中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [7]
化学研究所 [2]
力学研究所 [1]
采集方式
OAI收割 [10]
内容类型
期刊论文 [10]
发表日期
2024 [1]
2015 [1]
2013 [2]
2012 [2]
2011 [2]
2010 [1]
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Wintersweet-like Nanohybrids of Titanium-doped Cerium Vanadate Loaded with Polypyrrole for Tumor Theranostic
期刊论文
OAI收割
ADVANCED HEALTHCARE MATERIALS, 2024, 页码: 13
作者:
Lu, Qianyun
;
Wang, Xiaotong
;
Fan, Xin
;
Lin, Jinguo
;
Hu, Jiayi
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2024/07/08
cerium vanadate
chemodynamic therapy
polypyrrole
reactive oxygen species
theranostic
Fragment-Based Drug Discovery of 2-Thiazolidinones as BRD4 Inhibitors: 2. Structure-Based Optimization
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2015, 卷号: 58, 期号: 3, 页码: 1281-1297
作者:
Zhao, Lele
;
Wang, Yingqing
;
Cao, Danyan
;
Chen, Tiantian
;
Wang, Qi
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2019/01/08
Design, synthesis and SAR of piperidyl-oxadiazoles as 11 beta-hydroxysteroid dehydrogenase 1 inhibitors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 62, 页码: 1-10
作者:
Xia, Guangxin
;
You, Xiaodi
;
Liu, Lin
;
Liu, Haiyan
;
Wang, Jianfa
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2019/01/08
11 beta-HSD1 inhibitor
Oxadiazole
Bioisostere
SAR
Docking
Design and Synthesis of (R)-1-Arylsulfonylpiperidine-2-carboxamides as 11 beta-Hydroxysteroid Dehydrogenase Type 1 Inhibitors
期刊论文
OAI收割
CHEMMEDCHEM, 2013, 卷号: 8, 期号: 4, 页码: 577-581
作者:
Xia, Guangxin
;
Liu, Lin
;
Liu, Haiyan
;
Yu, Jianxin
;
Xu, Zhenmin
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2019/01/08
11-HSD1
diabetes
docking
inhibitors
Discovery of 2-Alkyl-1-arylsulfonylprolinamides as 11 beta-Hydroxysteroid Dehydrogenase Type 1 Inhibitors
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2012, 卷号: 3, 期号: 10, 页码: 793-798
作者:
Yu, Jianxin
;
Liu, Haiyan
;
Xia, Guangxin
;
Liu, Lin
;
Xu, Zhenmin
  |  
收藏
  |  
浏览/下载:148/0
  |  
提交时间:2019/01/08
metabolic syndrome
enzyme inhibitor
11 beta-hydroxysteroid dehydrogenase type 1
sulfonamide
2-alkylproline
prolinamide
Discovery of novel sulfonamides as potent and selective inhibitors against human and mouse 11 beta-hydroxysteroid dehydrogenase type 1
期刊论文
OAI收割
MOLECULAR AND CELLULAR ENDOCRINOLOGY, 2012, 卷号: 358, 期号: 1, 页码: 46-52
作者:
Xia, Guangxin
;
Liu, Lin
;
Xue, Mengzhu
;
Liu, Haiyan
;
Yu, Jianxin
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2019/01/08
11 beta-HSD1
Inhibitor
Sulfonamide
Diabetes
Docking
Potent and novel 11 beta-HSD1 inhibitors identified from shape and docking based virtual screening
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 卷号: 21, 期号: 19, 页码: 5739-5744
作者:
Xia, Guangxin
;
Xue, Mengzhu
;
Liu, Lin
;
Yu, Jianxin
;
Liu, Haiyan
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2019/01/08
11 beta-HSD1 inhibitor
Virtual screening
Docking
Shape similarity
Absolute Configurations and Stability of Cyclic Guanosine Mono-adducts with Glyoxal and Methylglyoxal
期刊论文
OAI收割
CHIRALITY, 2011, 卷号: 23, 期号: 7, 页码: 487-494
作者:
Lai, Congfang
;
Lin, Guangxin
;
Wang, Wenyue
;
Luo, Hai
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2019/04/09
Glyoxal/methylglyoxal
Guanosine Adduct
Circular Dichroism
Octant Rule
Diastereoisomer
Racemization
(S)-tert-Butyl 3-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine-1-carboxylate
期刊论文
OAI收割
ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE, 2010, 卷号: 66, 页码: O1576-U602
作者:
Liu, Lin
;
Xia, Guangxin
;
Liu, Xuejun
;
Xie, Jieshu
;
Shen, Jingkang
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2019/01/08
Desorption electrospray ionization
期刊论文
OAI收割
PROGRESS IN CHEMISTRY, 2008, 卷号: 20, 期号: 4, 页码: 594-601
作者:
Zhen, Xue
;
Bo, Qiu
;
Lin Guangxin
;
Lai Congfang
;
Hai, Luo
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2019/04/09
Desorption Electrospray Ionization (Desi)
Ambient Ionization
Ion Source
Surface Analysis
Detection Technique