中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
高能物理研究所 [7]
上海药物研究所 [6]
地质与地球物理研究所 [3]
大连化学物理研究所 [2]
中国科学院大学 [2]
自动化研究所 [2]
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OAI收割 [16]
iSwitch采集 [9]
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期刊论文 [25]
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2024 [2]
2021 [1]
2019 [4]
2017 [3]
2016 [1]
2014 [3]
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学科主题
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Breaking boundaries in radiology: redefining AI diagnostics via raw data ahead of reconstruction
期刊论文
OAI收割
Physics in Medicine & Biology, 2024, 卷号: 69, 期号: 7
作者:
He,Bingxi
;
Sun,Caixia
;
Li,Hailin
;
Wang,Yongbo
;
She,Yunlang
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2024/05/30
deep learning
sinogram
CT scans
lung cancer
raw data
From Signal to Knowledge: The Diagnostic Value of Raw Data in the Artificial Intelligence Prediction of Human Data for the First Time
期刊论文
OAI收割
ENGINEERING, 2024, 卷号: 34, 页码: 60-69
作者:
He, Bingxi
;
Guo, Yu
;
Zhu, Yongbei
;
Tong, Lixia
;
Kong, Boyu
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2024/09/09
Computed tomography
Diagnosis
Deep learning
Lung cancer
Raw data
Discovery of a Pyrimidinedione Derivative as a Potent and Orally Bioavailable Axl Inhibitor
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 7, 页码: 3956-3975
作者:
Zhang, Hefeng
;
Peng, Xia
;
Dai, Yang
;
Shao, Jingwei
;
Ji, Yinchun
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2021/06/11
Rational Design, synthesis and biological evaluation of novel triazole derivatives as potent and selective PRMT5 inhibitors with antitumor activity
期刊论文
OAI收割
JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN, 2019, 卷号: 33, 期号: 8, 页码: 775-785
作者:
Zhu, Kongkai
;
Shao, Jingwei
;
Tao, Hongrui
;
Yan, Xue
;
Luo, Cheng
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2020/07/01
PRMT5 inhibitor
Anti-proliferative
Cellular target validation
Design and synthesis
Response of aggregate associated organic carbon, nitrogen and phosphorous to re-vegetation in agro-pastoral ecotone of northern China
期刊论文
OAI收割
GEODERMA, 2019, 期号: 341, 页码: 172-180
作者:
Yufei Yao
;
Nannan Ge
;
Si Yu
;
Xiaorong Wei
;
Xiang Wang
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2020/06/11
Discovery of 2-substituted-N-(3-(3,4-dihydroisoquinolin-2(1H)-yl)-2-hydroxypropyl)-1,2,3,4-tetrahydroisoquinoline-6-carboxamide as potent and selective protein arginine methyltransferases 5 inhibitors: Design, synthesis and biological evaluation
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 164, 页码: 317-333
作者:
Shao, Jingwei
;
Zhu, Kongkai
;
Du, Daohai
;
Zhang, Yuanyuan
;
Tao, Hongrui
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2020/07/01
PRMT5 inhibitors
N-Substituted 1,2,3,4-tetrahydroisoquinoline derivatives
Anti-tumor
Targeting PRMT5 Activity Inhibits the Malignancy of Hepatocellular Carcinoma by Promoting the Transcription of HNF4 alpha
期刊论文
OAI收割
THERANOSTICS, 2019, 卷号: 9, 期号: 9, 页码: 2606-2617
作者:
Zheng, Bai-Nan
;
Ding, Chen-Hong
;
Chen, Shi-Jie
;
Zhu, Kongkai
;
Shao, Jingwei
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2020/07/01
PRMT5
HNF4 alpha
hepatocellular carcinoma
cancer stem cells
Potent, Selective, and Cell Active Protein Arginine Methyltransferase 5 (PRMT5) Inhibitor Developed by Structure-Based Virtual Screening and Hit Optimization
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 14, 页码: 6289-6304
作者:
Mao, Ruifeng
;
Shao, Jingwei
;
Zhu, Kongkai
;
Zhang, Yuanyuan
;
Ding, Hong
  |  
收藏
  |  
浏览/下载:99/0
  |  
提交时间:2019/01/08
Excellent wear resistance of plasma-sprayed amorphous Al2O3–Y3Al5O12ceramic coating
期刊论文
OAI收割
Surface and Coatings Technology, 2017, 卷号: 326, 页码: 96-102
作者:
Yang, Kai
;
Rong, Jian
;
Feng, Jingwei
;
Zhuang, Yin
;
Zhao, Huayu
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2018/12/29
Microstructure formed by suspension plasma spraying: From YSZ splat to coating
期刊论文
OAI收割
Ceramics International, 2017, 卷号: 43, 期号: 10, 页码: 7488-7496
作者:
Li, Dachuan
;
Feng, Jingwei
;
Zhao, Huayu
;
Liu, Chenguang
;
Zhang, Linlin
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2018/12/29