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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [52]
地质与地球物理研究所 [1]
采集方式
OAI收割 [53]
内容类型
期刊论文 [52]
会议论文 [1]
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2025 [4]
2024 [2]
2023 [4]
2022 [4]
2021 [3]
2020 [7]
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Discovery of 2-tetrahydroisoquinoline substituted quinazoline derivatives as lysine methyltransferase G9a inhibitors with in vivo antitumor efficacy
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 300, 页码: 15
作者:
Shao, Mengjie
;
Gao, Lixin
;
Xu, Jiahui
;
Zhu, Lingfeng
;
Lu, Yiting
  |  
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A pan-KRAS inhibitor and its derived degrader elicit multifaceted anti-tumor efficacy in
KRAS
-driven cancers
期刊论文
OAI收割
CANCER CELL, 2025, 卷号: 43, 期号: 10, 页码: 32
作者:
Feng, Juanjuan
;
Xiao, Xuanzheng
;
Xia, Xinting
;
Min, Jian
;
Tang, Weiying
  |  
收藏
  |  
Discovery of Hydrazineyl Amide Derivative of Pseudolaric Acid B for Reprogramming Tumor-Associated Macrophages Against Tumor Growth
期刊论文
OAI收割
MOLECULES, 2025, 卷号: 30, 期号: 10, 页码: 22
作者:
Peng, Xia
;
Yu, Siqi
;
Xu, Lin
;
Wang, Qinghua
;
Yang, Lin
  |  
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  |  
Design, Synthesis, and Pharmacological Evaluation of Quinazoline and Quinoline Derivatives as Potent ENPP1 Inhibitors for Cancer Immunotherapy
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 页码: 18
作者:
He, Jie
;
Ma, Xiaoyu
;
Sun, Jia
;
Chen, Manman
;
Xu, Lan
  |  
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  |  
Discovery of Urea Derivatives of Celastrol as Selective Peroxiredoxin 1 Inhibitors against Colorectal Cancer Cells
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 9, 页码: 7176-7196
作者:
Li, Yang
;
Zhu, Yuyuan
;
Shang, Fan-Fan
;
Xu, Lin
;
Jiang, Defang
  |  
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  |  
Design, Synthesis, and Pharmacological Evaluation of Spiro[carbazole-3,3′-pyrrolidine] Derivatives as cGAS Inhibitors for Treatment of Acute Lung Injury
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 24
作者:
Chen, Mingjie
;
Lei, Shuyue
;
Zhou, Zihua
;
Wang, Meng
;
Feng, Chunlan
  |  
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  |  
Design, Synthesis, and Pharmacological Evaluation of Isoindoline Analogues as New HPK1 Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 23, 页码: 16201-16221
作者:
Xie, Chenghu
;
Liu, Bo
;
Song, Zilan
;
Yang, Ye
;
Dai, Mengdi
  |  
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  |  
Photochemically controlled activation of STING by CAIX-targeting photocaged agonists to suppress tumor cell growth
期刊论文
OAI收割
CHEMICAL SCIENCE, 2023, 卷号: 14, 期号: 22, 页码: 5956-5964
作者:
Ding, Chunyong
;
Du, Mengyan
;
Xiong, Zhi
;
Wang, Xue
;
Li, Hongji
  |  
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  |  
Celastrol suppresses colorectal cancer via covalent targeting peroxiredoxin 1
期刊论文
OAI收割
Signal Transduction and Targeted Therapy, 2023, 卷号: 8, 期号: 3, 页码: 1159-1174
作者:
Xu, Heng
;
Zhao, Hongfang
;
Ding, Chunyong
;
Jiang, Defang
;
Zhao, Zijie
  |  
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  |  
Acid-Ionizable Iron Nanoadjuvant Augments STING Activation for Personalized Vaccination Immunotherapy of Cancer
期刊论文
OAI收割
ADVANCED MATERIALS, 2023, 页码: 15
作者:
Chen, Fangmin
;
Li, Tianliang
;
Zhang, Huijuan
;
Saeed, Madiha
;
Liu, Xiaoying
  |  
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