中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [7]
广州能源研究所 [1]
采集方式
OAI收割 [8]
内容类型
期刊论文 [8]
发表日期
2024 [3]
2022 [1]
2018 [1]
2016 [1]
2015 [1]
2010 [1]
更多
学科主题
energy & f... [1]
engineerin... [1]
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浏览/检索结果:
共8条,第1-8条
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Development of ketalized unsaturated saccharides as multifunctional cysteine-targeting covalent warheads
期刊论文
OAI收割
COMMUNICATIONS CHEMISTRY, 2024, 卷号: 7, 期号: 1, 页码: 10
作者:
Dong, Sanfeng
;
Huang, Hui
;
Li, Jintian
;
Li, Xiaomei
;
Bunu, Samuel Jacob
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/10/21
Discovery of Novel PROTAC Degraders of p300/CBP as Potential Therapeutics for Hepatocellular Carcinoma
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 4, 页码: 2466-2486
作者:
Chang, Qi
;
Li, Jiayi
;
Deng, Yue
;
Zhou, Ruilin
;
Wang, Bingwei
  |  
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2024/03/25
Design and synthesis of cantharidin derivative DCZ5418 as a TRIP13 inhibitor with anti-multiple myeloma activity
in
vitro
and
in
vivo
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 98, 页码: 7
作者:
Dong, Sanfeng
;
Hu, Ke
;
Shi, Yulong
;
Wang, Guanli
;
Yu, Dandan
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2024/02/19
Multiple myeloma
TRIP13 inhibitor
Cantharidin
DCZ5418
DCZ0415
Discovery of novel benzimidazole derivatives as potent p300 bromodomain inhibitors with anti-proliferative activity in multiple cancer cells
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2022, 卷号: 66, 页码: 16
作者:
Chen, Zonglong
;
Li, Jiayi
;
Yang, Hong
;
He, Yulong
;
Shi, Qiongyu
  |  
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2022/08/16
P300
Bromodomain inhibitors
CBP30
SBDD
Discovery of novel 2,4-diarylaminopyrimidine derivatives as potent and selective epidermal growth factor receptor (EGFR) inhibitors against L858R/T790M resistance mutation
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 152, 页码: 298-306
作者:
Yan, Qi
;
Chen, Yuzhe
;
Tang, Baiyou
;
Xiao, Qiang
;
Qu, Rong
  |  
收藏
  |  
浏览/下载:83/0
  |  
提交时间:2019/01/08
EGFR inhibitors
Pyrimidine derivatives
Mutant selective inhibitors
AZD9291
T790M
Discovery of 5-(methylthio)pyrimidine derivatives as L858R/T790M mutant selective epidermal growth factor receptor (EGFR) inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 12, 页码: 2673-2680
作者:
Xiao, Qiang
;
Qu, Rong
;
Gao, Dingding
;
Yan, Qi
;
Tong, Linjiang
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2019/01/08
5-(Methylthio)pyrimidine derivatives
Mutant selective inhibitors
Epidermal growth factor inhibitor
NSCLC
Structure-based drug design
Total Synthesis of Two Diastereomers of Megastigmane Glycoside Lauroside B
期刊论文
OAI收割
JOURNAL OF CARBOHYDRATE CHEMISTRY, 2015, 卷号: 34, 期号: 8, 页码: 445-459
作者:
Fu, Xiaozhe
;
Zhang, Mingming
;
Gao, Qi
;
Yang, Fengling
;
Li, Yingxia
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2019/01/08
Lauroside B
Megastigmane
Melanoma
NF-B
Diastereomers
Experimental study on a small scale of gas hydrate cold storage apparatus
期刊论文
OAI收割
applied energy, 2010, 卷号: 87, 期号: 11, 页码: 3340-3346
作者:
Xie, Yingming
;
Li, Gang
;
Liu, Daoping
;
Liu, Ni
;
Qi, Yingxia
收藏
  |  
浏览/下载:82/0
  |  
提交时间:2014/12/24
Gas hydrate
Cold storage
Heat exchanger
SDS
Hydration enhancement
Coolant