中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共328条,第1-10条 帮助

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Design, Synthesis, and Biological Evaluation of Pyrrolo[1,2-a]quinoxalin-4(5H)-one Derivatives as Potent and Orally Available Noncovalent Bruton's Tyrosine Kinase (BTK) Inhibitors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 8, 页码: 8841-8860
作者:  
Tian, Chaoquan;  Du, Husheng;  Sha, Wenjie;  Wu, Lingkang;  Yu, Zhixiao
  |  收藏  |  浏览/下载:10/0  |  提交时间:2025/05/27
IHCH9033, a novel class I HDAC inhibitor, synergizes with FLT3 inhibitor and rescues quizartinib resistance in FLT3-ITD AML via enhancing DNA damage response 期刊论文  OAI收割
EXPERIMENTAL HEMATOLOGY & ONCOLOGY, 2025, 卷号: 14, 期号: 1, 页码: 19
作者:  
Yao, Mingyue;  Yan, Wenzhong;  Wang, Yafang;  Zhao, Yu;  Xu, Xiaowei
  |  收藏  |  浏览/下载:23/0  |  提交时间:2025/04/01
Unraveling the CDK9/PP2A/ERK Network in Transcriptional Pause Release and Complement Activation in KRAS-mutant Cancers 期刊论文  OAI收割
ADVANCED SCIENCE, 2024, 页码: 20
作者:  
Wang, Yafang;  Xu, Lansong;  Ling, Lijun;  Yao, Mingyue
  |  收藏  |  浏览/下载:32/0  |  提交时间:2024/10/21
Highly accurate carbohydrate-binding site prediction with DeepGlycanSite 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2024, 卷号: 15, 期号: 1, 页码: 13
作者:  
He, Xinheng;  Zhao, Lifen
  |  收藏  |  浏览/下载:27/0  |  提交时间:2024/08/20
Computing the relative binding affinity of ligands based on a pairwise binding comparison network 期刊论文  OAI收割
Nature computational science, 2023, 卷号: 3, 期号: 10, 页码: 860-872
作者:  
Yu, Jie;  Li, Zhaojun;  Chen, Geng;  Kong, Xiangtai;  Hu, Jie
  |  收藏  |  浏览/下载:36/0  |  提交时间:2024/03/26
Structure-based development and preclinical evaluation of the SARS-CoV-2 3C-like protease inhibitor simnotrelvir 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 15
作者:  
Jiang, Xiangrui;  Su, Haixia;  Shang, Weijuan;  Zhou, Feng;  Zhang, Yan
  |  收藏  |  浏览/下载:51/0  |  提交时间:2024/03/25
Loops Mediate Agonist-Induced Activation of the Stimulator of Interferon Genes Protein 期刊论文  OAI收割
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2023, 页码: 9
作者:  
Li, Rui;  Chen, Lin;  He, Xinheng;  Cao, Duanhua;  Zhang, Zehong
  |  收藏  |  浏览/下载:32/0  |  提交时间:2023/12/11
αExtractor: a system for automatic extraction of chemical information from biomedical literature 期刊论文  OAI收割
SCIENCE CHINA-LIFE SCIENCES, 2023, 页码: 4
作者:  
Xiong, Jiacheng;  Liu, Xiaohong;  Li, Zhaojun;  Xiao, Hongzhong;  Wang, Guangchao
  |  收藏  |  浏览/下载:48/0  |  提交时间:2023/12/08
STING agonist-boosted mRNA immunization via intelligent design of nanovaccines for enhancing cancer immunotherapy 期刊论文  OAI收割
NATIONAL SCIENCE REVIEW, 2023, 卷号: 10, 期号: 10, 页码: 16
作者:  
Zhou, Lei;  Yi, Wenzhe;  Zhang, Zehong;  Shan, Xiaoting;  Zhao, Zitong
  |  收藏  |  浏览/下载:34/0  |  提交时间:2023/10/17
Spermine is a natural suppressor of AR signaling in castration-resistant prostate cancer 期刊论文  OAI收割
CELL REPORTS, 2023, 卷号: 42, 期号: 7, 页码: 24
作者:  
Li, Xiao;  Li, Fei;  Ye, Fei
  |  收藏  |  浏览/下载:44/0  |  提交时间:2023/10/17