中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
合肥物质科学研究院 [6]
成都山地灾害与环境研... [1]
上海药物研究所 [1]
近代物理研究所 [1]
采集方式
OAI收割 [9]
内容类型
期刊论文 [9]
发表日期
2021 [2]
2018 [3]
2017 [3]
2016 [1]
学科主题
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Radioactivity control strategy for the JUNO detector
期刊论文
OAI收割
JOURNAL OF HIGH ENERGY PHYSICS, 2021, 期号: 11, 页码: 39
作者:
Abusleme, Angel
;
Adam, Thomas
;
Ahmad, Shakeel
;
Ahmed, Rizwan
;
Aiello, Sebastiano
  |  
收藏
  |  
浏览/下载:139/0
  |  
提交时间:2022/01/07
Neutrino Detectors and Telescopes (experiments)
Multiscale Co-reconstruction of Lung Architectures and Inhalable Materials Spatial Distribution
期刊论文
OAI收割
ADVANCED SCIENCE, 2021, 页码: 14
作者:
  |  
收藏
  |  
浏览/下载:55/0
  |  
提交时间:2021/05/24
dry powder inhalation
fluorescence‐
micro optical sectioning tomography
inhaled materials
pulmonary drug delivery
three‐
dimensional rendering
Discovery of (E)-N-(4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-((3-(2-(pyridin-2-yl)vinyl)-1H-indazol-6-yl)thio)propanamide (CHMFL-ABL-121) as a highly potent ABL kinase inhibitor capable of overcoming a variety of ABL mutants including T315I for chronic myeloid leukemia
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 160, 页码: 61-81
作者:
Liu, Xuesong
;
Wang, Beilei
;
Chen, Cheng
;
Jiang, Zongru
;
Hu, Chen
  |  
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2019/01/11
ABL kinase
Kinase inhibitor
ABL mutant
CML
Laboratory Investigation of the Effect of Nano-Silica on Unconfined Compressive Strength and Frost Heaving Characteristics of Silty Clay
期刊论文
OAI收割
SOIL MECHANICS AND FOUNDATION ENGINEERING, 2018, 卷号: 55, 期号: 5, 页码: 352-357
作者:
Hu, Kai
;
Chen, Xiaoqing
;
Chen, Jiangang
;
Ren, Xiaochuan
  |  
收藏
  |  
浏览/下载:59/0
  |  
提交时间:2019/01/21
nano-silica
Unconfined Compressive Strength
Frost Heaving Characteristics
Discovery of 4-((N-(2-(dimethylamino)ethyl)acrylamido)methyl)-N-(4-methyl-3-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)phenyl)benzamide (CHMFL-PDGFR-159) as a highly selective type II PDGFR alpha kinase inhibitor for PDGFR alpha driving chronic eosinophilic leukemia
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 150, 期号: 无, 页码: 366-384
作者:
Wang, Qiang
;
Liu, Feiyang
;
Qi, Shuang
;
Qi, Ziping
;
Yan, Xiao-E.
  |  
收藏
  |  
浏览/下载:75/0
  |  
提交时间:2019/06/10
PDGFR kinase
Type II inhibitor
Kinase inhibitor
CEL
Discovery of 1-(4-(4-Amino-3-(4-(2-morpholinoethoxy)-phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)phenyl)-3-(5-(tert-butyl)isoxazol-3-yl)urea (CHMFL-FLT3-213) as a Highly Potent Type II FLT3 Kinase Inhibitor Capable of Overcoming a Variety of FLT3 Kinase Mutants in FLT3-ITD Positive AML
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 20, 页码: 8407-8424
作者:
Wang, Aoli
;
Li, Xixiang
;
Chen, Cheng
;
Wu, Hong
;
Qi, Ziping
  |  
收藏
  |  
浏览/下载:54/0
  |  
提交时间:2019/06/17
Discovery of N-(3-(5-((3-acrylamido-4-(morpholine-4-carbonyl) phenyl)amino)-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl)-4-(tert-butyl)benzamide (CHMFL-BTK-01) as a highly selective irreversible Bruton's tyrosine kinase (BTK) inhibitor
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 131, 页码: 107-125
作者:
Liang, Qianmao
;
Chen, Yongfei
;
Yu, Kailin
;
Chen, Cheng
;
Zhang, Shouxiang
  |  
收藏
  |  
浏览/下载:43/0
  |  
提交时间:2018/07/26
Btk
Irreversible Inhibitor
Kinase Inhibitor
Structure-activity Relationship
B-cell Lymphoma
Discovery of 2-((3-Acrylamido-4-methylphenyl)amino)-N-(2-methyl5-(3,4,5-trimethoxybenzamido)phenyI)-4-(methylamino)pyrimidine-5-carboxamide (CHMFL-BMX-078) as a Highly Potent and Selective Type II Irreversible Bone Marrow Kinase in the X Chromosome (BMX) Kinase Inhibitor
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 5, 页码: 1793-1816
作者:
Liang, Xiaofei
;
Lv, Fengchao
;
Wang, Beilei
;
Yu, Kailin
;
Wu, Hong
  |  
收藏
  |  
浏览/下载:883/0
  |  
提交时间:2018/07/04
Discovery of N-((1-(4-(3-(3-((6,7-Dimethoxyquinolin-3-yl)oxy)phenyl)ureido)-2-(trifluoromethyl)phenyl)piperidin-4-yl)methyl)propionamide (CHMFL-KIT-8140) as a Highly Potent Type II Inhibitor Capable of Inhibiting the T670I "Gatekeeper" Mutant of cKIT Kinase
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 18, 页码: 8456-8472
作者:
Li, Binhua
;
Wang, Aoli
;
Liu, Juan
;
Qi, Ziping
;
Liu, Xiaochuan
收藏
  |  
浏览/下载:45/0
  |  
提交时间:2017/11/21