中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [57]
采集方式
OAI收割 [57]
内容类型
期刊论文 [57]
发表日期
2025 [1]
2024 [2]
2023 [6]
2022 [5]
2021 [11]
2020 [11]
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B(MIDA)-directed site-selective intermolecular halofluoroalkylation of alkenes: synthesis of diversely functionalized building blocks
期刊论文
OAI收割
CHEMICAL SCIENCE, 2025, 页码: 8
作者:
Wu, Hengbo
;
Luo, Ruitong
;
Peng, Jingjing
;
Han, Zijian
;
Zhang, Renjie
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2025/04/01
Discovery of Phenylpyrazole Derivatives as a New Class of Selective Inhibitors of MCL-1 with Antitumor Activity
期刊论文
OAI收割
ACS OMEGA, 2024, 页码: 28
作者:
Gong, Qineng
;
Li, Chunpu
;
Wang, Haojie
;
Cao, Jinrui
;
Li, Zuo
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2024/07/12
Discovery, Optimization, and Evaluation of Novel Pyridin-2(1
H
)-one Analogues as Potent TRK Inhibitors for Cancer Treatment
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 2, 页码: 1168-1183
作者:
Xu, Zichao
;
Peng, Xia
;
Zhang, Renjie
;
Ji, Yinchun
;
You, Mengke
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2024/02/27
Structure-based drug discovery of novel fused- pyrazolone carboxamide derivatives as potent and selective AXL inhibitors
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13, 期号: 12, 页码: 4918-4933
作者:
Fang, Feifei
;
Dai, Yang
;
Wang, Hao
;
Ji, Yinchun
;
Liang, Xuewu
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2024/01/26
derivatives
Antitumor drug development
Potential AXL inhibitor
Antitumor activity
Structure-based drug design
Fused-pyrazolone carboxamide
Constructing N-Acyl/N-Sulfonyl Aza-Sulfur Derivatives from Amides/Sulfonamides and Thiophthalimides via Oxidant Regulation
期刊论文
OAI收割
ORGANIC LETTERS, 2023, 卷号: 25, 期号: 32, 页码: 6018-6023
作者:
Li, Yazhou
;
Wang, Yongkun
;
Fang, Feifei
;
Zhang, Yu
;
Li, Chunpu
  |  
收藏
  |  
浏览/下载:50/0
  |  
提交时间:2023/10/17
Late-Stage Functionalization for the Divergent Synthesis of Podophyllotoxin Derivatives by Rhodium Catalysis
期刊论文
OAI收割
CHEMISTRY-A EUROPEAN JOURNAL, 2023, 页码: 10
作者:
Zhao, Yue
;
Shen, Yangpeng
;
He, Jian
;
Li, Jing
;
Zhou, Shengbin
  |  
收藏
  |  
浏览/下载:292/0
  |  
提交时间:2023/10/17
anticancer
C-H bond activation
divergent synthesis
podophyllotoxin
late-stage functionalization
Rapid Access to Polysubstituted Tetrahydrocarbazol-4-ones via Sequential Selective C-H Functionalization from N-Nitrosoanilines
期刊论文
OAI收割
CHINESE JOURNAL OF CHEMISTRY, 2023, 页码: 1957-1962
作者:
Li, Chan
;
Yang, Yanchen
;
Fang, Feifei
;
Liu, Chaoyi
;
Li, Chunpu
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2023/10/17
C-H activation
Cross dehydrogenative coupling
Rhodium catalysis
Iridium catalysis
Alkenylation
Amaidiation
Heteroarylation
Rh(III)-Catalyzed Synthesis of Substituted Isoindoles through a Direct C-H Activation/[4+1] Annulation and Acyl Migration Cascade of Oxadiazolones with Diazo Compounds
期刊论文
OAI收割
ORGANIC LETTERS, 2023, 页码: 5
作者:
Yang, Xiaohao
;
Ren, Hairu
;
Zhou, Shengbin
;
Li, Chunpu
;
Liu, Chaoyi
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2023/10/17
Structural Optimization of Fibroblast Growth Factor Receptor Inhibitors for Treating Solid Tumors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 5, 页码: 3226-3249
作者:
Li, Chunpu
;
Dai, Yang
;
Kong, Xiangtai
;
Wang, Bao
;
Peng, Xia
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2024/03/27
Synthesis of maleimide-braced peptide macrocycles and their potential anti-SARS-CoV-2 mechanisms
期刊论文
OAI收割
CHEMICAL COMMUNICATIONS, 2022, 页码: 4
作者:
Li, Jian
;
Sun, Jina
;
Zhang, Xianglei
;
Zhang, Ruxue
;
Wang, Qian
  |  
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2023/04/10