 9, 页码: 7176-7196
作者:  
Li, Yang;  Zhu, Yuyuan;  Shang, Fan-Fan;  Xu, Lin;  Jiang, Defang
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Design, Synthesis, and Pharmacological Evaluation of Spiro[carbazole-3,3′-pyrrolidine] Derivatives as cGAS Inhibitors for Treatment of Acute Lung Injury 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 24
作者:  
Chen, Mingjie;  Lei, Shuyue;  Zhou, Zihua;  Wang, Meng;  Feng, Chunlan
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Design, Synthesis, and Pharmacological Evaluation of Isoindoline Analogues as New HPK1 Inhibitors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 23, 页码: 16201-16221
作者:  
Xie, Chenghu;  Liu, Bo;  Song, Zilan;  Yang, Ye;  Dai, Mengdi
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Photochemically controlled activation of STING by CAIX-targeting photocaged agonists to suppress tumor cell growth 期刊论文  OAI收割
CHEMICAL SCIENCE, 2023, 卷号: 14, 期号: 22, 页码: 5956-5964
作者:  
Ding, Chunyong;  Du, Mengyan;  Xiong, Zhi;  Wang, Xue;  Li, Hongji
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Celastrol suppresses colorectal cancer via covalent targeting peroxiredoxin 1 期刊论文  OAI收割
Signal Transduction and Targeted Therapy, 2023, 卷号: 8, 期号: 3, 页码: 1159-1174
作者:  
Xu, Heng;  Zhao, Hongfang;  Ding, Chunyong;  Jiang, Defang;  Zhao, Zijie
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Acid-Ionizable Iron Nanoadjuvant Augments STING Activation for Personalized Vaccination Immunotherapy of Cancer 期刊论文  OAI收割
ADVANCED MATERIALS, 2023, 页码: 15
作者:  
Chen, Fangmin;  Li, Tianliang;  Zhang, Huijuan;  Saeed, Madiha;  Liu, Xiaoying
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