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CAS IR Grid
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过程工程研究所 [23]
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期刊论文 [32]
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Potency Prediction of Covalent Inhibitors against SARS-CoV-2 3CL-like Protease and Multiple Mutants by Multiscale Simulations
期刊论文
OAI收割
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2024, 卷号: 64, 期号: 24, 页码: 9501-9516
作者:
Xiong, Muya
;
Nie, Tianqing
;
Li, Zhewen
;
Hu, Meiyi
;
Su, Haixia
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2025/01/06
Discovery of Novel Nonpeptidic and Noncovalent Small Molecule 3CL
pro
Inhibitors as anti-SARS-CoV-2 Drug Candidate
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 15, 页码: 12760-12783
作者:
Jiang, Zhidong
;
Feng, Bo
;
Chen, Lu
;
Nie, Tianqing
;
Chen, Shizhao
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2024/09/26
Design, synthesis and biological evaluation of betulinic acid derivatives as potential inhibitors of 3CL-protease of SARS-CoV-2
期刊论文
OAI收割
STEROIDS, 2024, 卷号: 202, 页码: 8
作者:
Liu, Yaowen
;
Nie, Tianqing
;
Hou, Jinjun
;
Long, Huali
;
Zhang, Zijia
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2024/03/13
3CLpro
SARS-CoV-2
Betulinic acid
Natural product
Inhibitory activity
Structure-based development and preclinical evaluation of the SARS-CoV-2 3C-like protease inhibitor simnotrelvir
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 15
作者:
Jiang, Xiangrui
;
Su, Haixia
;
Shang, Weijuan
;
Zhou, Feng
;
Zhang, Yan
  |  
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2024/03/25
Discovery and Mechanism Study of SARS-CoV-2 3C-like Protease Inhibitors with a New Reactive Group
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 18
作者:
Ren, Pengxuan
;
Li, Hui
;
Nie, Tianqing
;
Jian, Xiaoqin
;
Yu, Changyue
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2023/10/17
Discovery of novel non-peptidic and non-covalent small-molecule 3CL(pro) inhibitors as potential candidate for COVID-19 treatment
期刊论文
OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2023, 卷号: 8, 期号: 1, 页码: 4
作者:
Jiang, Zhidong
;
Feng, Bo
;
Zhang, Yumin
;
Nie, Tianqing
;
Liu, Hong
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2023/10/17
Discovery, synthesis and mechanism study of 2,3,5-substituted [1,2,4]-thiadiazoles as covalent inhibitors targeting 3C-Like protease of SARS-CoV-2
期刊论文
OAI收割
European journal of medicinal chemistry, 2023, 卷号: 249, 页码: 115129
作者:
Ren, Pengxuan
;
Yu, Changyue
;
Zhang, Ruxue
;
Nie, Tianqing
;
Hu, Qiaoyu
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2024/03/26
A 3D bioprinted decellularized extracellular matrix/gelatin/quaternized chitosan scaffold assembling with poly(ionic liquid)s for skin tissue engineering
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2022, 卷号: 220, 页码: 1253-1266
作者:
Xu, Jie
;
Fang, Huan
;
Su, Ya
;
Kang, Yue
;
Xu, Deli
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2023/02/24
Antibacterial
Hemostasis
Skin tissue engineering
Antibacterial
Hemostasis
Skin tissue engineering
Gelatin/sodium alginate hydrogel-coated decellularized porcine coronary to construct tissue blood vessels
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2022, 卷号: 209, 页码: 2070-2083
作者:
Du, Jing
;
Hu, Xueyan
;
Su, Ya
;
Wei, Tuo
;
Jiao, Zeren
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2023/02/24
Decellularized porcine coronary artery
Gelatin
sodium alginate
Bilayer scaffolds construct
Fibroblasts
Tissue engineered blood vessels
In silico screening-based discovery of novel covalent inhibitors of the SARS-CoV-2 3CL protease
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 231, 页码: 8
作者:
Xiong, Muya
;
Nie, Tianqing
;
Shao, Qiang
;
Li, Minjun
;
Su, Haixia
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2022/06/15
SARS-CoV-2 3C-Like protease
Covalent inhibitor
Virtual screening
Crystal structure